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Advanced Synthesis & Catalysis, ISSN 1615-4150, 12/2019, Volume 361, Issue 23, pp. 5428 - 5439
A convenient approach to the multigram synthesis of functionalized 1,2‐disubstituted cyclopropyltrifluoroborates was developed, based on Pd(II)‐ or... 
Cyclopropanes | Diazoalkanes | Organoboron compounds | Chan-Lam reaction | Suzuki-Miyaura reaction | REAGENTS | H BORYLATION | CYCLOPROPANATION | CHEMISTRY, ORGANIC | AUXILIARY | SUZUKI-MIYAURA | SCALE SYNTHESIS | PROTECTING GROUP | DRUGS | CHEMISTRY, APPLIED | Coupling (molecular) | Couplings | Stereoselectivity | Synthesis | Copper
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 11/2017, Volume 2017, Issue 43, pp. 6450 - 6456
Syntheses of bicyclo[1.1.1]pentane‐derived azides and terminal alkynes – interesting substrates for click reactions – are described. With a few exceptions,... 
Azides | Propellane | Cage compounds | Click chemistry | Nitrogen heterocycles | Alkynes | CUBANES | EXPEDIENT SYNTHESIS | BRIDGEHEAD | CHEMISTRY, ORGANIC | TINKERTOY CONSTRUCTION SET | RING-SYSTEM | AZIDE | RECEPTOR ANTAGONIST | MEDICINAL CHEMISTRY | BIOORTHOGONAL REACTIONS | BIOCONJUGATION
Journal Article
Synthesis, ISSN 0039-7881, 05/2018, Volume 50, Issue 10, pp. 1973 - 1978
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 12/2018, Volume 59, Issue 52, pp. 4611 - 4615
[Display omitted] •Synthesis of azabicyclo[5.1.0]octane(methanoazepane)-derived amino acids and diamines is reported.•The Corey–Chaikovsky cyclopropanation is... 
Bicyclic compounds | Diamines | Amino acids | Azepane | Cyclopropane | Pyrrolidine | ASYMMETRIC-SYNTHESIS | MICHAEL ADDITION-REACTIONS | CHEMISTRY, ORGANIC | ALPHA-AMINO-ACIDS | INTERNAL DOUBLE-BOND | NI(II) COMPLEXES | HALOESTER | POTENT | STEREOSELECTIVE-SYNTHESIS | INHIBITOR | HOMOLOGATION | Proline | Alkaloids | Cyclopropane compounds | Resveratrol
Journal Article
Synthesis, ISSN 0039-7881, 04/2015, Volume 47, Issue 8, pp. 1123 - 1130
Abstract The synthesis of optically pure (1 S ,4 S )-2,5-diazabicyclo[2.2.1]heptane-1-carboxylic acid starting from easily available ‘chiral pool’ l... 
paper | SUBSTITUTION | ANALOGS | amino acids | CHEMISTRY, ORGANIC | BETA-AMINO-ACID | DENDRIMERS | PROTEIN-STRUCTURE PREDICTION | PEPTIDOMIMETICS | PEPTIDES | Strecker reaction | bicyclic compounds | SEQUENCE | SECONDARY STRUCTURE PREDICTION | BEARING | molecular rigidity | nucleophilic cyclization
Journal Article
Synlett, ISSN 0936-5214, 02/2014, Volume 25, Issue 3, pp. 355 - 358
Abstract A scalable synthesis was developed of 3,5-methanoni­pecotic acid (3-azabicyclo[3.1.1]heptane-1-carboxylic acid), a rare example of a conformationally... 
letter | conformation | bicyclic compounds | heterocycles | amino acids | 2,4-METHANOPROLINE | ANALOGS | CHEMISTRY, ORGANIC | AQUEOUS-SOLUTION | MEDICINAL CHEMISTRY | HAIRPIN FORMATION | PEPTIDOMIMETICS | PEPTIDES | DIVERSITY | STEREOSELECTIVE-SYNTHESIS | INHIBITORS
Journal Article
Tetrahedron: Asymmetry, ISSN 0957-4166, 12/2017, Volume 28, Issue 12, pp. 1817 - 1822
[Display omitted] An approach to the synthesis and resolution of five- and six-membered lactams (i.e., 5-oxopyrrolidine- and 6-oxopiperidine-3-carboxylic... 
ASYMMETRIC-SYNTHESIS | ENANTIOMERS | GAMMA-LACTAMS | DEBENZYLATION | CHEMISTRY, PHYSICAL | BETA-PROLINE | AMIDES
Journal Article
Synthesis (Germany), ISSN 0039-7881, 04/2015, Volume 47, Issue 8, pp. 1123 - 1130
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 09/2019, Volume 2019, Issue 33, pp. 5624 - 5635
Preparation of 2,2‐disubstituted and 2‐monosubstituted alkenylboronic acid esters from aliphatic and aromatic ketones and aldehydes by the boron‐Wittig... 
