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1. Full Text Efficient solid-phase chemical synthesis of 5′-triphosphates of DNA, RNA, and their analogues
by Zlatev, Ivan and Lavergne, Thomas and Debart, Françoise and Vasseur, Jean-Jacques and Manoharan, Muthiah and Morvan, François
Organic Letters, ISSN 1523-7060, 05/2010, Volume 12, Issue 10, pp. 2190 - 2193
A robust, reproducible, and scalable method for the solid-phase synthesis of 5'-triphosphates of DNA, RNA, and their chemically modified analogues using... 
CHEMISTRY, ORGANIC | SUPPORT | RIG-I | PANHANDLE | Organophosphonates - chemical synthesis | DNA - chemistry | Nucleic Acid Conformation | RNA - chemistry | Organophosphonates - chemistry | Solid Phase Extraction
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2. Full Text Synthesis of nucleoside phosphate and phosphonate prodrugs
by Pradere, Ugo and Garnier-Amblard, Ethel C and Coats, Steven J and Amblard, Franck and Schinazi, Raymond F
Chemical Reviews, ISSN 0009-2665, 2014, Volume 114, Issue 18, pp. 9154 - 9218
REPLICATION IN-VITRO | TOXIC LIPONUCLEOTIDE ANALOGS | HEPATITIS-C VIRUS | ANTI-HIV ACTIVITY | ACYCLOVIR DIPHOSPHATE DIMYRISTOYLGLYCEROL | LIPOPHILIC NUCLEOTIDE PRODRUGS | POSSIBLE ANTIVIRAL AGENTS | PRELIMINARY BIOLOGICAL EVALUATION | PHOSPHORAMIDATE PROTIDE TECHNOLOGY | CHEMISTRY, MULTIDISCIPLINARY | ARYL PHOSPHOTRIESTER DERIVATIVES | Prodrugs - chemical synthesis | Organophosphonates - chemical synthesis | Nucleosides - chemistry | Nucleosides - chemical synthesis | Phosphates - chemistry | Nucleosides | Chemical properties | Research | Phosphonates | Review
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3. Full Text Synthesis of Side-Chain Modified Polypeptides
by Deming, Timothy J
Chemical Reviews, ISSN 0009-2665, 2016, Volume 116, Issue 3, pp. 786 - 808
ACID-N-CARBOXYANHYDRIDES | POLY-L-LYSINE | CELL-PENETRATING PROPERTIES | DRUG-DELIVERY | ALPHA-AMINO-ACIDS | L-METHIONINE | RING-OPENING POLYMERIZATION | L-GLUTAMATE DERIVATIVES | CARBOBENZOXYMETHYL-L-CYSTEINE | WATER-SOLUBLE POLYPEPTIDES | CHEMISTRY, MULTIDISCIPLINARY | Peptides - chemical synthesis | Peptides - chemistry | Organophosphonates - chemistry | Phosphates - chemistry | Sulfhydryl Compounds - chemistry | Cysteine - chemistry | Cycloaddition Reaction | Alkylation | Esterification | Usage | Polypeptides | Chemical properties | Research | Biomimetics | Chemical synthesis
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4. Full Text Synthesis of β-aminophosphonates and -phosphinates
by Palacios, Francisco and Alonso, Concepción and de los Santos, Jesús M
Chemical Reviews, ISSN 0009-2665, 03/2005, Volume 105, Issue 3, pp. 899 - 931
P-C BOND | B RECEPTOR ANTAGONISTS | CATALYTIC ASYMMETRIC AMINOHYDROXYLATION | STATE ANALOG INHIBITORS | RING-OPENING REACTIONS | EFFICIENT SYNTHESIS | ORGANIC PHOSPHORUS-COMPOUNDS | ALPHA-HYDROXY PHOSPHONATES | ORGANOPHOSPHORUS COMPOUNDS | ASPARTIC-ACID DERIVATIVES | CHEMISTRY, MULTIDISCIPLINARY | Amines - chemistry | Organophosphorus Compounds - chemical synthesis | Models, Chemical | Oxidation-Reduction | Carbon - chemistry | Organophosphonates - chemical synthesis | Organophosphonates - pharmacology | Heterocyclic Compounds - chemistry | Nitrogen - chemistry | Phosphinic Acids - pharmacology | Imines - chemistry | Organophosphorus Compounds - pharmacology | Phosphinic Acids - chemical synthesis | Amino acids | Phosphorus compounds | Chemical properties | Chemical synthesis
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5. Full Text Silver-catalyzed synthesis of 3-phosphorated coumarins via radical cyclization of alkynoates and dialkyl H -phosphonates
by Mi, Xia and Wang, Chenyang and Huang, Mengmeng and Zhang, Jianye and Wu, Yusheng and Wu, Yangjie
Organic Letters, ISSN 1523-7060, 06/2014, Volume 16, Issue 12, pp. 3356 - 3359
Ag2CO3-catalyzed difunctionalization of alkynes via a radical phosphonation and C-H functionalization tandem process was developed to synthesize various... 
