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European Journal of Medicinal Chemistry, ISSN 0223-5234, 04/2019, Volume 167, pp. 269 - 290
ATP competitive inhibitors of DNA gyrase and topoisomerase IV have great therapeutic potential, but none of the described synthetic compounds has so far... 
GyrB | ParE | ATP competitive | N-phenylpyrrolamide | Inhibitor | Antibacterial | Topoisomerase IV | DNA gyrase | DESIGN | CHEMISTRY, MEDICINAL | ACID | ANALOGS | N-PHENYL-4,5-DIBROMOPYRROLAMIDES | DISCOVERY | ATPASE INHIBITORS | BIOLOGICAL EVALUATION | TOPOISOMERASE | PHENYLINDOLAMIDES | Methicillin | Biological products | Escherichia coli | DNA | Staphylococcus aureus infections | Bacteria | Liquid chromatography
Journal Article
Toxicology Letters, ISSN 0378-4274, 10/2017, Volume 280, pp. S111 - S111
Journal Article
Environmental Toxicology and Pharmacology, ISSN 1382-6689, 10/2016, Volume 47, p. 182
Structural analogs of bisphenol A are commonly used as its alternatives in industrial and commercial applications. Nevertheless, the question arises whether... 
Mass production | Endocrine system | Toxicity | Estrogen | Detoxification | Literature reviews | Analogs | Bisphenol A | Receptors | Metabolites | Bisphenols | Phenols | Metabolic pathways | Plastics
Journal Article
Expert Opinion on Therapeutic Patents, ISSN 1354-3776, 03/2019, Volume 29, Issue 3, pp. 171 - 180
Introduction: The bacterial topoisomerases DNA gyrase and topoisomerase IV are validated targets for development of novel antibacterial agents.... 
Antibacterial compounds | ATP-competitive inhibitors | DNA gyrase B | topoisomerase IV | PARE | DESIGN | CHEMISTRY, MEDICINAL | GYRB | EFFICACY | UREA INHIBITORS | CANDIDATE | DISCOVERY | BIOLOGICAL EVALUATION | PHARMACOLOGY & PHARMACY | Index Medicus
Journal Article
Farmacevtski Vestnik, ISSN 0014-8229, 12/2016, Volume 67, Issue 6, pp. 386 - 396
Journal Article
Bioorganic & Medicinal Chemistry Letters, ISSN 0960-894X, 2010, Volume 20, Issue 3, pp. 958 - 962
Journal Article
Journal Article
Journal Article
Current Topics in Medicinal Chemistry, ISSN 1568-0266, 2014, Volume 14, Issue 1, pp. 130 - 151
Journal Article
Farmacevtski Vestnik, ISSN 0014-8229, 2014, Volume 65, Issue 2, pp. 118 - 128
Journal Article
Journal Article
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