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7-substituted indoles (35) 35
chemistry, organic (32) 32
indole (13) 13
derivatives (10) 10
indoles (10) 10
room-temperature (10) 10
chemistry (8) 8
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catalysis (7) 7
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activation (6) 6
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7-substituted indole (5) 5
bond activation (5) 5
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cyclization (5) 5
thallation (5) 5
2,3-disubstituted indoles (4) 4
alkaloids (4) 4
arenes (4) 4
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heterocyclic compounds (4) 4
indolines (4) 4
research (4) 4
2-substituted indoles (3) 3
alkenylation (3) 3
bond (3) 3
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chemistry, applied (3) 3
formyl group (3) 3
heck reaction (3) 3
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indol (3) 3
letter (3) 3
n-pivaloylindoles (3) 3
nitroarenes (3) 3
nonrearranged monoterpenoid unit (3) 3
regioselectivity (3) 3
rhodium (3) 3
substituted indoles (3) 3
sulfonyl azides (3) 3
tripeptide (3) 3
vinyl grignard-reagents (3) 3
3,4-differentially substituted indoles (2) 2
7-substituted 1,4-dihydro-4-oxo-1--1,8-naphthyridine-3-carboxylic acids (2) 2
7-substituted coumarins (2) 2
7-substituted indolines (2) 2
agents (2) 2
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clavicipitic acid (2) 2
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homogeneous catalysis (2) 2
indoles - chemistry (2) 2
initiated cyclizations (2) 2
isatin (2) 2
keton (2) 2
ketones (2) 2
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Organic and Biomolecular Chemistry, ISSN 1477-0520, 2016, Volume 14, Issue 21, pp. 4804 - 4808
Iridium(III)-catalyzed direct C7-sulfonamidation of indoles with sulfonyl azides is described. The developed method has good compatibility with diverse... 
ANTIVIRAL AGENTS | CHELATION-ASSISTANCE | DIRECT ARYLATION | SULFONYL AZIDES | 7-SUBSTITUTED INDOLES | C-H AMIDATION | CHEMISTRY, ORGANIC | BOND ACTIVATION | N-PIVALOYLINDOLES | CLAVICIPITIC ACID | NONREARRANGED MONOTERPENOID UNIT
Journal Article
Organic & biomolecular chemistry, ISSN 1477-0520, 06/2016, Volume 14, Issue 21, pp. 4804 - 4808
Iridium(iii)-catalyzed direct C7-sulfonamidation of indoles with sulfonyl azides is described. The developed method has good compatibility with diverse... 
Journal Article
ACS Catalysis, ISSN 2155-5435, 09/2017, Volume 7, Issue 9, pp. 5618 - 5627
The indole scaffold will continue to play a vital part in the future of drug discovery and agrochemical development. Because of this, the necessity for elegant... 
regioselectivity | heteroaromatics | indole | homogeneous catalysis | C-H functionalization | DIRECTING GROUP | ROOM-TEMPERATURE | 7-SUBSTITUTED INDOLES | NATURAL-PRODUCTS | BOND FUNCTIONALIZATIONS | CHEMISTRY, PHYSICAL | INTERNAL ALKYNES | MILD CONDITIONS | RUTHENIUM CATALYSIS | REGIOSELECTIVE SYNTHESIS | 2,3-DISUBSTITUTED INDOLES
Journal Article
Current Organic Chemistry, ISSN 1385-2728, 01/2005, Volume 9, Issue 2, pp. 163 - 178
Due to the potent biological activity exhibited by various indole derivatives, there is a continuous demand for novel synthetic procedures in this area. In... 