REGIOSELECTIVE PHOSPHONATION | FUNCTIONALIZATION | PHOSPHORUS-CENTERED RADICALS | DIENES | P BOND FORMATION | PHOSPHONYLATION | C-P | CHEMISTRY, ORGANIC | PHOSPHITES | ALKYNES | DERIVATIVES | Organophosphonates - chemical synthesis | Cyclization | Stereoisomerism | Coumarins - chemical synthesis | Organophosphonates - chemistry | Carbonates - chemistry | Coumarins - chemistry | Alkynes - chemistry | Molecular Structure | Catalysis | Silver Compounds - chemistry
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6. Full Text Fluorinated phosphonates: Synthesis and biomedical application
by Romanenko, Vadim D and Kukhar, Valery P
Chemical Reviews, ISSN 0009-2665, 09/2006, Volume 106, Issue 9, pp. 3868 - 3935
CARBOHYDRATE DIFLUOROMETHYLENE-PHOSPHONATES | PURINE-NUCLEOSIDE PHOSPHORYLASE | BETA-KETO PHOSPHONATES | WADSWORTH-EMMONS REACTION | ALPHA-AMINO PHOSPHONATES | SOLID-PHASE SYNTHESIS | MULTISUBSTRATE ANALOG INHIBITORS | HIV-1 REVERSE-TRANSCRIPTASE | CHEMISTRY, MULTIDISCIPLINARY | PROTEIN-TYROSINE-PHOSPHATASE | ALPHA,ALPHA-DIFLUORO FUNCTIONALIZED PHOSPHONATES | Antiviral Agents - pharmacology | Stereoisomerism | Antibodies - chemistry | Antineoplastic Agents - chemical synthesis | Enzyme Inhibitors - pharmacology | Hydrocarbons, Fluorinated - chemistry | Antineoplastic Agents - chemistry | Enzyme Inhibitors - chemical synthesis | Platelet Aggregation Inhibitors - chemical synthesis | Organophosphonates - chemical synthesis | Organophosphonates - pharmacology | Antiviral Agents - chemistry | Enzyme Inhibitors - chemistry | Organophosphonates - chemistry | Platelet Aggregation Inhibitors - chemistry | Antiviral Agents - chemical synthesis | Platelet Aggregation Inhibitors - pharmacology | Antineoplastic Agents - pharmacology | Molecular Structure | Catalysis | Atomic properties | Chemical properties | Fluorine | Phosphonates
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7. Aminophosphonic acids and derivatives. Synthesis and biological applications
by Orsini, F and Sello, G and Sisti, M
Current Medicinal Chemistry, ISSN 0929-8673, 2010, Volume 17, Issue 3, pp. 264 - 289
In recent years, phosphonic acids and their derivatives have received increasing attention as analogues of a series of naturally occurring phosphates and as... 
