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British Journal of Pharmacology, ISSN 0007-1188, 02/1999, Volume 126, Issue 3, pp. 665 - 672
We have tested our prediction that AM630 is a CB2 cannabinoid receptor ligand and also investigated whether L759633 and L759656, are CB2 receptor agonists.... 
AM630 | CB2‐selective ligands | L759656 | CB2‐selective inverse agonist | [35S]‐GTPγS | CB2‐selective agonist | cyclic AMP | Cannabinoid CB1 and CB2 receptors | L759633 | Cannabinoid CB | selective agonist | receptors | Cyclic AMP | selective ligands | and CB | selective inverse agonist | S]-GTPγS | ANTAGONIST | cannabinoid CB1 and CB2 receptors | [S-35]-GTP gamma S | CB2-selective agonist | CB2-selective ligands | CB2-selective inverse agonist | PHARMACOLOGY | PHARMACOLOGY & PHARMACY | BINDING | BRAIN | Guanosine 5'-O-(3-Thiotriphosphate) - pharmacology | Cannabinoids - antagonists & inhibitors | Humans | Bornanes - pharmacology | Tritium | Benzoxazines | Receptors, Drug - agonists | Cyclohexanols - metabolism | Chromans - pharmacology | Indoles - pharmacology | Cyclohexanols - pharmacology | Radioligand Assay | Naphthalenes - metabolism | Cannabinoids - metabolism | Cyclic AMP - metabolism | CHO Cells | Pyrazoles - pharmacology | Cricetinae | Colforsin - pharmacology | Morpholines - pharmacology | Morpholines - metabolism | Pyrazoles - metabolism | Receptors, Drug - metabolism | Naphthalenes - pharmacology | Binding, Competitive - drug effects | Guanosine 5'-O-(3-Thiotriphosphate) - metabolism | Animals | Bornanes - metabolism | Receptors, Cannabinoid | Receptors, Drug - antagonists & inhibitors | Papers | [35S]-GTPγS
Journal Article
Journal Article
British Journal of Pharmacology, ISSN 0007-1188, 05/2019, Volume 176, Issue 10, pp. 1481 - 1491
Journal Article
Journal Article
ACS Medicinal Chemistry Letters, ISSN 1948-5875, 02/2018, Volume 9, Issue 2, pp. 120 - 124
Biaryl amides as new RORγt modulators were discovered. The crystal structure of biaryl amide agonist 6 in complex with RORγt ligand binding domain (LBD) was... 
CHEMISTRY, MEDICINAL | inverse agonist | NUCLEAR RECEPTORS | ROR gamma t | TARGETING TH17 CELLS | agonist | cocrystal structure | DISCOVERY | AUTOIMMUNE | POTENT | DISEASES | Th17 cell differentiation | MULTIPLE-SCLEROSIS | INTERLEUKIN-17 | DIFFERENTIATION | ANTAGONISTS | biaryl amides
Journal Article
Neurobiology of Disease, ISSN 0969-9961, 2007, Volume 30, Issue 1, pp. 74 - 83
Abstract Narcolepsy is characterized by excessive daytime sleepiness (EDS), cataplexy, direct onsets of rapid eye movement (REM) sleep from wakefulness (DREMs)... 
Neurology | Histamine | Sleep disorders | Somnolence | Wakefulness | receptor inverse agonist | Narcolepsy | Orexin
Journal Article
Journal Article
Journal Article
Journal Article
Science Signaling, ISSN 1945-0877, 10/2013, Volume 6, Issue 298, pp. ra93 - ra93
Journal Article
16.