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benzamidines - chemical synthesis (98) 98
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Journal of Organic Chemistry, ISSN 0022-3263, 11/2013, Volume 78, Issue 22, pp. 11342 - 11348
The first example of a copper-catalyzed cascade reaction of (2-aminophenyl)methanols with aldehydes using the combination of cerium nitrate hexahydrate and... 
SYSTEM | NITROARENES | DESIGN | 2-SUBSTITUTED QUINAZOLINES | BENZAMIDINES | BIOLOGICAL EVALUATION | CHEMISTRY, ORGANIC | AEROBIC OXIDATION | INHIBITORS | ARYLBORONIC ACIDS | WATER | Quinazolines - chemical synthesis | Molecular Structure | Copper - chemistry | Catalysis | Quinazolines - chemistry | Pyrimidines | Chemical properties | Research | Copper | Chemical synthesis
Journal Article
Organic Letters, ISSN 1523-7060, 06/2014, Volume 16, Issue 11, pp. 2888 - 2891
An iodine-catalyzed oxidative cross-coupling of C-H/N-H has been demonstrated. This simple and efficient approach constructed α-ketoimides in good to excellent... 
Iodine - chemistry | Oxidation-Reduction | Benzamidines - chemical synthesis | Ketones - chemistry | Hydrochloric Acid - chemistry | Molecular Structure | Catalysis | Benzamidines - chemistry
Journal Article
Journal of the American Chemical Society, ISSN 0002-7863, 10/2009, Volume 131, Issue 41, pp. 14699 - 14702
Journal Article
Chemistry - A European Journal, ISSN 0947-6539, 07/2012, Volume 18, Issue 29, pp. 8882 - 8885
Journal Article
Organic Letters, ISSN 1523-7060, 09/2010, Volume 12, Issue 17, pp. 3963 - 3965
Journal Article
Bioorganic & Medicinal Chemistry, ISSN 0968-0896, 05/2015, Volume 23, Issue 10, pp. 2328 - 2343
Hepatocyte growth factor activator (HGFA), matriptase and hepsin are all S1 trypsin-like serine endopeptidases. HGFA is a plasma protease while hepsin and... 
Cell-signaling | Structure-based drug design | Peptidomimetic | Hepsin | HGF | Receptor tyrosine kinase | Enzyme inhibitor | Therapeutic | MSP | Benzamidine | RON | Small-molecule | Serine protease | Matriptase | c-MET | HGFA | Cancer | Growth factor | SINGLE-CHAIN PRECURSOR | HEPATOCYTE GROWTH-FACTOR | RAY CRYSTAL-STRUCTURE | TRANSMEMBRANE SERINE-PROTEASE | PROSTATE-CANCER | MACROPHAGE-STIMULATING PROTEIN | C-MET INHIBITOR | NAFAMOSTAT MESILATE | CHEMISTRY, MEDICINAL | BIOCHEMISTRY & MOLECULAR BIOLOGY | CHEMISTRY, ORGANIC | FACTOR ACTIVATOR HGFA | SUNFLOWER TRYPSIN INHIBITOR-1 | Phenylalanine - analogs & derivatives | Benzamidines - chemical synthesis | Antineoplastic Agents - chemical synthesis | Humans | Neoplasm Proteins - antagonists & inhibitors | Structure-Activity Relationship | Urea - chemistry | Protease Inhibitors - pharmacology | Urea - analogs & derivatives | Drug Design | Antineoplastic Agents - pharmacology | Amidines - chemical synthesis | Catalytic Domain | Recombinant Proteins - chemistry | Neoplasm Proteins - chemistry | Serine Endopeptidases - chemistry | Enzyme Assays | Peptidomimetics - chemistry | Benzamidines - pharmacology | Arginine - chemistry | Guanidines - chemistry | High-Throughput Screening Assays | Phenylalanine - chemical synthesis | Piperazines - chemical synthesis | Molecular Docking Simulation | Protease Inhibitors - chemical synthesis | Kinetics | Chemical properties | Protease inhibitors | Proteases | Analysis
Journal Article
Journal Article
Journal Article
Russian Journal of Organic Chemistry, ISSN 1070-4280, 7/2019, Volume 55, Issue 7, pp. 1047 - 1052
Ten N(N′)-arylbenzamidines were synthesized in 60–77% yield by one-pot microwave-assisted reaction of the corresponding N-arylbenzamides with aniline or... 
lipoxygenase | Chemistry | α-glucosidase | reverse transcriptase | N -substituted benzamidines | acetylcholinesterase | Organic Chemistry | alpha-glucosidase | PEPTIDES | UREASE | N-substituted benzamidines | ANTIOXIDANT ACTIVITIES | DNA | CHEMISTRY, ORGANIC | UNUSUAL AMINO-ACIDS | DERIVATIVES | Ammonia | Powders | Enzyme inhibitors | Aniline | Hydrogen | DNA polymerases | Copper oxide | Cuprite
Journal Article
Bioorganic & Medicinal Chemistry, ISSN 0968-0896, 2011, Volume 19, Issue 7, pp. 2156 - 2167
Journal Article