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chemistry, organic (199) 199
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European Journal of Organic Chemistry, ISSN 1434-193X, 06/2019, Volume 2019, Issue 24, pp. 3949 - 3954
A facile and general method for the synthesis of indole‐1‐carboxamides was developed via copper(I)‐catalyzed N‐carboxamidation of indoles with isocyanates... 
Isocyanates | Carboxamidation | Synthesis design | Indole derivatives | Homogeneous catalysis | 2-SUBSTITUTED INDOLES | ANNULATION | CHEMISTRY, ORGANIC | SALTS | CONSTRUCTION | BIOLOGICAL EVALUATION | INHIBITORS | DERIVATIVES | EFFICIENT | C-H AMINATION | CYCLIZATION | Copper | Methods
Journal Article
Advanced Synthesis & Catalysis, ISSN 1615-4150, 10/2008, Volume 350, Issue 14‐15, pp. 2153 - 2167
In the past decade alkynes have become attractive starting materials for the synthesis of a variety of indole derivatives. This review summarizes the... 
hydrazines | indoles | nitroarenes | anilines | alkynes | isonitriles | Hydrazines | Anilines | Indoles | Nitroarenes | Isonitriles | Alkynes | 2-SUBSTITUTED INDOLES | ONE-POT SYNTHESIS | CHEMISTRY, ORGANIC | TERMINAL ALKYNES | INTERNAL ALKYNES | HIGHLY EFFICIENT PROMOTERS | COUPLING REACTION | PHOSPHORUS-ACIDS | CHEMISTRY, APPLIED | 2,3-DISUBSTITUTED INDOLES | SUBSTITUTED INDOLES | HECK REACTION
Journal Article
Tetrahedron, ISSN 0040-4020, 2011, Volume 67, Issue 38, pp. 7195 - 7210
The indole alkaloids, ranging from lysergic acid to vincristine, have long inspired organic synthesis chemists. Interest in developing new methods for indole... 
INDOLE-3-CARBOXYLIC ACID-DERIVATIVES | 2-SUBSTITUTED INDOLES | ONE-POT SYNTHESIS | CATALYZED SYNTHESIS | REGIOSELECTIVE SYNTHESIS | CHEMISTRY, ORGANIC | ALLENE INTRAMOLECULAR CYCLOADDITION | 2,3-DISUBSTITUTED INDOLES | SUBSTITUTED INDOLES | C-H AMINATION | 3-SUBSTITUTED INDOLES | LSD (Drug)
Journal Article
Chemical communications (Cambridge, England), ISSN 1359-7345, 09/2015, Volume 51, Issue 73, pp. 13898 - 13901
A simple, efficient and practical metal-free C-H sulfenylation process at the C2 position of non-protected indoles has been developed. 2-Thioindoles were... 
Indoles - chemistry | Molecular Structure | Succinimides - chemistry
Journal Article
European Journal of Organic Chemistry, ISSN 1434-193X, 08/2019, Volume 2019, Issue 30, pp. 4844 - 4854
Herein, we report a new transition‐metal‐free robust and cost‐effective method for synthesis of 1,2‐disubstituted indoles from easily available unactivated... 
Heterocycles | Amides | Indoles | Cyclization | Intramolecular condensation | 2-SUBSTITUTED INDOLES | ONE-POT SYNTHESIS | ARYLATION | EFFICIENT SYNTHESIS | CHEMISTRY, ORGANIC | PD-CATALYZED SYNTHESIS | EXCESS N-BUTYLLITHIUM | REGIOSELECTIVE SYNTHESIS | MODULAR SYNTHESIS | SUBSTITUTED INDOLES | C-H
Journal Article
Chemical Communications : Chem Comm, ISSN 1359-7345, 01/2018, Volume 54, Issue 14, pp. 1676 - 1685
Recent advances in transition metal-catalyzed selective C–H functionalization of indoles have garnered tremendous attention. Great efforts have been devoted to... 
Regioselectivity | Indoles
Journal Article
Chemical Communications, ISSN 1359-7345, 2/2018, Volume 54, Issue 14, pp. 1676 - 1685
Recent advances in transition metal-catalyzed selective C-H functionalization of indoles have garnered tremendous attention. Great efforts have been devoted to... 