Boron‐Wittig olefination | Boronic esters | Alkenes | Organoboron compounds | Boron-Wittig olefination | HYDROBORATION | DIVERSIFICATION | ESTERS | CHEMISTRY, ORGANIC | CARBANIONS | ALKYNES | BORYLATION | Methane | Ketones | Aldehydes
Journal Article
Journal of Organic Chemistry, ISSN 0022-3263, 03/2018, Volume 83, Issue 6, pp. 3265 - 3274
Facile synthesis of 5-fluoropyrazoles by direct fluorination of pyrazoles with N-fluorobenzenesulfonimide (NFSI) was elaborated. This approach was used to... 
CYCLOADDITION | SUBSTITUTION | 3-COMPONENT SYNTHESIS | NANO2 | REGIOSELECTIVE SYNTHESIS | CHEMISTRY | CHEMISTRY, ORGANIC | FLUORINATED PYRAZOLES | ALKYNES | IN-SITU GENERATION | ACCESS
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 03/2018, Volume 83, Issue 6, pp. 3265 - 3274
Facile synthesis of 5-fluoropyrazoles by direct fluorination of pyrazoles with N-fluoro­benzene­sulfonimide (NFSI) was elaborated. This approach was used to... 
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 05/2014, Volume 55, Issue 22, pp. 3312 - 3315
[Display omitted] An efficient method for the preparation of Boc-protected 4,5-methano-β-proline—a novel bicyclic cyclopropane-containing β-amino acid—was... 
Bicyclic compounds | Proline analogues | Simmons–Smith reaction | Cyclopropane | β-Amino acids | Simmons-Smith reaction | ANALOGS | CHEMISTRY, ORGANIC | ALPHA-AMINO-ACIDS | RECEPTOR | EQUIVALENTS | BETA | beta-Amino acids | PEPTIDES | PYRROLIDINES | FOLDAMERS | DERIVATIVES | PROLINE | Tetrahedrons | Itaconic acid | Synthesis (chemistry) | Construction | Isomers
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 05/2014, Volume 55, Issue 22, p. 3312
Display Omitted 
Proline
Journal Article
Tetrahedron: Asymmetry, ISSN 0957-4166, 12/2015, Volume 26, Issue 21-22, pp. 1268 - 1272
[Display omitted] The synthesis of both racemic and enantiomerically pure (1R,6S)-3,4-methanonipecotic acid, a cyclopropane-containing β-amino acid, which is a... 
HAIRPIN FORMATION | AMINO-ACID | DYSOXYLUM-LENTICELLARE | EVOLVING ROLE | NATURAL-PRODUCTS | DRUG DISCOVERY | CHEMISTRY, ORGANIC | CHEMISTRY, PHYSICAL | BETA-PEPTIDES | STEM | CHEMISTRY, INORGANIC & NUCLEAR | Enantiomers | Resveratrol | Malic acid | Amino acids | Drug discovery | Cyclopropane compounds
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 10/2014, Volume 55, Issue 43, pp. 5970 - 5972
An unusual rearrangement of a 1-oxa-6-azaspiro[2.5]octane derivative giving access to novel 5-substituted 2-azabicyclo[3.1.0]hexanes is described. The... 
Bicyclic compounds | Cyclopropanes | Conformational restriction | β-Amino acids | Epoxides | DESIGN | beta-Amino acids | AMINO-ACIDS | Cyclopropanes Epoxides | CHEMISTRY, ORGANIC | INHIBITOR | PROLINE | Tetrahedrons | Amino acids | Synthesis (chemistry) | Derivatives
Journal Article
Angewandte Chemie International Edition, ISSN 1433-7851, 11/2016, Volume 55, Issue 47, pp. 14788 - 14792
A conformationally restricted monofluorinated α‐amino acid, (3‐fluorobicyclo[1.1.1]pentyl)glycine (F‐Bpg), was designed as a label for the structural analysis... 
peptides | solid-state NMR spectroscopy | amino acids | fluorine | propellanes | Membrane lipids | Nuclear magnetic resonance spectroscopy | Fluorides | Peptides | Glycine
Journal Article
Angewandte Chemie (International ed. in English), ISSN 1433-7851, 11/2016, Volume 55, Issue 47, pp. 14788 - 14792
A conformationally restricted monofluorinated α-amino acid, (3-fluorobicyclo[1.1.1]pentyl)glycine (F-Bpg), was designed as a label for the structural analysis... 
Journal Article
RSC Advances, ISSN 2046-2069, 2016, Volume 6, Issue 27, pp. 22737 - 22748
Differentiation of identical electrophilic functional groups (carboxylates) by a strategically placed internal nucleophile (an amino group) in cyclic... 
CHEMISTRY, MULTIDISCIPLINARY | DIVERSITY-ORIENTED SYNTHESIS | PEPTIDES
Journal Article
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