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Journal of Pharmaceutical and Biomedical Analysis, ISSN 0731-7085, 2010, Volume 53, Issue 3, pp. 603 - 608
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 08/2014, Volume 12, Issue 29, pp. 5407 - 5426
Journal Article
European Journal of Medicinal Chemistry, ISSN 0223-5234, 01/2018, Volume 144, pp. 672 - 681
Antagonists addressing selectively NMDA receptors containing the GluN2B subunit are of particular interest for the treatment of various neurological disorders... 
Docking studies | Ifenprodil binding site | GluN2B antagonists | Structure-affinity relationships | Affinity | Cytoprotective activity | Selectivity | NMDA receptor | Structure-activity relationships | GLUN2B SUBUNIT | ACTIVATION | CHEMISTRY, MEDICINAL | MECHANISM | SYNAPTIC PLASTICITY | METABOLISM | IN-VIVO | SELECTIVE NMDA | DERIVATIVES | BINDING
Journal Article
ChemMedChem, ISSN 1860-7179, 08/2014, Volume 9, Issue 8, p. 1697
  In accordance with a novel strategy for generating the 2-benzazepine scaffold by connecting C6-C1 and C3-N building blocks, a set of 5-phenylsulfanyl- and... 
Binding sites
Journal Article
ISSN 2040-2503, 8/2017, Volume 8, Issue 8, pp. 1697 - 175
It has been reported that bioisosteric replacement of an 1,2,4-oxadiazole ring by an 1,3,4-oxadiazole ring leads to higher polarity, reduced metabolic... 
Journal Article
MedChemComm, ISSN 2040-2503, 08/2017, Volume 8, Issue 8, p. 1697
It has been reported that bioisosteric replacement of an 1,2,4-oxadiazole ring by an 1,3,4-oxadiazole ring leads to higher polarity, reduced metabolic... 
Journal Article
ISSN 1477-0520, 7/2014, Volume 12, Issue 29, pp. 547 - 5426
A large set of tetrahydro-2-benzazepines with an α-hydroxy or α-(aryl)alkoxy substituted benzyl moiety in the 5-position was prepared according to the recently... 
Journal Article
Journal Article
ASSAY and Drug Development Technologies, ISSN 1540-658X, 08/2012, Volume 10, Issue 4, pp. 365 - 374
The standard assay for the determination of σ 1 receptor affinities of novel compounds is a competitive binding assay using [ 3 H]-(+)-pentazocine as... 
Original Articles
Journal Article
Journal Article
Archiv der Pharmazie, ISSN 0365-6233, 01/2014, Volume 347, Issue 1, pp. 21 - 31
Journal Article
Journal Article