X
Search Filters
Format Format
Subjects Subjects
Subjects Subjects
X
Sort by Item Count (A-Z)
Filter by Count
humans (20) 20
index medicus (16) 16
animals (10) 10
chemistry, medicinal (9) 9
female (9) 9
adult (8) 8
gaba (7) 7
male (7) 7
receptors, gaba-a - metabolism (7) 7
analysis (6) 6
middle aged (6) 6
rats (6) 6
3-isoxazolol gaba antagonists (5) 5
aged (5) 5
structure-activity relationship (5) 5
subtypes (5) 5
agonists (4) 4
binding sites (4) 4
drug design (4) 4
glutamate (4) 4
pharmacology (4) 4
time factors (4) 4
tooth loss (4) 4
accurate docking (3) 3
analogs (3) 3
antagonists (3) 3
follow-up studies (3) 3
imidazole-4-acetic acid (3) 3
logistic models (3) 3
longitudinal studies (3) 3
mice (3) 3
models, molecular (3) 3
outcomes (3) 3
postmenopausal women (3) 3
prospective studies (3) 3
pyrazoles - chemistry (3) 3
receptors (3) 3
receptors, gaba-a - chemistry (3) 3
research (3) 3
risk (3) 3
structure–activity relationships (3) 3
tooth loss - epidemiology (3) 3
4--1-hydroxypyrazoles (2) 2
4-piol (2) 2
activation (2) 2
affinity (2) 2
aged, 80 and over (2) 2
analysis of variance (2) 2
binding (2) 2
biochemistry & molecular biology (2) 2
bone density (2) 2
cancer (2) 2
carcinoma (2) 2
cell line (2) 2
chemotherapy (2) 2
chi-square distribution (2) 2
cohort studies (2) 2
cross-sectional studies (2) 2
derivatives (2) 2
dose-response relationship, drug (2) 2
ecology (2) 2
ecosystems (2) 2
emergency medical care (2) 2
emergency medical services (2) 2
emergency medicine (2) 2
emergency services (2) 2
endocrinology & metabolism (2) 2
environmental sciences (2) 2
gaba receptor (2) 2
gaba receptors (2) 2
gaba-a receptor agonists - chemistry (2) 2
gaba-a receptor agonists - pharmacology (2) 2
gabaa receptor (2) 2
glide (2) 2
glycine (2) 2
history (2) 2
hospitals (2) 2
identification (2) 2
imidazoles - chemistry (2) 2
imidazoles - pharmacology (2) 2
in vitro techniques (2) 2
injuries (2) 2
kidney - drug effects (2) 2
life sciences (2) 2
ligands (2) 2
management (2) 2
mass (2) 2
membrane potentials - drug effects (2) 2
men (2) 2
metacarpal bone mineral density (2) 2
mice, inbred balb c (2) 2
mineral density (2) 2
modulation (2) 2
odds ratio (2) 2
oncology (2) 2
osteoporosis (2) 2
osteoporosis - complications (2) 2
patients (2) 2
periodontal diseases - epidemiology (2) 2
pharmacology & pharmacy (2) 2
more...
Library Location Library Location
Language Language
Publication Date Publication Date
Click on a bar to filter by decade
Slide to change publication date range


Journal Article
European Journal of Medicinal Chemistry, ISSN 0223-5234, 10/2018, Volume 158, p. 311
To access, purchase, authenticate, or subscribe to the full-text of this article, please visit this link: http://dx.doi.org/10.1016/j.ejmech.2018.08.094 The... 
Triazoles | Analysis | GABA | Investigations
Journal Article
JOURNAL OF MEDICINAL CHEMISTRY, ISSN 0022-2623, 06/2019, Volume 62, Issue 12, pp. 5797 - 5809
Given the heterogeneity within the gamma-amino-butyric acid (GABA) receptor and transporter families, a detailed insight into the pharmacology is still... 
GLYCINE | CHEMISTRY, MEDICINAL | ANALOGS | SUBTYPES | PHARMACOLOGICAL CHARACTERIZATION | GLUTAMATE | ANTAGONISTS | BINDING | SELECTIVITY | AGONISTS | MODULATION
Journal Article
Journal of Neuroscience, ISSN 0270-6474, 12/2014, Volume 34, Issue 49, pp. 16256 - 16272
In the present study, the orthosteric GABA sub(A) receptor (GABA sub(A)R) ligand 4,5,6,7-tetrahydroisothiazolo [5,4-c]pyridin-3-ol (Thio-THIP) was found to... 
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 02/2013, Volume 56, Issue 3, pp. 1211 - 1227
The isoxazol-3-one tautomer of the bicyclic isoxazole, 5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepin-3-ol (THAZ), has previously been shown to be a weak GABAA... 
INVERSE AGONISTS | ACID ANALOGS | SEROTONIN 5-HT2C RECEPTOR | 2-TRIAL MEMORY TASK | CHEMISTRY, MEDICINAL | AFFINITY | GLUTAMATE | DRUG DEVELOPMENT | FUNCTIONAL-CHARACTERIZATION | BINDING | DISCOVERY
Journal Article
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 03/2019, Volume 62, Issue 5, pp. 2798 - 2813
Gabazine, a gamma-aminobutyric acid type A (GABA(A)) receptor antagonist, has previously been reported to inhibit the binding of [H-3]NCS-382, a representative... 
POTENT | DESIGN | ACTIVATION | CHEMISTRY, MEDICINAL | SUBTYPES | PHARMACOLOGY | 3-ISOXAZOLOL GABA(A) ANTAGONISTS | RECEPTORS | DERIVATIVES | AGONISTS | MODULATION
Journal Article
ChemMedChem, ISSN 1860-7179, 10/2016, Volume 11, Issue 20, pp. 2299 - 2310
The ρ‐containing γ‐aminobutyric acid type A receptors (GABAARs) play an important role in controlling visual signaling. Therefore, ligands that selectively... 
imidazole-4-acetic acid | GABAC receptors | retinal vascular tone | ρ GABAA receptors | structure–activity relationships
Journal Article
ChemMedChem, ISSN 1860-7179, 10/2016, Volume 11, Issue 20, pp. 2299 - 2310
The rho -containing gamma -aminobutyric acid typeA receptors (GABA sub(A)Rs) play an important role in controlling visual signaling. Therefore, ligands that... 
Journal Article
ChemMedChem, ISSN 1860-7179, 10/2016, Volume 11, Issue 20, p. 2299
  The ρ-containing [gamma]-aminobutyric acid typeA receptors (GABAARs) play an important role in controlling visual signaling. Therefore, ligands that... 
Acids
Journal Article
ACS CHEMICAL NEUROSCIENCE, ISSN 1948-7193, 11/2019, Volume 10, Issue 11, pp. 4669 - 4684
Journal Article
ChemMedChem, ISSN 1860-7179, 11/2014, Volume 9, Issue 11, p. 2475
  A series of bioisosteric N1- and N2-substituted 5-(piperidin-4-yl)-3-hydroxypyrazole analogues of the partial GABAAR agonists 4-PIOL and 4-PHP have been... 
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 04/2010, Volume 53, Issue 8, pp. 3417 - 3421
A series of substituted 1-hydroxypyrazole analogues of the GABAA receptor partial agonist 5-(4-piperidyl)-3-isoxazolol (4-PIOL) have been synthesized and... 
Journal Article
Journal Article
No results were found for your search.

Cannot display more than 1000 results, please narrow the terms of your search.