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chemistry, organic (24) 24
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ISSN 1477-0520, 7/2019, Volume 17, Issue 26, pp. 6432 - 644
A highly regioselective metal-free direct C-H thiolation of 2-pyridones with disulfides or thiols has been developed. A combination of persulfate and a... 
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 2018, Volume 16, Issue 15, pp. 2697 - 2704
The persulfate-meditated oxidative C-N bond coupling of the C-H bond of quinoxalinones and the N-H bond of NH-sulfoximines is reported. The reaction proceeds... 
IN-VITRO | AMINATION | MILD CONDITIONS | RADICAL CYCLIZATION | DRUG DISCOVERY | CHEMISTRY, ORGANIC | QUINOXALIN-2(1H)-ONES | INHIBITORS | DERIVATIVES | TRANSITION-METAL-FREE | ALDOSE REDUCTASE | Hydrogen bonds | Substrates | Coupling
Journal Article
Advanced Synthesis & Catalysis, ISSN 1615-4150, 09/2018, Volume 360, Issue 17, pp. 3345 - 3355
A facile and efficient oxidative C−H acylation of N‐substituted pyrazolones using α‐oxocarboxylic acids as an acyl group source was developed. A combination of... 
decarboxylative coupling | α-oxocarboxylic acid | Copper | pyrazolone | acylation | SELECTIVE OXIDATION | SULFOXIMINES | CHEMISTRY, ORGANIC | alpha-oxocarboxylic acid | COPPER-OXIDE | AMINES | LIGHT PHOTOREDOX CATALYSIS | KETO ACIDS | IODINE-MAGNESIUM EXCHANGE | N BOND FORMATION | CHEMISTRY, APPLIED | CARBOXYLIC-ACIDS | ACTIVATED PERSULFATE | Pyrazolones | Decarboxylation | Potassium persulfate | Acylation
Journal Article
ISSN 1477-0520, 1/2018, Volume 16, Issue 3, pp. 424 - 432
A highly efficient protocol for a direct thiolation of N -substituted pyrazolones with diaryl disulfides is described. Using a combination of DABCO and silver(... 
Journal Article
ORGANIC & BIOMOLECULAR CHEMISTRY, ISSN 1477-0520, 07/2019, Volume 17, Issue 26, pp. 6432 - 6440
A highly regioselective metal-free direct C-H thiolation of 2-pyridones with disulfides or thiols has been developed. A combination of persulfate and a... 
C-H ALKYLATION | THIOLS | ACID | ARYLATION | BOND FUNCTIONALIZATION | SYNTHETIC METHODS | ARYL SULFIDES | CHEMISTRY, ORGANIC | SULFUR | DIRECT ACCESS | ENANTIOSELECTIVE SULFENYLATION
Journal Article
ISSN 1477-0520, 5/2017, Volume 15, Issue 2, pp. 432 - 4327
A copper-catalyzed oxidative decarboxylative coupling of α-keto acids with NH -sulfoximines has been developed. With CuBr as the catalyst and K 2 S 2 O 8 as... 
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 04/2015, Volume 80, Issue 7, pp. 3447 - 3454
Journal Article
ISSN 1477-0520, 4/2018, Volume 16, Issue 15, pp. 2697 - 274
The persulfate-meditated oxidative C-N bond coupling of the C-H bond of quinoxalinones and the N-H bond of NH -sulfoximines is reported. The reaction proceeds... 
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 2017, Volume 15, Issue 20, pp. 4320 - 4327
A copper-catalyzed oxidative decarboxylative coupling of alpha-keto acids with NH-sulfoximines has been developed. With CuBr as the catalyst and K2S2O8 as the... 
HETEROAROMATIC CARBOXYLIC-ACIDS | ARYL BROMIDES | AROYLATION | PALLADIUM | PHOTOREDOX | ARYLATION | CHEMISTRY, ORGANIC | OXOCARBOXYLIC ACIDS | C-H ACTIVATION | ORTHO-ACYLATION | NH-SULFOXIMINES
Journal Article
Synthesis, ISSN 0039-7881, 06/2018, Volume 50, Issue 12, pp. 2337 - 2346
Abstract A highly efficient iodine-catalyzed oxidative cross-dehydrogenative coupling reaction of quinoxalinones and indoles has been developed. Without the... 
paper | oxidative coupling | iodine | quinoxalinone | indole | metal-free | TYROSINE KINASE-ACTIVITY | MOLECULAR-IODINE | ONE-POT SYNTHESIS | EFFICIENT SYNTHESIS | CHEMISTRY, ORGANIC | C-H ACTIVATION | SIMPLE ARENES | N BOND FORMATION | GROWTH-FACTOR | PART 2 | DERIVATIVES
Journal Article
Organic & biomolecular chemistry, ISSN 1477-0520, 01/2018, Volume 16, Issue 3, pp. 424 - 432
A highly efficient protocol for a direct thiolation of N-substituted pyrazolones with diaryl disulfides is described. Using a combination of DABCO and... 