Aminophosphonates | Synthesis | Asymmetric synthesis | Aminophosphonic acids | Biological activity | CHEMISTRY, MEDICINAL | KABACHNIK-FIELDS REACTION | SOLVENT-FREE CONDITIONS | ONE-POT SYNTHESIS | BIOCHEMISTRY & MOLECULAR BIOLOGY | METABOTROPIC GLUTAMATE RECEPTORS | CATALYZED ENANTIOSELECTIVE HYDROPHOSPHONYLATION | DIPEPTIDYL PEPTIDASE IV | MATRIX-METALLOPROTEINASE INHIBITORS | PHARMACOLOGY & PHARMACY | ALPHA-AMINO-PHOSPHONATES | MICROWAVE-ASSISTED SYNTHESIS | TRANSITION-STATE ANALOG | Antiviral Agents - pharmacology | Stereoisomerism | Antineoplastic Agents - chemical synthesis | Humans | Enzyme Inhibitors - pharmacology | Enzyme Inhibitors - chemical synthesis | Anti-Bacterial Agents - chemical synthesis | Organophosphonates - chemical synthesis | Organophosphonates - pharmacology | Animals | Antiviral Agents - chemical synthesis | Anti-Bacterial Agents - pharmacology | Antineoplastic Agents - pharmacology
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8. Full Text Palladium‐Catalyzed Difluoroalkylation of Aryl Boronic Acids: A New Method for the Synthesis of Aryldifluoromethylated Phosphonates and Carboxylic Acid Derivatives
by Feng, Zhang and Min, Qiao‐Qiao and Xiao, Yu‐Lan and Zhang, Bo and Zhang, Xingang
Angewandte Chemie International Edition, ISSN 1433-7851, 02/2014, Volume 53, Issue 6, pp. 1669 - 1673
The palladium‐catalyzed difluoroalkylation of aryl boronic acids with bromodifluoromethylphosphonate, bromodifluoroacetate, and further derivatives has been... 
difluoroalkylation | palladium | aryl boronic acids | cross‐coupling | fluorine | cross-coupling | HALIDES | COPPER-MEDIATED DIFLUOROMETHYLATION | FLUOROALKYLATION | BOND FORMATION | REDUCTIVE ELIMINATION | CHEMISTRY, MULTIDISCIPLINARY | PROTEIN-TYROSINE | CROSS-COUPLING REACTIONS | FACILE | Electron Transport | Carboxylic Acids - chemistry | Organophosphonates - chemistry | Boronic Acids - chemistry | Catalysis | Palladium - chemistry | Boronic Acids - chemical synthesis | Fluorine - chemistry | Electrons | Palladium | Fluorides | Analysis | Methods | Phosphonates | Acids | Synthesis | Pathways | Catalysts | Aromatic compounds | Derivatives | Carboxylic acids | Single electrons
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9. Full Text Enantioselective organocatalytic conjugate addition of aldehydes to vinyl sulfones and vinyl phosphonates as challenging michael acceptors
by Sulzer-Mossé, Sarah and Alexakis, Alexandre and Mareda, Jiri and Bollot, Guillaume and Bernardinelli, Gerald and Filinchuk, Yaroslav
Chemistry - A European Journal, ISSN 0947-6539, 03/2009, Volume 15, Issue 13, pp. 3204 - 3220
Chiral amines with a pyrrolidine framework catalyze the enantioselective conjugate addition of a broad range of aldehydes to various vinyl sulfones and vinyl... 
Michael addition | Amines | Asymmetric synthesis | Aldehydes | Organocatalysis | ORGANIC-SYNTHESIS | ASYMMETRIC-SYNTHESIS | amines | QUATERNARY CARBON CENTERS | CHEMISTRY, MULTIDISCIPLINARY | CHIRAL IMINES | organocatalysis | aldehydes | asymmetric synthesis | NATURAL-PRODUCT SYNTHESIS | CATALYZED REDUCTIVE DESULFONYLATION | C-C | STEREOSELECTIVE-SYNTHESIS | ALPHA,BETA-UNSATURATED SULFONES | NITRO-OLEFINS | Amines - chemistry | Vinyl Compounds - chemical synthesis | Vinyl Compounds - chemistry | Models, Chemical | Aldehydes - chemical synthesis | Stereoisomerism | Pyrrolidines - chemistry | Organophosphonates - chemical synthesis | Combinatorial Chemistry Techniques | Sulfones - chemistry | Organophosphonates - chemistry | Molecular Structure | Catalysis | Aldehydes - chemistry | Sulfones - chemical synthesis
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10. Full Text Synthesis and applications of masked oxo-sulfinamides in asymmetric synthesis
by Edupuganti, Ramakrishna and Davis, Franklin A
ORGANIC & BIOMOLECULAR CHEMISTRY, ISSN 1477-0520, 7/2012, Volume 1, Issue 26, pp. 521 - 531
This short perspective reports on the synthesis and applications of a class of chiral amino carbonyl compounds, masked oxo-sulfinamides where the amine is... 
