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Journal of Molecular Graphics and Modelling, ISSN 1093-3263, 03/2016, Volume 64, pp. 121 - 130
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 03/2018, Volume 61, Issue 5, pp. 2124 - 2130
Starting from 1–4 and 7 structural templates, analogues based on bioisosteric replacements (5a–c vs 1, 2 and 6 vs 7) were synthesized for completing the SAR... 
CRYSTAL-STRUCTURES | POTENT | CHEMISTRY, MEDICINAL
Journal Article
Current Pharmaceutical Design, ISSN 1381-6128, 2002, Volume 8, Issue 8, pp. 615 - 657
Journal Article
European Journal of Medicinal Chemistry, ISSN 0223-5234, 04/2018, Volume 150, pp. 698 - 718
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 09/2013, Volume 54, Issue 39, pp. 5387 - 5390
We developed a novel and convenient stereoselective path for the preparation of pyrrolo-1,5-benzoxazepinones (PBOs). This innovative route envisaged the... 
Aryl–alkyl ether | Menthol | Pyrrolo-1,5-benzoxazepinones | Stereoselective synthesis | Aryl-alkyl ether | Pyrrolo-15-benzoxazepinones | DESIGN | ENANTIOSELECTIVE SYNTHESIS | CHIRAL AUXILIARIES | CHEMISTRY, ORGANIC | IDENTIFICATION | ONE-STEP | POTENT | ALPHA-HYDROXY ACIDS | ANTIVIRAL ACTIVITY | INHIBITORS | DERIVATIVES | Tetrahedrons | Biological | Access routes | Ethers | Employment
Journal Article
Journal Article
Investigational New Drugs, ISSN 0167-6997, 10/2016, Volume 34, Issue 5, pp. 663 - 676
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 03/2013, Volume 54, Issue 10, pp. 1233 - 1235
As a part of our work in the development of novel antimalarials, we were interested in elaborating an appropriate synthetic strategy for the preparation of... 
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 03/2013, Volume 54, Issue 10, pp. 1233 - 1235
As a part of our work in the development of novel antimalarials, we were interested in elaborating an appropriate synthetic strategy for the preparation of... 
Tetrahedrons | Strategy | Exposure | Dehydration | Scaffolds
Journal Article
Journal Article
Chemical Biology & Drug Design, ISSN 1747-0277, 02/2019, Volume 93, Issue 2, pp. 139 - 146
This study describes the activity of five natural hydroxycinnamic acids and derived compound: caffeic (1), rosmarinic (2), chlorogenic (3), and... 
natural products | molecular modeling | arginase inhibition | polyamines | enzyme kinetics | Leishmania amazonensis | CHEMISTRY, MEDICINAL | INHIBITS PROMASTIGOTE | BIOCHEMISTRY & MOLECULAR BIOLOGY | FLAVONOIDS | TRYPANOTHIONE | QUERCETIN | IN-VITRO | AMASTIGOTES | METABOLISM | GROWTH | NITRIC-OXIDE | REDUCTASE
Journal Article
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 03/2013, Volume 54, Issue 10, pp. 1233 - 1235
As a part of our work in the development of novel antimalarials, we were interested in elaborating an appropriate synthetic strategy for the preparation of... 
Endoperoxide | Trimethylsilyl triflate | Lactol | DIHYDROPLAKORTIN | DESIGN | ANALOGS | POTENT ANTIMALARIAL AGENTS | CHEMISTRY, ORGANIC | CLOTRIMAZOLE SCAFFOLD | YINGZHAOSU-A | PEROXIDES | LACTONES | BIOLOGICAL EVALUATION | INNOVATIVE PHARMACOPHORE
Journal Article
Journal Article