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PLoS ONE, ISSN 1932-6203, 02/2013, Volume 8, Issue 2, p. e56132
Journal Article
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 10/2017, Volume 2017, Issue 39, pp. 5921 - 5934
Most known β2‐selective proteasome inhibitors suffer from relatively poor cell permeability as the result of a net positive charge caused by the basic moiety... 
Proteasomes | Amino acids | Inhibitors | Asymmetric synthesis | Peptidomimetics | Structure‐activity relationships | Structure-activity relationships | TRYPSIN-LIKE SITES | CHEMISTRY, ORGANIC | BORTEZOMIB | CARFILZOMIB | AMINO-ACIDS | SUBSTRATE | MYELOMA CELLS | Synthesis | Permeability | Hydrogen-ion concentration | Lysine | Organic compounds
Journal Article
Journal Article
Cancer Cell, ISSN 1535-6108, 12/2013, Volume 24, Issue 6, pp. 691 - 693
An elegant paper by Anchoori and colleagues in this issue of describes an irreversible inhibitor of Rpn13, one of the ubiquitin receptors on the 26S proteasome... 
ONCOLOGY | CANCER | CELL BIOLOGY | Animals | Membrane Glycoproteins - antagonists & inhibitors | Proteasome Inhibitors - pharmacology | Humans | Female | Piperidones - pharmacology | Neoplasms - drug therapy | Ubiquitin | Enzyme inhibitors
Journal Article
Current Opinion in Chemical Biology, ISSN 1367-5931, 12/2014, Volume 23, pp. 16 - 22
Specialized variants of the constitutive 20S proteasome in the immune system like the immunoproteasomes and the thymoproteasome contain active site-bearing... 
MULTIPLE-MYELOMA | IMMUNE-RESPONSE | CELLS | SELECTIVE INHIBITOR | BIOPHYSICS | IMMUNOPROTEASOME | BIOCHEMISTRY & MOLECULAR BIOLOGY | SITES | RESISTANCE | LMP7 | BORTEZOMIB | EXPRESSION | Animals | Antigen Presentation | Proteasome Inhibitors - pharmacology | Humans | Substrate Specificity | Proteasome Endopeptidase Complex - immunology | Immunologic Factors - pharmacology
Journal Article
Journal Article