NITROARENES | METHODOLOGY | NITRO-COMPOUNDS | 7-SUBSTITUTED INDOLES | VINYL GRIGNARD-REAGENTS | CHEMISTRY, ORGANIC | SUBSTITUTED INDOLES | DERIVATIVES | GENERAL-METHOD | CONJUGATE ADDITION | ALKALOIDS
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 08/1996, Volume 61, Issue 17, pp. 5804 - 5812
Journal Article
Angewandte Chemie International Edition, ISSN 1433-7851, 01/2016, Volume 55, Issue 1, pp. 321 - 325
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 02/2015, Volume 80, Issue 3, pp. 1946 - 1951
Journal Article
Synthesis, ISSN 0039-7881, 10/2006, Volume 2006, Issue 20, pp. 3467 - 3477
Abstract Traditional strategies in indole chemistry do not allow high-yielding access to some substitution patterns such as 3,5,7-trisubstituted indoles. We... 
paper | Heck reaction | Palladium | Indoles | 2-vinylanilines | Larock's cyclisation | 7-SUBSTITUTED INDOLES | CHEMISTRY, ORGANIC | indoles | ARYL HALIDES | COUPLING REACTION | palladium | SUBSTITUTED INDOLES | 2,3-DISUBSTITUTED INDOLES | INTRAMOLECULAR HECK REACTION | CYCLIZATION | REGIOCONTROLLED SYNTHESIS | ALKALOIDS
Journal Article
Organic Letters, ISSN 1523-7060, 08/2003, Volume 5, Issue 16, pp. 2829 - 2832
Bartoli indole synthesis has been performed for the first time on solid supports. Starting from Merrifield resin, immobilization of five nitro benzoic acids... 
TRACELESS | PHASE SYNTHESIS | NITROARENES | 7-SUBSTITUTED INDOLES | CHEMISTRY, ORGANIC | RECEPTOR | 2,3-DISUBSTITUTED INDOLES | SUBSTITUTED INDOLES | ANTAGONISTS | DERIVATIVES | CYCLIZATION
Journal Article
Advanced Synthesis & Catalysis, ISSN 1615-4150, 02/2015, Volume 357, Issue 2‐3, pp. 594 - 600
Journal Article
Synlett, ISSN 0936-5214, 12/2005, Volume 2005, Issue 20, pp. 3071 - 3074
Abstract Traditional strategies in indole chemistry do not allow high yielding access to some substitution patterns such as 3,5,7-trisubstituted indoles. We... 
letter | Heck reaction | Anilines | Palladium | Hydroxybenzimidazole | Indoles | BASES | REAGENTS | 7-SUBSTITUTED INDOLES | CHEMISTRY, ORGANIC | anilines | indoles | ARYL HALIDES | CESIUM | CHEMISTRY | palladium | POTASSIUM | 2,3-DISUBSTITUTED INDOLES | hydroxybenzimidazole | DERIVATIVES
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 01/2016, Volume 81, Issue 2, pp. 396 - 403
The rhodium­(III)-catalyzed intermolecular C7-thiolation and selenation of indolines with disulfides and diselenides were developed. This protocol relies on... 
ALIPHATIC AMIDES | ROOM-TEMPERATURE | C(SP)-H BONDS | ACTIVATION | C-7 POSITION | 7-SUBSTITUTED INDOLES | CHEMISTRY, ORGANIC | OXIDATIVE ANNULATION | DIRECT THIOLATION | C-H BONDS | CATALYZED DIRECTED SULFENYLATION | Ruthenium | Chemical properties | Catalysis | Research | Indole
Journal Article
Synthesis, ISSN 0039-7881, 12/2007, Volume 2007, Issue 24, pp. 3851 - 3857
Abstract A new approach to the synthesis of cyclopenta[G]indole derivatives possessing structural features of natural alkaloids, such as trikentrins and... 
paper | Ring contraction | Cyclopenta[g]indoles | Thallium trinitrate | (+/-)-CIS-TRIKENTRIN-A | OXIDATION | ORGANIC-SYNTHESIS | cyclopenta[g]indoles | 7-SUBSTITUTED INDOLES | CHEMISTRY, ORGANIC | DIASTEREOSELECTIVE TOTAL-SYNTHESIS | NODULISPORIC-ACID | thallium trinitrate | ABSOLUTE STRUCTURES | REARRANGEMENT | THALLIUM | ring contraction | 1,2-DIHYDRONAPHTHALENES
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 10/2016, Volume 81, Issue 20, pp. 9878 - 9885
The rhodium­(III)-catalyzed direct C–H functionalization of various indolines with 1,4,2-dioxazol-5-ones as new amidating agents is described. This... 
