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Journal Article
Journal Article
PURINERGIC SIGNALLING, ISSN 1573-9538, 03/2013, Volume 9, Issue 1, pp. 91 - 100
The concept of functional selectivity offers great potential for the development of drugs that selectively activate a specific intracellular signaling pathway.... 
Biased signaling | Adenosine | ANALOGS | ARRESTIN-BIASED AGONISM | Beta-arrestin | HIGH-AFFINITY | HIGH-POTENCY | NEUROSCIENCES | 7-TRANSMEMBRANE RECEPTORS | A RECEPTOR | PROFILE | GTP gamma S | Functional selectivity | BIOLOGICAL EVALUATION | ANTAGONISTS | DERIVATIVES | Adenosine A receptor
Journal Article
Journal Article
MedChemComm, ISSN 2040-2503, 06/2015, Volume 6, Issue 6, pp. 991 - 1002
Increasing evidence points to the possibility of one or more secondary binding sites being involved in the interaction of catecholamines on their receptors.... 
BETA-2-ADRENERGIC RECEPTOR | CHEMISTRY, MEDICINAL | STRUCTURE-BASED DISCOVERY | STRUCTURAL BASIS | ARRESTIN-BIASED AGONISM | BIOCHEMISTRY & MOLECULAR BIOLOGY | BETA-1-ADRENERGIC RECEPTOR | PROTEIN-COUPLED RECEPTORS | ADRENERGIC-RECEPTOR | ALLOSTERIC MODULATION | BETA-ADRENERGIC RECEPTOR
Journal Article
Journal of Biomolecular Structure and Dynamics, ISSN 0739-1102, 08/2019, Volume 37, Issue 12, pp. 3206 - 3225
Journal Article
by Zhang, J and Liu, X and Wang, SQ and Liu, GY and Xu, WR and Cheng, XC and Wang, RL
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, ISSN 0739-1102, 2017, Volume 35, Issue 12, pp. 2665 - 2680
It has been reported previously that some angiotensin II receptor blockers not only antagonize angiotensin II type 1 receptor (AT(1)R), but also exert... 
AT RECEPTOR | telmisartan | IN-SILICO | BIOCHEMISTRY & MOLECULAR BIOLOGY | molecular dynamics | ARRESTIN-BIASED LIGAND | ADMET | HYPERTENSIVE PATIENTS | DIABETIC-PATIENTS | BIOPHYSICS | PPAR | STRUCTURAL BASIS | INSULIN-RESISTANCE | FUNCTIONAL SELECTIVITY | SP docking | PPAR-GAMMA AGONISTS | MOLECULAR-DYNAMICS SIMULATIONS | ATR
Journal Article
Journal of Pharmacological Sciences, ISSN 1347-8613, 2013, Volume 122, Issue 1, pp. 1 - 9
[Abstract]. β-Arrestin-biased agonists are a new class of drugs with promising therapeutic effects. The molecular mechanisms of β-arrestin-biased agonists are... 
Journal Article