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Neuropharmacology, ISSN 0028-3908, 07/2018, Volume 136, Issue Pt C, pp. 427 - 437
Journal Article
Nature Communications, ISSN 2041-1723, 2015, Volume 6, Issue 1, pp. 10156 - 10156
Journal Article
Journal Article
Angewandte Chemie International Edition, ISSN 1433-7851, 01/2013, Volume 52, Issue 2, pp. 508 - 516
Journal Article
Angewandte Chemie, ISSN 1433-7851, 01/2013, Volume 52, Issue 2, pp. 508 - 516
  Cell-membrane-spanning Gprotein coupled receptors (GPCRs) belong to the most important therapeutic target structures. Endogenous transmitters bind from the... 
Proteins | Binding sites | Drugs | Binding | Receptors | Side effects | Activation | Selectivity | Modulators
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 01/2015, Volume 58, Issue 2, pp. 560 - 576
Aiming to design partial agonists for a G-protein-coupled receptor based on dynamic ligand binding, we synthesized three different series of bipharmacophoric... 
Receptor, Muscarinic M1 - agonists | Animals | Cricetulus | Muscarinic Agonists - pharmacology | Drug Design | Structure-Activity Relationship | CHO Cells | Muscarinic Agonists - chemical synthesis
Journal Article
Science Signaling, ISSN 1945-0877, 10/2013, Volume 6, Issue 298, pp. ra93 - ra93
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 08/2014, Volume 57, Issue 15, pp. 6739 - 6750
Journal Article