CANCER-CELLS | AGENT | PALLADIUM | CATALYSIS | ACTIVATION | C-7 POSITION | MICROTUBULE | 7-SUBSTITUTED INDOLES | NATURAL-PRODUCTS | BOND FUNCTIONALIZATIONS | CHEMISTRY, ORGANIC
Journal Article
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, ISSN 1434-193X, 01/2017, Issue 4, pp. 840 - 845
An efficient method for the CF3-carbenoid C-7 functionalization of N-pyrimidylindolines has been developed. This protocol uses readily available methyl... 
Diazo compounds | ROOM-TEMPERATURE | Fluorine | 7-SUBSTITUTED INDOLES | NATURAL-PRODUCTS | CHEMISTRY, ORGANIC | Carbenoids | C-H functionalization | IN-SITU GENERATION | H BOND ACTIVATION | MEDICINAL CHEMISTRY | Nitrogen heterocycles | COUPLING REACTION | METHYL 3,3,3-TRIFLUORO-2-DIAZOPROPIONATE | Indoles | AMINO-ACID-DERIVATIVES
Journal Article
ADVANCED SYNTHESIS & CATALYSIS, ISSN 1615-4150, 04/2018, Volume 360, Issue 8, pp. 1644 - 1649
A Cu(I)-catalyzed regioselective cross-dehydrogenative coupling of indoline with a variety aryl and alkyl carboxylic acids is described. The divergent process... 
ROOM-TEMPERATURE | C-H BOND | C-7 POSITION | Indole | 7-SUBSTITUTED INDOLES | EXPEDIENT SYNTHESIS | CHEMISTRY, ORGANIC | CARBONYL-COMPOUNDS | DIRECT ACCESS | C-H functionalization | copper catalysis | acyloxylation | COUPLING REACTION | N-PIVALOYLINDOLES | CHEMISTRY, APPLIED | cross-dehydrogenative coupling | AROMATIC CARBOXYLIC-ACIDS
Journal Article
Tetrahedron, ISSN 0040-4020, 1999, Volume 55, Issue 30, pp. 9151 - 9162
Directed lithiation of 1-acylindole derivatives was investigated. It was discovered that a bulky 2,2-diethylbutanoyl (DEB) group could promote unusual C-7... 
SUBSTITUTION | PROTEIN-KINASE-C | LYNGBYATOXIN-A TELEOCIDIN-A-1 | ANALOGS | 7-SUBSTITUTED INDOLES | COMPLEXES | CHEMISTRY | INDOLINES | CHEMISTRY, ORGANIC | CONGENERS | ETODOLAC
Journal Article
Organic Letters, ISSN 1523-7060, 11/2014, Volume 16, Issue 22, pp. 6020 - 6023
An improved method for the dehydrogenative C–H/C–H cross-coupling at the C-7 position of indolines containing a urea as a directing group is reported. The new... 
FUNCTIONALIZATION | ROOM-TEMPERATURE | CATALYZED ORTHO-ARYLATION | 7-SUBSTITUTED INDOLES | DIRECT OLEFINATION | CHEMISTRY, ORGANIC | SODIUM PERSULFATE | BOND ACTIVATION | OXIDATIVE ARYLATION | PALLADIUM CATALYSIS | SIMPLE ARENES
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 2018, Volume 16, Issue 5, pp. 693 - 697
A rhodium(III)-catalyzed direct cross-coupling reaction of indolines with maleimides via C-H bond activation was developed. This protocol displays good... 
DIRECTING GROUP | FUNCTIONALIZATION | ANTICANCER ACTIVITY | C-7 POSITION | ALLYLIC CARBONATES | 7-SUBSTITUTED INDOLES | ALKYLATION | CHEMISTRY, ORGANIC | BOND | C-H ACTIVATION | (HETERO)ARENES
Journal Article
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