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Tetrahedron, ISSN 0040-4020, 11/2012, Volume 68, Issue 44, pp. 9035 - 9044
A facile, efficient, and general synthetic method for a wide range of medicinally useful 2-carboxylate derivatives of acridinols, quinolinols, and... 
Regioselective | Silver-catalyzed | Diketoacid | Electrophilic cyclization | Enolates | VERSATILE ACCESS | TOPOISOMERASE-II | TANDEM SYNTHESIS | CHEMISTRY, ORGANIC | FUROQUINOLINE | IN-VITRO | HETEROCYCLES | INHIBITORS | EFFICIENT | ANTIMICROBIAL ACTIVITY | CYCLIZATION
Journal Article
Antiviral Research, ISSN 0166-3542, 10/2016, Volume 134, pp. 236 - 243
Journal Article
Bulletin of the Korean Chemical Society, ISSN 0253-2964, 07/2013, Volume 34, Issue 7, pp. 1953 - 1954
Journal Article
Chinese Journal of Chemistry, ISSN 1001-604X, 09/2004, Volume 22, Issue 9, pp. 978 - 983
In order to provide a facile and practical access to structurally diverse aryl beta-diketoacids, An improved and highly efficient oxalylation method was... 
Aryl β-diketoacid | Dimethyl oxalate | Oxalylation | Sodium tert-butoxide | Bis-diketoacid | HIV-1 integrase inhibitor | oxalylation | CELLS | DESIGN | REPLICATION | aryl beta-diketoacid | ACIDS | sodium tert-butoxide | dimethyl oxalate | DERIVATIVES | CHEMISTRY, MULTIDISCIPLINARY | bis-diketoacid
Journal Article
Journal Article
Journal Article
Current Topics in Medicinal Chemistry, ISSN 1568-0266, 07/2007, Volume 7, Issue 13, pp. 1251 - 1272
Replication of the human immunodeficiency virus (HIV) is dependent upon the enzyme HIV integrase (IN), one of three essential enzymes encoded in the viral... 
Integrase | 1,6-naphthyridine | Strand transfer | HIV | Diketoacid | AIDS | Diaryldiketone | STRAND-TRANSFER | CHEMISTRY, MEDICINAL | ACID | PROTEIN | STABLE COMPLEX | ACTIVE-SITE | diketoacid | RETROVIRAL DNA INTEGRATION | integrase | VIRAL REPLICATION | strand transfer | IN-VITRO | POTENT | diaryidiketone | IMMUNODEFICIENCY-VIRUS TYPE-1
Journal Article
Virologie, ISSN 1267-8694, 12/2007, Volume 11, pp. S163 - S173
Journal Article
Tetrahedron, ISSN 0040-4020, 2004, Volume 60, Issue 31, pp. 6479 - 6486
A simple and efficient oxalylation of aryl methyl ketones was accomplished with dimethyl oxalate in the presence of sodium methoxide. The unpreviously reported... 
Antiviral agents | Tautomerism | HIV integrase inhibitors | Diketoacids | tautomerism | CELLS | REPLICATION | diketoacids | antiviral agents | CHEMISTRY, ORGANIC | AGENTS | HIV-1 INTEGRASE INHIBITORS | DERIVATIVES
Journal Article
Journal Article
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