AMINO CARBONYL-COMPOUNDS | ORGANIC-SYNTHESIS | ACID-DERIVATIVES | SULFUR-NITROGEN | FORMAL SYNTHESIS | ENANTIOSPECIFIC SYNTHESIS | TERT-BUTANESULFINAMIDE | CHEMISTRY, ORGANIC | ANTI-1,3-AMINO ALCOHOLS | N-SULFINYL IMINES | COCAINE C-1 ANALOGS | Amines - chemistry | Amides - chemical synthesis | Amino Acids - chemistry | Heterocyclic Compounds - chemical synthesis | Pipecolic Acids - chemical synthesis | Proline - chemical synthesis | Amino Acids - chemical synthesis | Chemistry Techniques, Synthetic - methods | Organophosphonates - chemical synthesis | Heterocyclic Compounds - chemistry | Imines - chemistry | Imines - chemical synthesis | Amino Alcohols - chemistry | Tropanes - chemistry | Amino Alcohols - chemical synthesis | Tropanes - chemical synthesis | Amines - chemical synthesis | Cocaine - analogs & derivatives | Pyrrolidines - chemistry | beta-Lactams - chemistry | Proline - chemistry | Sulfonium Compounds - chemical synthesis | Pyrrolidines - chemical synthesis | Sulfonium Compounds - chemistry | Organophosphonates - chemistry | beta-Lactams - chemical synthesis | Amides - chemistry | Cocaine - chemical synthesis | Pipecolic Acids - chemistry
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11. Full Text Direct phosphonylation of aromatic azaheterocycles
by Van Der Jeught, Sarah and Stevens, Christian V
Chemical Reviews, ISSN 0009-2665, 06/2009, Volume 109, Issue 6, pp. 2672 - 2702
HETEROAROMATIC NUCLEOPHILIC-SUBSTITUTION | PALLADIUM-CATALYZED SYNTHESIS | MICHAELIS-ARBUZOV-REACTION | CONTAINING HETEROCYCLIC-COMPOUNDS | WITTIG-HORNER REACTION | FREE-RADICAL PHOSPHONATION | MONOMERIC METHYL METAPHOSPHATE | CHEMISTRY, MULTIDISCIPLINARY | REISSERT TYPES REACTION | TRIALKYL PHOSPHITES | PHOSPHORUS-CARBON BOND | Agrochemicals - chemical synthesis | Organophosphonates - chemical synthesis | Heterocyclic Compounds - chemistry | Aza Compounds - chemical synthesis | Organophosphonates - chemistry | Aza Compounds - chemistry | Heterocyclic Compounds - chemical synthesis | Agrochemicals - chemistry | Chemistry, Pharmaceutical
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12. Full Text Catalytic Aldol-Cyclization Cascade of 3-Isothiocyanato Oxindoles with α-Ketophosphonates for the Enantioselective Synthesis of β-Amino-α-hydroxyphosphonates
by Kayal, Satavisha and Mukherjee, Santanu
Organic Letters, ISSN 1523-7060, 11/2015, Volume 17, Issue 21, pp. 5508 - 5511
A cascade aldol cyclization reaction between 3-isothiocyanato oxindoles and alpha-ketophosphonates has been developed for the synthesis of... 
