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Bioorganic & Medicinal Chemistry Letters, ISSN 0960-894X, 02/2020, Volume 30, Issue 3, p. 126838
[Display omitted] A series of indane-type acetamide and propanamide analogues were investigated as TRPV1 antagonists. The analysis of structure–activity... 
Vanilloid receptor 1 | TRPV1 antagonist | Analgesic | VANILLOID-1 ANTAGONISTS | CHEMISTRY, MEDICINAL | 2-(3-FLUORO-4-METHYLSULFONAMIDOPHENYL)PROPANAMIDES | PYRIDINE | C-REGION ANALOGS | 2-(3-FLUORO-4-METHYLSULFONYLAMINOPHENYL)PROPANAMIDES | CHEMISTRY, ORGANIC | CAPSAICIN RECEPTOR | PAIN | PHARMACOLOGY
Journal Article
Journal Article
Journal Article
Journal of Medicinal Chemistry, ISSN 0022-2623, 10/2012, Volume 55, Issue 19, pp. 8392 - 8408
Journal Article
Journal Article
European Journal of Pharmacology, ISSN 0014-2999, 03/2020, Volume 871, p. 172934
The TRPV1 ion channel is a neuronal sensor that plays an important role in nociception and neuropathic as well as inflammatory pain. In clinical trials,... 
TRPV1 | Analgesics | Hyperthermia | Body temperature regulation | ACTIVATION | ANTAGONIST | CAPSAICIN 8-PERCENT PATCH | PAIN | VR1 | PHARMACOLOGY | NEURONS | PHARMACOLOGY & PHARMACY | CHANNELS | HYPERALGESIA
Journal Article
European Journal of Pharmacology, ISSN 0014-2999, 10/1998, Volume 359, Issue 2-3, pp. 143 - 150
The effect of the Poly (adenosine 5′-diphosphate ribose) synthetase (PARS) inhibitor 3-aminobenzamide on (i) infarct size caused by regional myocardial... 
PARS (Poly (adenosine 5′-diphosphate ribose) synthetase) | Heart | Cardiomyoblast, human | Reperfusion injury | Oxygen radical | Pig | PARS (Poly (adenosine 5'-diphosphate ribose) synthetase) | POLY(ADP-RIBOSE) POLYMERASE | CELLS | ACTIVATION | DNA STRAND-BREAKS | PEROXYNITRITE | PARS (poly (adenosine 5 '-diphosphate ribose) synthetase) | reperfusion injury | oxygen radical | heart | FREE-RADICALS | cardiomyoblast | METABOLISM | NITRIC-OXIDE | PHARMACOLOGY & PHARMACY | human | SUPEROXIDE-DISMUTASE | Oxidants - pharmacology | Heart Rate - drug effects | Poly(ADP-ribose) Polymerases - drug effects | Myocardial Reperfusion Injury - pathology | Benzamides - therapeutic use | Swine | Myocardial Infarction - pathology | Heart Rate - physiology | Myocardial Infarction - physiopathology | Benzamides - pharmacology | Blood Pressure - drug effects | Blood Pressure - physiology | Cell Death - drug effects | Myocardial Reperfusion Injury - drug therapy | Eukaryotic Cells - enzymology | Cells, Cultured | Enzyme Inhibitors - pharmacology | Hydrogen Peroxide - pharmacology | Myocardium - pathology | Enzyme Inhibitors - therapeutic use | Poly(ADP-ribose) Polymerase Inhibitors | Eukaryotic Cells - pathology | Myocardial Reperfusion Injury - physiopathology | Myocardium - cytology | Myocardium - enzymology | Animals | Eukaryotic Cells - drug effects | Hemodynamics
Journal Article
British Journal of Pharmacology, ISSN 0007-1188, 08/1995, Volume 115, Issue 7, pp. 1175 - 1181
Journal Article