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animals (3) 3
enzyme activation (3) 3
index medicus (3) 3
phosphorylation (3) 3
amino acid sequence (2) 2
ampk, amp-activated protein kinase (2) 2
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mapkap-k, mapk-activated protein kinase (2) 2
msk, mitogen- and stress-activated protein kinase (2) 2
research article (2) 2
rsk, p90 ribosomal s6 kinase (2) 2
3-phosphoinositide-dependent protein kinase 1 (1) 1
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camp and calcium responsive element binding protein (1) 1
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creb, cyclic amp response element binding protein (1) 1
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fgf-r, fibroblast-growth-factor receptor (1) 1
fkbp, fk506-binding protein (1) 1
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gak, cyclin g-associated kinase (1) 1
gsk3, glycogen synthase kinase 3 (1) 1
gst, glutathione (1) 1
gst, glutathione s-transferase (1) 1
gst, glutathione transferase (1) 1
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hipk, homeodomain-interacting protein kinase (1) 1
his6, hexahistidine (1) 1
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ikk, inhibitory κb kinase (1) 1
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Biochemical Journal, ISSN 0264-6021, 12/2007, Volume 408, Issue 3, pp. 297 - 315
The specificities of 65 compounds reported to be relatively specific inhibitors of protein kinases have been profiled against a panel of 70-80 protein kinases.... 
Drug discovery | Kinase profiling | Protein kinase | Anti-cancer drugs | Inhibitor specificity | RHO-ASSOCIATED KINASE | TUMOR PROGRESSION | FAMILY-MEMBERS | BIOCHEMISTRY & MOLECULAR BIOLOGY | CELL-PROLIFERATION | protein kinase | P38 MAP KINASE | CYCLIN-DEPENDENT KINASES | RECEPTOR TYROSINE KINASES | drug discovery | kinase profiling | SB 203580 | anti-cancer drugs | ISOFORMS IN-VITRO | P90 RSK | inhibitor specificity | Amino Acid Sequence | Cell Line | Phosphorylation | Recombinant Proteins - antagonists & inhibitors | Animals | Mitogen-Activated Protein Kinases - antagonists & inhibitors | Humans | Drug Design | Protein Kinase Inhibitors - pharmacology | Enzyme Activation | Mitogen-Activated Protein Kinases - metabolism | Spodoptera | Index Medicus | Yes1, Yamaguchi sarcoma viral oncogene homologue 1 | CSK, C-terminal Src kinase | Lck, lymphocyte cell-specific protein-tyrosine kinase | EGF, epidermal growth factor | FGF-R, fibroblast-growth-factor receptor | PAK, p21-activated protein kinase | PDK, 3-phosphoinositide-dependent protein kinase | PI3K, phosphatidylinositol (phosphoinositide) 3-kinase | NEK, NIMA (never in mitosis in Aspergillus nidulans)-related kinase | RSK, p90 ribosomal S6 kinase | HEK-293 cells, human embryonic kidney-293 cells | VEGF, vascular endothelial growth factor (vasoendothelial growth factor) | EF2K, elongation-factor-2 kinase | CK, casein kinase | PTEN, phosphatase and tensin homologue deleted on chromosome 10 | ERK, extracellular-signal-regulated kinase | ATM, ataxia telangiectasia mutated | SRPK, serine-arginine protein kinase | IL-1, interleukin 1 | MNK, MAPK-integrating protein kinase | ROCK, Rho-dependent protein kinase | CaMKK, CaMK kinase | GST, glutathione transferase | MKK1, MAPK kinase-1 (also called MEK1, MAPK or ERK kinase 1) | GAK, cyclin G-associated kinase | FMK, fluoromethylketone | MST, mammalian homologue Ste20-like kinase | PKA, cAMP-dependent protein kinase | FKBP, FK506-binding protein | PPAR, peroxisome-proliferator-activated receptor | IKK, inhibitory κB kinase | PH, pleckstrin homology | MBP, myelin basic protein | AICAR, aminoimidazole-4-carboxamide-1-β-D-ribofuranoside | MAPKAP-K, MAPK-activated protein kinase | Sf21, Spodoptera frugiperda (fall armyworm) 21 | MARK, microtubule-affinity-regulating kinase | PIM, provirus integration site for Moloney murine leukaemia virus | LPS, lipopolysaccharide | MSK, mitogen- and stress-activated protein kinase | MAPK, mitogen-activated protein kinase | MELK, maternal embryonic leucine-zipper kinase | His6, hexahistidine | CAK, cyclin-dependent kinase-activating kinase | Eph-A2, Ephrin A2 receptor | PLK, polo-like kinase | ATF2, activating transcription factor 2 | PKD, protein kinase D | Src, sarcoma kinase | AMPK, AMP-activated protein kinase | MMS, methyl methanesulfonate | CHK, checkpoint kinase | JNK, c-Jun N-terminal kinase | TORC1, mTOR (mammalian target of rapamycin)–raptor (regulatory associated protein of mTOR) complex | BRSK, brain-specific kinase | RIP2, receptor-interacting protein 2 | IGF-1, insulin-like growth factor-1 | S6K1, S6 kinase 1 | DYRK, dual-specificity tyrosine-phosphorylated and -regulated kinase | HIPK, homeodomain-interacting protein kinase | ZMP, aminoimidazole-4-carboxamide-1-β-D-ribofuranoside monophosphate | PRAK, p38-regulated activated kinase | PKC, protein kinase C | Src-I1, Src inhibitor 1 | TANK, TRAF (tumour-necrosis-factor-receptor-associated factor)-family-member-associated nuclear factor κB activator | NFAT, nuclear factor for activated T-cells | PHK, phosphorylase kinase | GSK3, glycogen synthase kinase 3 | PKB, protein kinase B (also called Akt) | CaMK, calmodulin-dependent kinase | CDK, cyclin-dependent protein kinase | NDRG, N-myc downstream-regulated gene | SmMLCK, smooth-muscle myosin light-chain kinase | TBK1, TANK-binding kinase 1 | PRK, protein kinase C-related kinase | SGK, serum- and glucocorticoid-induced kinase
Journal Article
Biochemical Journal, ISSN 0264-6021, 04/2005, Volume 387, Issue 2, pp. 507 - 517
MSK1 (mitogen- and stress-activated protein kinase) is a kinase activated in cells downstream of both the ERK1/2 (extracellular-signal-regulated kinase) and... 
MSK2 | Mitogen- and stress-activated protein kinase (MSK1) | 3-Phosphoinositide-dependent protein kinase 1 (PDK1) | P38 | Extracellular-signal-regulated kinase (ERK) | P90 ribosomal S6 kinase (RSK) | Amino Acid Sequence | Cell Line | Phosphorylation | Mutagenesis, Site-Directed | Humans | Molecular Sequence Data | Ribosomal Protein S6 Kinases, 90-kDa - chemistry | Ribosomal Protein S6 Kinases, 90-kDa - metabolism | Animals | Mitogen-Activated Protein Kinase 3 - metabolism | p38 Mitogen-Activated Protein Kinases - metabolism | Enzyme Activation | Mitogens | Mitogen-Activated Protein Kinase 1 - metabolism | Index Medicus | mitogen- and stress-activated protein kinase (MSK1) | 3-phosphoinositide-dependent protein kinase 1 (PDK1) | PDK1, 3-phosphoinositide-dependent protein kinase 1 | GST, glutathione S-transferase | HEK-293 cells, human embryonic kidney 293 cells | RSK, p90 ribosomal S6 kinase | extracellular-signal-regulated kinase (ERK) | ERK, extracellular-signal-regulated kinase | MALDI–TOF, matrix-assisted laser-desorption ionization–time of flight | PEI, polyethyleneimine | p38 | DMEM, Dulbecco's modified Eagle's medium | MAPKAP-K, MAPK-activated protein kinase | MEF, mouse embryonic fibroblast | PH domain, pleckstrin homology domain | MSK, mitogen- and stress-activated protein kinase | p90 ribosomal S6 kinase (RSK) | PIP3, phosphatidylinositol 3,4,5-trisphosphate | MAPK, mitogen-activated protein kinase | PKA, PKB, PKC and PKG, protein kinases A, B, C and G respectively | TFA, trifluoroacetic acid
Journal Article
FEBS Letters, ISSN 0014-5793, 1998, Volume 439, Issue 3, pp. 287 - 290
Journal Article
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