THIOCARBAMATE CATALYSTS | ISOTHIOCYANATO OXINDOLES | ASYMMETRIC-SYNTHESIS | PHOSPHONIC ACID-DERIVATIVES | CHEMISTRY, ORGANIC | CINCHONA ORGANOCATALYSTS | ORGANOPHOSPHORUS COMPOUNDS | POLYCYCLIC SPIROOXINDOLES | HIGHLY EFFICIENT | MICHAEL ADDITION | BIFUNCTIONAL ORGANOCATALYSTS | Stereoisomerism | Indoles - chemical synthesis | Thiourea - chemistry | Quinine - chemistry | Organophosphonates - chemical synthesis | Cyclization | Isothiocyanates - chemistry | Spiro Compounds - chemical synthesis | Organophosphonates - chemistry | Molecular Structure | Catalysis | Indoles - chemistry | Spiro Compounds - chemistry | Aldehydes - chemistry
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13. Full Text Structure-guided design, synthesis, and evaluation of guanine-derived inhibitors of the eIF4E mRNA-cap interaction
by Chen, Xiaoqi and Kopecky, David J and Mihalic, Jeff and Jeffries, Shawn and Min, Xiaoshan and Heath, Julie and Deignan, Jeff and Lai, Sujen and Fu, Zice and Guimaraes, Cristiano and Shen, Shanling and Li, Shyun and Johnstone, Sheree and Thibault, Stephen and Xu, Haoda and Cardozo, Mario and Shen, Wang and Walker, Nigel and Kayser, Frank and Wang, Zhulun
Journal of Medicinal Chemistry, ISSN 0022-2623, 04/2012, Volume 55, Issue 8, pp. 3837 - 3851
The eukaryotic initiation factor 4E (eIF4E) plays a central role in the initiation of gene translation and subsequent protein synthesis by binding the 5'... 
TRANSPORT | CHEMISTRY, MEDICINAL | CYCLIN D1 | ANALOGS | DEPENDENT TRANSLATION | INITIATION-FACTOR 4E | TRANSLATION INITIATION | EUKARYOTIC TRANSLATION | BINDING PROTEIN | CANCER | EXPRESSION | Guanosine Monophosphate - pharmacology | Rabbits | Guanine - analogs & derivatives | Humans | Eukaryotic Initiation Factor-4E - metabolism | Models, Molecular | Crystallography, X-Ray | Structure-Activity Relationship | RNA Caps - metabolism | Reticulocytes - metabolism | Organophosphonates - chemical synthesis | Eukaryotic Initiation Factor-4E - chemistry | Organophosphonates - pharmacology | Animals | Reticulocytes - drug effects | Guanine - pharmacology | Drug Design | Guanosine Monophosphate - analogs & derivatives | Inhibitory Concentration 50 | RNA Caps - chemistry | Protein Biosynthesis - drug effects | Phosphorous Acids | Guanosine Monophosphate - chemical synthesis | Guanine - chemical synthesis
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14. Full Text Rhodium carbene routes to oxazoles and thiazoles. Catalyst effects in the synthesis of oxazole and thiazole carboxylates, phosphonates, and sulfones
by Shi, Baolu and Blake, Alexander J and Lewis, William and Campbell, Ian B and Judkins, Brian D and Moody, Christopher J
Journal of Organic Chemistry, ISSN 0022-3263, 01/2010, Volume 75, Issue 1, pp. 152 - 161
Dirhodium tetraacetate catalyzed reaction of alpha-diazo-beta-keto-carboxylates and -phosphonates with arenecarboxamides gives 2-aryloxazole-4-carboxylates and... 
DIAZO ROUTE | BIS-OXAZOLE | DIAZONAMIDE-A | FRAGMENT | CHEMISTRY, ORGANIC | ALPHA-AMINO-ACID | FUNCTIONALIZED OXAZOLES | PEPTIDE MIMETICS | BETA-KETO-ESTERS | N-H INSERTION | THIOPEPTIDE ANTIBIOTICS | Magnetic Resonance Spectroscopy | Methane - analogs & derivatives | Stereoisomerism | Carboxylic Acids - chemical synthesis | Structure-Activity Relationship | Oxazoles - chemistry | Organophosphonates - chemical synthesis | Oxazoles - chemical synthesis | Thiazoles - chemical synthesis | Sulfones - chemistry | Carboxylic Acids - chemistry | Organophosphonates - chemistry | Methane - chemistry | Thiazoles - chemistry | Molecular Structure | Catalysis | Rhodium - chemistry | Sulfones - chemical synthesis | Oxazoles | Rhodium | Phosphonates | Chemical properties | Structure | Carbenes | Sulfones
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15. Full Text Copper-catalyzed aerobic oxidative coupling of terminal alkynes with H-phosphonates leading to alkynylphosphonates
by Gao, Yuxing and Wang, Gang and Chen, Lu and Xu, Pengxiang and Zhao, Yufen and Zhou, Yongbo and Han, Li-Biao
Journal of the American Chemical Society, ISSN 0002-7863, 06/2009, Volume 131, Issue 23, pp. 7956 - 7957
Copper catalyzed the aerobic oxidative coupling of terminal alkynes with H-phosphonates to afford alkynylphosphonates in high yields. 
