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European Journal of Organic Chemistry, ISSN 1434-193X, 09/2019, Volume 2019, Issue 34, pp. 5937 - 5949
An approach to all isomeric 3‐pyridylcyclobutane‐derived building blocks, i.e. ketones, alcohols and amines, is described. Synthesis of the title compounds... 
Lead‐oriented synthesis | Heterocycles | Alkaloids | Pyridine | Cyclobutane | CONSTRUCTION | ARYLATION | Lead-oriented synthesis | CHEMISTRY, ORGANIC | OPTIMIZATION | INHIBITORS | DERIVATIVES | Alcohols
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 06/2019, Volume 2019, Issue 23, pp. 3744 - 3750
An approach to the synthesis of spirocyclic diazirines from cyclic ketones was examined on a series of carbo‐ and heterocyclic substrates containing the amine... 
Diazirines | Heterocycles | Photoaffinity probes | Synthesis design | Spiro compounds | ELUCIDATION | DESIGN | CHEMISTRY, ORGANIC | LIGAND | PROBES
Journal Article
Advanced Synthesis & Catalysis, ISSN 1615-4150, 12/2019, Volume 361, Issue 23, pp. 5428 - 5439
A convenient approach to the multigram synthesis of functionalized 1,2‐disubstituted cyclopropyltrifluoroborates was developed, based on Pd(II)‐ or... 
Cyclopropanes | Diazoalkanes | Organoboron compounds | Chan-Lam reaction | Suzuki-Miyaura reaction | REAGENTS | H BORYLATION | CYCLOPROPANATION | CHEMISTRY, ORGANIC | AUXILIARY | SUZUKI-MIYAURA | SCALE SYNTHESIS | PROTECTING GROUP | DRUGS | CHEMISTRY, APPLIED | Coupling (molecular) | Couplings | Stereoselectivity | Synthesis | Copper
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 10/2019, Volume 2019, Issue 37, pp. 6417 - 6421
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 05/2019, Volume 2019, Issue 18, pp. 2884 - 2898
An approach to synthesis of 2‐, 4‐, and 5‐bromooxazoles is described. The method was optimized, and its scope was extended to all three isomeric parents, as... 
Suzuki coupling | Heterocycles | Regioselectivity | Bromination | Oxazole | ANTIBIOTICS | STRUCTURAL ELUCIDATION | CHEMISTRY, ORGANIC | ABSOLUTE STEREOCHEMISTRY | STREPTOCHLORIN | POTENT | METHODOLOGY | INHIBITORS | DERIVATIVES | ANTIMICROBIAL ACTIVITY
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 11/2018, Volume 2018, Issue 40, pp. 5596 - 5604
An efficient approach to synthesis of various substituted 3‐azabicyclo[3.2.0]heptane‐derived building blocks based on [3+2] cycloaddition of... 
Bicyclic compounds | Cycloaddition | Parallel synthesis | Pyrrolidine | Cyclobutene | 2+2 PHOTOCYCLOADDITION | AMINO | 1,3-DIPOLAR CYCLOADDITION | CHEMISTRY, ORGANIC | PHOTOCHEMICAL-SYNTHESIS | EVP
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 06/2018, Volume 2018, Issue 22, pp. 2753 - 2761
The reaction of chloroximes that have a protected amino group and active methylene nitriles under basic conditions has been shown to give functionalized... 
Amino acids | Synthetic methods | Nitrogen heterocycles | Enantioselectivity | Regioselectivity | DESIGN | BUILDING-BLOCKS | ALKYLATION | AKP-001 | DIVERGENT SYNTHESIS | CHEMISTRY, ORGANIC | SULFONAMIDES | AMINOISOXAZOLES | INHIBITORS | DERIVATIVES | EFFICIENT | Nitriles | Drug discovery
Journal Article
Journal of Fluorine Chemistry, ISSN 0022-1139, 01/2020, Volume 229, p. 109407
•An approach to a series of diazolyl α,α-difluoroacetates is developed.•The strategy is based on deoxofluorination of diazolyl glyoxylates with morph-DAST.•Two... 
Deoxofluorination | gem-Difluorinated compounds | Azoles | Nitrogen heterocycles | Building blocks | ASYMMETRIC-SYNTHESIS | ACIDS | TRIFLUORIDE | CHEMISTRY, ORGANIC | CONVENIENT | FLUORINATION | DISCOVERY | CHEMISTRY, INORGANIC & NUCLEAR | OPTIMIZATION | BEARING | INHIBITORS | DERIVATIVES | Cyanide | Amides | Nitriles | Carboxylic acids | Chemical synthesis | Alcohols
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 05/2019, Volume 2019, Issue 18, pp. 2869 - 2869
The Front Cover shows Bromooxazoles – a widely exploited class of compounds which is known for many decades (depicted as a medieval Knight) in the quest for... 
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 11/2018, Volume 2018, Issue 40, pp. 5585 - 5595
An approach to 4‐hetarylisoxazole‐derived amines and other related 3,4‐disubstituted isoxazoles which relies on [3+2] cycloaddition of amino acid‐derived... 
Isoxazole | [3+2] Cycloaddition | Nitrogen heterocycles | Push‐Pull Enamines | Push-Pull Enamines | ISOXAZOLES | DESIGN | SAR | CHEMISTRY, ORGANIC | OPTIMIZATION | INHIBITORS | ANTAGONISTS | DISCOVERY | Amino acids
Journal Article
Tetrahedron, ISSN 0040-4020, 08/2015, Volume 71, Issue 33, p. 5169
Display Omitted 
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 06/2018, Volume 2018, Issue 22, pp. 2727 - 2727
The Cover Feature shows the retrosynthetic disconnection of 5‐amino‐3‐(piperidin‐4‐yl)isoxazole‐4‐carbonitrile, a representative of functionalized... 
Journal Article
Advanced Synthesis & Catalysis, ISSN 1615-4150, 09/2017, Volume 359, Issue 18, pp. 3077 - 3077
The front cover image, provided by Pavel Nosik, Andriy Gerasov, Sergey Ryabukhin, Oleksandr Grygorenko, and Dmitriy Volochnyuk illustrates the synthesis of... 
cycloaddition | bicyclic compounds | difluorocarbene | Ruppert–Prakash reagent | cycloalkanes | Amines | Alkenes | Chemical synthesis | Substrates
Journal Article