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Biochemistry, ISSN 0006-2960, 05/2007, Volume 46, Issue 20, pp. 5960 - 5971
Journal Article
Molecular Cancer Therapeutics, ISSN 1535-7163, 12/2011, Volume 10, Issue 12, pp. 2426 - 2436
Journal Article
eLife, ISSN 2050-084X, 07/2016, Volume 5, Issue 2016
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 11/2011, Volume 54, Issue 21, pp. 7579 - 7587
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 06/2013, Volume 56, Issue 11, pp. 4597 - 4610
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 02/2016, Volume 59, Issue 3, pp. 985 - 1002
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 02/2018, Volume 61, Issue 3, pp. 989 - 1000
Antibody–drug conjugates (ADCs) have become an important therapeutic modality for oncology, with three approved by the FDA and over 60 others in clinical... 
ANTICANCER ACTIVITY | ATTACHMENT SITE | POTENT | CHEMISTRY, MEDICINAL | STABILITY | INHIBITORS | ADCS | NEXT-GENERATION | CANCER-THERAPY | CATHEPSIN-B | STRATEGIES
Journal Article
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 02/2010, Volume 53, Issue 3, pp. 1086 - 1097
Journal Article
Bioorganic & Medicinal Chemistry Letters, ISSN 0960-894X, 06/2019, Volume 29, Issue 12, pp. 1522 - 1531
Disruption of interleukin-13 (IL-13) signaling with large molecule antibody therapies has shown promise in diseases of allergic inflammation. Given that IL-13... 
Janus Kinase | JAK | Atopic dermatitis | Structure-based design | Interleukin-13 | IL-13 | JAK2 | JAK1 | Asthma | CHEMISTRY, MEDICINAL | CHEMISTRY, ORGANIC | IDENTIFICATION | Viral antibodies | Antibodies | Mutual fund industry | Interleukins
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 11/2011, Volume 54, Issue 22, pp. 7815 - 7833
Journal Article
ACS Medicinal Chemistry Letters, ISSN 1948-5875, 04/2016, Volume 7, Issue 4, pp. 351 - 356
Inhibition of phosphoinositide 3-kinase (PI3K) signaling is an appealing approach to treat brain tumors, especially glioblastoma multiforme (GBM). We... 
kinase inhibitor | CNS | blood-brain barrier penetration | PI3K | oncology | POTENT | CHEMISTRY, MEDICINAL
Journal Article
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