DUAL C-H | ROOM-TEMPERATURE | 2-SUBSTITUTED INDOLES | C-3 ARYLATION | DICTYODENDRINS F | SELECTIVE ARYLATION | N-PIVALOYLINDOLES | H BOND FUNCTIONALIZATION | CHEMISTRY, MULTIDISCIPLINARY | ORTHO-METALATION | CATALYZED DIRECT ARYLATION
Journal Article
Tetrahedron, ISSN 0040-4020, 2012, Volume 68, Issue 5, pp. 1393 - 1400
An impregnated copper on magnetite catalyst is a versatile system for different domino Sonogashira-cyclization processes between 2-iodophenol and different... 
C–C coupling | Heterogeneous catalysis | Palladium | Cyclization | Copper | Domino reaction | C-C coupling | 2-SUBSTITUTED INDOLES | LIGAND-FREE | ONE-POT SYNTHESIS | CHEMISTRY, ORGANIC | INTERNAL ALKYNES | CROSS-COUPLING REACTIONS | NANO-POWDER MAGNETITE | RECYCLABLE CATALYST | VINYL IODIDES | HETEROGENEOUS CATALYSTS | WATER | Furans | Magnetite
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 07/2016, Volume 81, Issue 13, pp. 5450 - 5463
Disubstituted benzo­[b]­furans were synthesized by ortho-selective Sonogashira coupling of dichlorophenols and terminal alkynes, followed by cyclization and... 
2-SUBSTITUTED INDOLES | COUPLING REACTIONS | 4-SUBSTITUTED INDOLES | COMBINATORIAL SYNTHESIS | INTRAMOLECULAR HYDROAMINATION | SONOGASHIRA REACTION | EFFICIENT SYNTHESIS | CHEMISTRY, ORGANIC | OLIGOARENE-TYPE PHOSPHINES | C-H ACTIVATION | GRIGNARD-REAGENTS
Journal Article
Organic Letters, ISSN 1523-7060, 07/2008, Volume 10, Issue 13, pp. 2617 - 2620
A new LDA-induced anionic N−C carbamoyl migration of 2-arylindoles (7) is reported. Treatment of N-carbamoylindoles 10 and 13, readily available by direct and... 
FUNCTIONALIZATION | 2-SUBSTITUTED INDOLES | METHODOLOGY | FRIES REARRANGEMENT | ESTERS | QUINOLINES | CHEMISTRY, ORGANIC | PYRIDINES | ACCESS | STRATEGIES | Metals - chemistry | Benzene - chemistry | Indoles - chemical synthesis | Models, Molecular | Molecular Structure | Anions - chemistry | Indoles - chemistry | Carbamates - chemistry
Journal Article
Chemistry – A European Journal, ISSN 0947-6539, 06/2018, Volume 24, Issue 31, pp. 7964 - 7969
Journal Article
Chemical Communications, ISSN 1359-7345, 07/2015, Volume 51, Issue 73, pp. 13898 - 13901
A simple, efficient and practical metal-free C-H sulfenylation process at the C2 position of non-protected indoles has been developed. 2-Thioindoles were... 
2-SUBSTITUTED INDOLES | 3-INDOLYL SULFIDES | ACID-CATALYZED ISOMERIZATION | TUBULIN POLYMERIZATION | CHLORIDES | INHIBITORS | CHEMISTRY, MULTIDISCIPLINARY | EFFICIENT SULFENYLATION | Indoles
Journal Article
Chemistry – An Asian Journal, ISSN 1861-4728, 05/2018, Volume 13, Issue 10, pp. 1327 - 1334
An asymmetric aza‐Friedel–Crafts alkylation reaction between indoles and indolenines that were derived in situ from 3‐indolinone‐2‐carboxylates has been... 
alkylation | indoles | asymmetric synthesis | Mannich reaction | synthetic methods | 2-SUBSTITUTED INDOLIN-3-ONES | ENANTIOSELECTIVE SYNTHESIS | (+/-)-TRIGONOLIIMINE C | CHEMISTRY, MULTIDISCIPLINARY | 2-MONOSUBSTITUTED INDOLIN-3-ONES | MANNICH REACTIONS | TRANSITION-METAL | C-SP3-H BOND ADJACENT | RECENT PROGRESS | CHIRAL BRONSTED ACID | N-BOC KETIMINES
Journal Article