CARBON BOND FORMATION | ANALOG | ONE-POT SYNTHESIS | CHEMISTRY, MULTIDISCIPLINARY | BIARYLS | Organophosphonates - chemical synthesis | Alkynes - chemical synthesis | Aerobiosis | Copper - chemistry | Oxidation-Reduction | Organophosphonates - chemistry | Alkynes - chemistry | Catalysis | Oxidation-reduction reaction | Chemical properties | Copper | Analysis | Phosphonates
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16. Full Text Discovery of a series of phosphonic acid-containing thiazoles and orally bioavailable diamide prodrugs that lower glucose in diabetic animals through inhibition of fructose-1,6-bisphosphatase
by Dang, Qun and Liu, Yan and Cashion, Daniel K and Kasibhatla, Srinivas Rao and Jiang, Tao and Taplin, Frank and Jacintho, Jason D and Li, Haiqing and Sun, Zhili and Fan, Yi and Dare, Jay and Tian, Feng and Li, Wenyu and Gibson, Tony and Lemus, Robert and Van Poelje, Paul D and Potter, Scott C and Erion, Mark D
Journal of Medicinal Chemistry, ISSN 0022-2623, 01/2011, Volume 54, Issue 1, pp. 153 - 165
Oral delivery of previously disclosed purine and benzimidazole fructose-1,6 bisphosphatase (FBPase) inhibitors via prodrugs failed, which was likely due to... 
FRUCTOSE 1,6-BISPHOSPHATASE | DESIGN | POTENT | CHEMISTRY, MEDICINAL | HYPERGLYCEMIA | OXAZOLES | RATS | CS-917 | AMP MIMICS | DERIVATIVES | Diabetes Mellitus, Experimental - drug therapy | Amides - chemical synthesis | Humans | Biological Availability | Male | Structure-Activity Relationship | Blood Proteins - metabolism | Thiazoles - pharmacokinetics | Diabetes Mellitus, Experimental - blood | Alanine - analogs & derivatives | Organophosphonates - chemical synthesis | Amides - pharmacokinetics | Alanine - pharmacology | Amides - pharmacology | Hypoglycemic Agents - pharmacokinetics | Alanine - pharmacokinetics | Administration, Oral | Rats | Rats, Sprague-Dawley | Hypoglycemic Agents - pharmacology | Organophosphonates - pharmacokinetics | Diabetes Mellitus, Type 2 - blood | Organophosphonates - pharmacology | Animals | Prodrugs - pharmacokinetics | Thiazoles - chemical synthesis | Hypoglycemic Agents - chemical synthesis | Alanine - chemical synthesis | Prodrugs - chemical synthesis | Protein Binding | Fructose-Bisphosphatase - antagonists & inhibitors | Mice | Thiazoles - pharmacology | Diabetes Mellitus, Type 2 - drug therapy | Prodrugs - pharmacology
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17. Full Text The synthesis of tenofovir and its analogues via asymmetric transfer hydrogenation
by Zhang, Qian and Ma, Bai-Wei and Wang, Qian-Qian and Wang, Xing-Xing and Hu, Xia and Xie, Ming-Sheng and Qu, Gui-Rong and Guo, Hai-Ming
Organic Letters, ISSN 1523-7060, 04/2014, Volume 16, Issue 7, pp. 2014 - 2017
A series of tenofovir analogues with potential antiviral and immunobiologically active compounds were synthesized through an asymmetric transfer hydrogenation... 
