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British journal of pharmacology, ISSN 0007-1188, 10/2013, Volume 170, Issue 4, pp. 893 - 907
internalization | receptor signalling | cannabinoid receptor | desensitization | allosteric modulator | Life Sciences & Biomedicine | Pharmacology & Pharmacy | Science & Technology | Humans | Cannabinoid Receptor Agonists - pharmacology | Dose-Response Relationship, Drug | Cyclohexanols - metabolism | Transfection | Piperidines - pharmacology | HEK293 Cells | Cannabinoid Receptor Antagonists - pharmacology | Indoles - pharmacology | Cyclohexanols - pharmacology | Cyclic AMP - metabolism | Potassium Channels, Inwardly Rectifying - drug effects | Rats | Protein Transport | Receptor, Cannabinoid, CB1 - metabolism | Animals | Receptor, Cannabinoid, CB1 - genetics | Membrane Potentials | Signal Transduction - drug effects | Receptor, Cannabinoid, CB1 - drug effects | Cell Line, Tumor | Ligands | Mice | Phenylurea Compounds - pharmacology | Pyridines - pharmacology | Kinetics | Potassium Channels, Inwardly Rectifying - metabolism | Cyclohexanol | Urea | Chemical properties | Studies | Binding sites | Index Medicus | Research Papers
Journal Article
The Journal of pharmacology and experimental therapeutics, ISSN 0022-3565, 07/2013, Volume 346, Issue 1, pp. 2 - 10
Life Sciences & Biomedicine | Pharmacology & Pharmacy | Science & Technology | Dopamine Plasma Membrane Transport Proteins - metabolism | Allosteric Regulation | Humans | Dopamine Plasma Membrane Transport Proteins - chemistry | Brain - metabolism | Nerve Tissue Proteins - chemistry | Dopamine - secretion | Protein Isoforms - metabolism | Protein Isoforms - agonists | Protein Isoforms - chemistry | Membrane Transport Modulators - pharmacology | Neurons - secretion | Biological Transport - drug effects | Neurons - metabolism | Neurons - drug effects | Dopamine - metabolism | Nerve Tissue Proteins - antagonists & inhibitors | Dopamine Plasma Membrane Transport Proteins - agonists | Nerve Tissue Proteins - agonists | Brain - drug effects | Dopamine Plasma Membrane Transport Proteins - antagonists & inhibitors | Nerve Tissue Proteins - metabolism | Brain - secretion | Animals | Ligands | Protein Conformation | Protein Isoforms - antagonists & inhibitors
Journal Article
Advanced drug delivery reviews, ISSN 0169-409X, 2003, Volume 55, Issue 1, pp. 151 - 164
P-glycoprotein | Multidrug resistance (MDR) | Multidrug resistant protein (MRP) | Block copolymer | Blood–brain barrier | Blood-brain barrier | Life Sciences & Biomedicine | Pharmacology & Pharmacy | Science & Technology | Humans | ATP-Binding Cassette, Sub-Family B, Member 1 - metabolism | ATP-Binding Cassette, Sub-Family B, Member 1 - antagonists & inhibitors | Blood-Brain Barrier - drug effects | Membrane Transport Modulators | Drug Carriers | Brain - blood supply | Poloxamer - toxicity | Biological Transport, Active | Pharmaceutical Preparations - metabolism | Animals | Poloxamer - pharmacology | Endothelium, Vascular - metabolism | Drug-Related Side Effects and Adverse Reactions | Membrane Transport Proteins - antagonists & inhibitors | ATP-Binding Cassette Transporters - metabolism | Membrane Transport Proteins - metabolism | ATP-Binding Cassette Transporters - antagonists & inhibitors | Index Medicus
Journal Article
Trends in pharmacological sciences (Regular ed.), ISSN 0165-6147, 2011, Volume 32, Issue 12, pp. 726 - 733
Advanced Basic Science | Life Sciences & Biomedicine | Pharmacology & Pharmacy | Science & Technology | Allosteric Regulation - drug effects | Receptors, N-Methyl-D-Aspartate - antagonists & inhibitors | Membrane Transport Modulators - chemistry | Humans | Protein Subunits - agonists | Receptors, N-Methyl-D-Aspartate - metabolism | Protein Subunits - metabolism | Membrane Transport Modulators - metabolism | Animals | Protein Isoforms - metabolism | Protein Isoforms - agonists | Protein Isoforms - chemistry | Receptors, N-Methyl-D-Aspartate - chemistry | Membrane Transport Modulators - pharmacology | Receptors, N-Methyl-D-Aspartate - agonists | Membrane Transport Modulators - therapeutic use | Ligands | Protein Conformation | Protein Subunits - antagonists & inhibitors | Protein Subunits - chemistry | Binding Sites | Protein Isoforms - antagonists & inhibitors | Methyl aspartate | Nervous system diseases | Pharmacology | Index Medicus
