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Accounts of Chemical Research, ISSN 0001-4842, 10/2016, Volume 49, Issue 10, pp. 2080 - 2090
The transition-metal-catalyzed asymmetric cyclopropanation of olefins with diazoacetates has become one of the most important methods for the synthesis of... 
STEREOSELECTIVE CYCLOPROPANATION | CYCLOPROPYLPHOSPHONATES | BELACTOSIN | INHIBITORS | ASYMMETRIC INTRAMOLECULAR CYCLOPROPANATION | DERIVATIVES | CHEMISTRY, MULTIDISCIPLINARY
Journal Article
Angewandte Chemie International Edition, ISSN 1433-7851, 12/2016, Volume 55, Issue 49, pp. 15406 - 15410
Journal Article
Chemistry Letters, ISSN 0366-7022, 6/2015, Volume 44, Issue 6, pp. 818 - 820
Highly stereoselective Reformatsky reaction and Pd-catalyzed arylation using 1-(alkoxycarbonyl)cyclopropylzinc bromide proceeded to give the trans-adduct as... 
REAGENT | HALIDES | REFORMATSKY-TYPE REACTION | ACID | SCOPE | ESTERS | EXPANSION | CATALYZED ALPHA-ARYLATION | MIYAURA COUPLING PROCESSES | BELACTOSIN | CHEMISTRY, MULTIDISCIPLINARY
Journal Article
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, ISSN 1433-7851, 06/2015, Volume 54, Issue 27, pp. 7810 - 7814
Broad-spectrum proteasome inhibitors are applied as anticancer drugs, whereas selective blockage of the immunoproteasome represents a promising therapeutic... 
20S PROTEASOME | inhibitors | immunoproteasome | lactones | COMPLEX | BELACTOSIN-C | BIOLOGICAL-ACTIVITY | MODE | CRYSTAL-STRUCTURES | CHEMISTRY, MULTIDISCIPLINARY | cytotoxicity | lead structures | Permeability | Lactones | Protease inhibitors
Journal Article
by Gu, XJ and Ma, ST
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY, ISSN 1871-5206, 2018, Volume 18, Issue 12, pp. 1656 - 1673
Background: The 26S proteasome is a proteolytic complex of multimeric protease, which operates at the executive end of the Ubiquitin-Proteasome System (UPS)... 
MULTIPLE-MYELOMA | CHEMISTRY, MEDICINAL | CRYSTAL-STRUCTURE | peptide inhibitors | SARs | NONPEPTIDIC BELACTOSIN DERIVATIVES | OPEN-LABEL | design strategy | inhibitory activity | 20S PROTEASOME | BORONIC ACIDS | 26S proteasome | ubiquitin-proteasome system | ONCOLOGY | PRECLINICAL MODELS | BIOLOGICAL EVALUATION | SELECTIVE INHIBITORS | CORE PARTICLE
Journal Article
The Journal of Organic Chemistry, ISSN 0022-3263, 07/2008, Volume 73, Issue 13, pp. 5198 - 5201
An enantioselective unified strategy for the syntheses of the oxylipin class of natural products was accomplished. Our strategy relies on three catalytic... 
BIOMIMETIC SYNTHESIS | OXYLIPINS | CLAVULARIA-VIRIDIS | BELACTOSIN-C | ACID | CONSTANOLACTONE-A | NEOHALICHOLACTONE | SULTAM DIRECTED ALDOL | CHEMISTRY, ORGANIC | STEREOSELECTIVE-SYNTHESIS | STRUCTURE REVISION | Chemical properties | Catalysis | Hydrogenation | Analysis | Propane
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 11/2013, Volume 54, Issue 48, pp. 6596 - 6598
Nitrocyclopropanation of amino-acid derived enones has led to a series of cyclopropyl peptidomimetics suitable for further elaboration to compounds with the... 
Weinreb amide | Nitrocyclopropanation | Cyclopropane | Peptidomimetic | SYSTEM | NITROCOMPOUNDS | DESIGN | REDUCTION | ACIDS | CHEMISTRY, ORGANIC | BELACTOSIN | GENERAL PROCEDURE | Tetrahedrons | Synthesis (chemistry) | Biological | Organic compounds
Journal Article
Organic Letters, ISSN 1523-7060, 05/2006, Volume 8, Issue 11, pp. 2261 - 2263
Dichloromethane serves as a novel electrophilic carbene equivalent which adds to an enamine double bond. The presence of other alkene moieties in the enamine... 
ALKENES | KETONES | METAL CARBENE COMPLEXES | CHEMISTRY, ORGANIC | METHYLENATION | OLEFINS | ALDEHYDES | AID | BELACTOSIN-A | DERIVATIVES | VINYL ETHERS
Journal Article
Journal Article
Australian Journal of Chemistry, ISSN 0004-9425, 2013, Volume 66, Issue 9, pp. 1105 - 1111
A concise synthesis of both E-isomers of 2S-amino-3-(2'-aminomethyl-cyclopropyl) propionic acid, new methano-L-lysines, is described. The synthetic route... 
ANTAGONIST | MUSHROOM | LIGANDS | ALLYLIC ALCOHOLS | BIOLOGICAL EVALUATION | CYCLOPROPANATION | ALPHA-AMINO-ACIDS | NATURAL OCCURRENCE | BELACTOSIN | CHEMISTRY, MULTIDISCIPLINARY | AMANITA-CASTANOPSIDIS-HONGO
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 08/2012, Volume 10, Issue 31, pp. 6363 - 6374
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 2010, Volume 51, Issue 50, pp. 6500 - 6502
Journal Article
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