IN-VITRO | N-6-SUBSTITUTED ADENINES | AROMATIC KETONES | KINETIC RESOLUTION | COUPLING REACTION | CHEMISTRY, ORGANIC | RUTHENIUM(II) COMPLEX | PYRIMIDINE-BASES | ENANTIOMERIC N-(2-PHOSPHONOMETHOXYPROPYL) DERIVATIVES | HUMAN-IMMUNODEFICIENCY-VIRUS | ACYCLIC NUCLEOSIDE PHOSPHONATES | Antiviral Agents - pharmacology | Adenine - analogs & derivatives | Adenine - chemical synthesis | Adenine - pharmacology | Adenine - chemistry | Hydrogenation | Tenofovir | Organophosphonates - chemical synthesis | Organophosphonates - pharmacology | Combinatorial Chemistry Techniques | Antiviral Agents - chemistry | Organophosphonates - chemistry | Antiviral Agents - chemical synthesis | Molecular Structure | Catalysis
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18. Full Text Review on modern advances of chemical methods for the introduction of a phosphonic acid group
by Demmer, Charles S and Krogsgaard-Larsen, Niels and Bunch, Lennart
Chemical Reviews, ISSN 0009-2665, 12/2011, Volume 111, Issue 12, pp. 7981 - 8006
GRB2 SH2 DOMAIN | TYROSINE-PHOSPHATASE 1B | ANALOGS | BOND FORMATION | H-PHOSPHONATES | ALDEHYDES | PALLADIUM-CATALYZED HYDROPHOSPHORYLATION | INHIBITORS | EFFICIENT | CHEMISTRY, MULTIDISCIPLINARY | DISCOVERY | Chemistry, Organic - methods | Nickel - chemistry | Manganese - chemistry | Molybdenum | Carbon - chemistry | Organophosphonates - chemical synthesis | Phosphorous Acids - chemistry | Copper - chemistry | Zinc Oxide - chemistry | Chemical Phenomena | Organophosphonates - chemistry | Catalysis | Palladium - chemistry | Palladium catalysts | Carbonyl compounds | Usage | Analysis | Organophosphorus compounds | Chemical properties | Ring formation (Chemistry) | Structure
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19. Full Text Organocatalytic enantioselective synthesis of α-hydroxy phosphonates
by Samanta, Sampak and Zhao, Cong-Gui
Journal of the American Chemical Society, ISSN 0002-7863, 06/2006, Volume 128, Issue 23, pp. 7442 - 7443
Tertiary alpha-hydroxy phosphonates have been synthesized in good yields and high enantiomeric purity (up to 99% ee) through a novel l-proline-catalyzed cross... 
ASPERGILLUS-NIGER | ORGANIC-CHEMISTRY | ENANTIOMERIC EXCESS | ASYMMETRIC-SYNTHESIS | REDUCTION | KETOPHOSPHONATES | ENZYMES | HYDROLYSIS | HYDROXYALKYLPHOSPHONATES | DERIVATIVES | CHEMISTRY, MULTIDISCIPLINARY | Organophosphonates - chemical synthesis | Molecular Structure | Catalysis | Enzyme Inhibitors - chemical synthesis | Hydroxy Acids - chemistry | Stereoisomerism
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20. Full Text Synthesis and antitumor activities of novel thiourea α-aminophosphonates from dehydroabietic acid
by Huang, Xiao-Chao and Wang, Meng and Wang, Heng-Shan and Pan, Ying-Ming and Yao, Gui-Yang and Tian, Xiao-Yan and Qin, Jiang-Ke and Zhang, Ye
European Journal of Medicinal Chemistry, ISSN 0223-5234, 11/2013, Volume 69, pp. 508 - 520
A series of novel thiourea α-aminophosphonate derivatives containing DHA structure was designed and synthesized as antitumor agents. Their inhibitory... 
Thiourea | Cytotoxicity | Dehydroabietic acid | α-Aminophosphonate | Apoptosis | ANTICANCER ACTIVITY | CHEMISTRY, MEDICINAL | alpha-Aminophosphonate | DNA | DRUGS | Cell Survival - drug effects | Apoptosis - drug effects | Antineoplastic Agents - chemical synthesis | Humans | Diterpenes, Abietane - chemistry | Structure-Activity Relationship | Thiourea - pharmacology | Antineoplastic Agents - chemistry | Hep G2 Cells | Dose-Response Relationship, Drug | Organophosphonates - chemical synthesis | Organophosphonates - pharmacology | Thiourea - chemical synthesis | Organophosphonates - chemistry | Cell Line, Tumor | Antineoplastic Agents - pharmacology | Cell Proliferation - drug effects | Molecular Structure | Thiourea - analogs & derivatives | Drug Screening Assays, Antitumor
Journal Article