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Annals of the New York Academy of Sciences, ISSN 0077-8923, 11/2019, Volume 1456, Issue 1
Journal Article
Basic & clinical pharmacology & toxicology, ISSN 1742-7835, 07/2019
Journal Article
Bone, ISSN 8756-3282, 01/2020, Volume 130, p. 115079
Infusion of the incretin hormone glucose-dependent insulinotropic polypeptide (GIP) suppresses the bone resorption marker carboxy-terminal type 1 collagen... 
Glucose-dependent insulinotropic polypeptide receptor antagonist | Glucose-dependent insulinotropic polypeptide | Gut-bone axis
Journal Article
ISSN 0040-4020, 2017
We here report the preparation of a new 2,6,8-trisubstituted bicyclic tripeptidomimetic scaffold through TFA-mediated cyclization of a linear precursor... 
CXCR4 antagonist | Scaffold | Tripeptidomimetic
Journal Article
Journal of Leukocyte Biology, ISSN 0741-5400, 08/2018, Volume 104, Issue 2, pp. 423 - 434
Chemokine–chemokine receptor (CKR) interactions are traditionally described by a two‐step/two‐site mechanism that details the major contact points between... 
chemokine | CCR6 | two‐step/two‐site paradigm | CCL20 | mutagenesis | chemokine receptor | two-step/two-site paradigm | ACTIVATION | RECOGNITION | CC-CHEMOKINE | RECEPTOR | CXCR4 | IMMUNOLOGY | MACROPHAGE INFLAMMATORY PROTEIN-3-ALPHA/CCL20 | CELL BIOLOGY | INHIBITION | ANTAGONISTS | HEMATOLOGY | EXPRESSION | LYMPHOCYTES
Journal Article
Diabetologia, ISSN 0012-186X, 02/2018, Volume 61, Issue 2, p. 413
To access, purchase, authenticate, or subscribe to the full-text of this article, please visit this link: http://dx.doi.org/10.1007/s00125-017-4447-4... 
Journal Article
ISSN 0968-0896, 2017
Here we report a series of close analogues of our recently published scaffold-based tripeptidomimetic CXCR4 antagonists, containing positively charged... 
CXCR4 antagonist | Peptidomimetic | Scaffold
Journal Article
European Journal of Immunology, ISSN 0014-2980, 07/2014, Volume 44, Issue 7, pp. 1904 - 1912
Journal Article
Frontiers in Immunology, ISSN 1664-3224, 2014, Volume 5
Biased signaling or functional selectivity occurs when a 7TM receptor preferentially activates one of several available pathways. It can be divided into three... 
Biased signaling | Chemokine system | b-arrestin recruitment | Ligand/receptor/tissue bias | Pathway-specific drug development | 7TM-receptor | 7TM structure-function | G protein coupling | biased signaling | chemokine system | ligand/receptor/tissue bias
Journal Article
Physiological Reports, 03/2018, Volume 6, Issue 6, pp. e13657 - n/a
The current available insulin therapies decrease blood glucose but are associated with the risk of developing hypoglycemia. Glucagon is a counter regulatory... 
glucagon | Diabetes | insulin | hypoglycemia | Hepatocytes | Glucagon | Glycogen | Diabetes mellitus | Liver | Rodents | Cyclic AMP | Glucose | Hypoglycemia | Insulin | Blood
Journal Article
ISSN 1464-3391, 2014
Structure–activity relationship studies of the cyclopentapeptide CXCR4 antagonists (cyclo(-l-/d-Arg1-Arg2-2-Nal3-Gly4-d-Tyr5-)) suggest that the... 
Cyclopentapeptide | CXCR4 antagonist | Peptidomimetic | Scaffold
Journal Article
Frontiers in immunology, ISSN 1664-3224, 2014, Volume 5, p. 277
Biased signaling or functional selectivity occurs when a 7TM-receptor preferentially activates one of several available pathways. It can be divided into three... 
Journal Article