Journal Article
Organic & biomolecular chemistry, ISSN 1477-0520, 01/2016, Volume 14, Issue 2, pp. 590 - 597
A new synthesis of sulfonamides has been developed via an iodine-catalyzed sulfonylation of amines with arylsulfonyl hydrazides. This metal-free strategy... 
Journal Article
ISSN 1477-0520, 12/2015, Volume 14, Issue 2, pp. 59 - 597
A new synthesis of sulfonamides has been developed via an iodine-catalyzed sulfonylation of amines with arylsulfonyl hydrazides. This metal-free strategy... 
Journal Article
Applied Catalysis A, General, ISSN 0926-860X, 01/2018, Volume 549, pp. 134 - 140
[Display omitted] •A rapid one-pot catalytic process for the synthesis of double-capped oligoesters from lactones is described.•A double-capped... 
Caprolactone | Transesterification | Oligoesters | Double-capped oligolactones | L-LACTIDE | CHEMISTRY, PHYSICAL | OLIGOMERS | POLYLACTIDES | ENVIRONMENTAL SCIENCES | BIODEGRADABLE POLYMERS | POLY(LACTIC ACID) | RING-OPENING POLYMERIZATION | ALCOHOLYSIS | Polymerization | Amides | Lithium compounds
Journal Article
Organic Letters, ISSN 1523-7060, 04/2009, Volume 11, Issue 7, pp. 1511 - 1514
A method for the direct arylation of benzotriazepines is reported, employing an aryl iodide as the coupling partner, copper iodide as the catalyst, and lithium... 
H BOND ACTIVATION | FUNCTIONALIZATION | POTENT | QUINOLINES | CHEMISTRY, ORGANIC | INHIBITORS | PYRIDINES | ANTAGONISTS | ALKENYLATION | DISCOVERY | Iodides - chemistry | Molecular Structure | Copper - chemistry | Catalysis | Benzazepines - chemical synthesis | Benzazepines - chemistry
Journal Article
Organic & Biomolecular Chemistry, ISSN 1477-0520, 01/2019, Volume 17, Issue 26, pp. 6432 - 6440
A highly regioselective metal-free direct C–H thiolation of 2-pyridones with disulfides or thiols has been developed. A combination of persulfate and a... 
Sulfide | Thiols | Regioselectivity | Lithium chloride | Metals | Lithium chlorides
Journal Article
Organic Letters, ISSN 1523-7060, 07/2010, Volume 12, Issue 13, pp. 2978 - 2981
An efficient method is reported for the preparation of multicyclic pyridines and quinolines by a rhodium-catalyzed intramolecular C−H bond functionalization... 
ROUTE | CYCLOADDITION | ACETYLENES | ACTIVATION | DIRECT ARYLATION | HETEROCYCLES | ONE-POT SYNTHESIS | CHEMISTRY, ORGANIC | RUTHENIUM | KINASE INHIBITORS | ALKYNES | Quinolines - chemical synthesis | Cyclization | Pyridines - chemistry | Stereoisomerism | Quinolines - chemistry | Pyridines - chemical synthesis | Molecular Structure
Journal Article
Synthesis, ISSN 0039-7881, 04/2013, Volume 45, Issue 7, pp. 936 - 942
Abstract A practical protocol for the one-pot synthesis of N-substituted 2-aminoazole derivatives is described, employing simple azole substrates, nitrogen... 
paper | carbon-nitrogen bond formation | benzoxazole | iodine | N-substituted 2-aminoazoles | one-pot synthesis | AZOLES | CHEMISTRY, ORGANIC | C-H BONDS | DISCOVERY | AMINATION | OREXIN RECEPTOR ANTAGONIST | OXIDANT | BENZOXAZOLES
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 04/2019, Volume 2019, Issue 16, pp. 2759 - 2766
A novel copper‐catalyzed direct C–H thiolation and thiocyanation of uracils using disulfides and thiocyanate salts respectively as coupling partners are... 
Thiocyanation | Copper | Uracil | Thiolation | Disulfides | INSERTION | PYRAZOLONES | CHEMISTRY, ORGANIC | SULFUR | INDOLES | BIOLOGICAL EVALUATION | INHIBITORS | DERIVATIVES | EFFICIENT | CYCLIZATION
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 02/2020, Volume 2020, Issue 8, pp. 961 - 970
Metal‐free approach for direct C–H thiolation and thiocyanation of N‐substituted pyrazolones with disulfides and thiocyanate salts, respectively, are... 
Thiocyanation | Pyrazolone | Metal‐free | Thiolation | Disulfide | Metal-free | ARYL SULFIDES | CHEMISTRY, ORGANIC | SULFENYLATION | DIRECT ACCESS | INDOLES | FUNCTIONALIZATION | S BOND FORMATION | HETEROCYCLES | REGIOSELECTIVE SYNTHESIS | DIMETHYL-SULFOXIDE | DERIVATIVES
Journal Article
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