Journal Article
Current medicinal chemistry, ISSN 0929-8673, 05/2008, Volume 15, Issue 11, pp. 1126 - 1146
BK channel blockers | BK channel openers | KCa1.1 | BK channels | Maxi-K channels | BK channel modulators | Pharmacology & Pharmacy | Biochemistry & Molecular Biology | Life Sciences & Biomedicine | Chemistry, Medicinal | Science & Technology | Membrane Transport Modulators - chemistry | Humans | Large-Conductance Calcium-Activated Potassium Channels - agonists | Potassium Channel Blockers - therapeutic use | Clinical Trials as Topic | Large-Conductance Calcium-Activated Potassium Channels - antagonists & inhibitors | Animals | Large-Conductance Calcium-Activated Potassium Channels - physiology | Membrane Transport Modulators - pharmacology | Membrane Transport Modulators - therapeutic use | Molecular Structure | Drug Evaluation, Preclinical | Potassium Channel Blockers - chemistry | Potassium Channel Blockers - pharmacology
Journal Article
Pflügers Archiv, ISSN 0031-6768, 7/2015, Volume 467, Issue 7, pp. 1417 - 1430
Biomedicine | Ca 2+ activated Cl − channels (CaCCs) | Human Physiology | Bestrophin-1 | Patch clamp | Inhibitor | TMEM16A | CHO cells | Life Sciences & Biomedicine | Physiology | Science & Technology | Anoctamin-1 | Cricetinae | Flufenamic Acid - pharmacology | Chloride Channels - antagonists & inhibitors | Cricetulus | 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid - pharmacology | Humans | Nitrobenzoates - pharmacology | Neoplasm Proteins - antagonists & inhibitors | Neoplasm Proteins - metabolism | Chloride Channels - metabolism | Animals | Bestrophins | Eye Proteins - metabolism | Tannins - pharmacology | Membrane Transport Modulators - pharmacology | Niflumic Acid - pharmacology | Eye Proteins - antagonists & inhibitors | CHO Cells | Index Medicus
Journal Article
Journal of medicinal chemistry, ISSN 0022-2623, 08/2017, Volume 60, Issue 16, pp. 7199 - 7205
Pyridines - chemistry | Humans | Imidazoles - chemistry | Male | Structure-Activity Relationship | ATP-Binding Cassette Transporters - genetics | Membrane Transport Proteins - genetics | HEK293 Cells | Imidazoles - chemical synthesis | Imidazoles - metabolism | Drug Stability | Pyridines - chemical synthesis | PPAR alpha - genetics | Imidazoles - pharmacology | Receptors, Cytoplasmic and Nuclear - genetics | Rats, Sprague-Dawley | Hep G2 Cells | Cholesterol 7-alpha-Hydroxylase - genetics | Animals | Pyridines - metabolism | Sterol Regulatory Element Binding Protein 1 - genetics | Zolpidem | Molecular Docking Simulation | Pyridines - pharmacology | HeLa Cells | ATP Binding Cassette Transporter, Subfamily B, Member 11 | Receptors, Cytoplasmic and Nuclear - metabolism | Index Medicus
Journal Article
Current topics in medicinal chemistry, ISSN 1568-0266, 07/2016, Volume 16, Issue 16, pp. 1764 - 1791
Atrial and Ventricular arrhythmia | Atrial fibrillation | Ivabradine | Drug design | Hyperpolarization-activated current | Selectivity | HCN channels | Parkinson’s disease | Pharmacology & Pharmacy | Life Sciences & Biomedicine | Chemistry, Medicinal | Science & Technology | Membrane Transport Modulators - chemistry | Animals | Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels - metabolism | Humans | Membrane Transport Modulators - pharmacology | Drug Design | Molecular Structure | Membrane Transport Modulators - chemical synthesis | Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels - antagonists & inhibitors
Journal Article