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Molecular and cellular endocrinology, ISSN 0303-7207, 2007, Volume 275, Issue 1, pp. 71 - 78
Mechanisms of action | SEGRA | Non-genomic | mGCR | Glucocorticoid | cGCR | Genomic | Endocrinology & Metabolism | Life Sciences & Biomedicine | Science & Technology | Cell Biology | Animals | Anti-Inflammatory Agents - pharmacology | Humans | Glucocorticoids - pharmacology | Immunosuppressive Agents - pharmacology | Cell Membrane - drug effects | Receptors, Glucocorticoid - agonists | Index Medicus
Journal Article
Cell (Cambridge), ISSN 0092-8674, 2011, Volume 145, Issue 2, pp. 224 - 241
Biochemistry & Molecular Biology | Life Sciences & Biomedicine | Science & Technology | Cell Biology | Promoter Regions, Genetic | Animals | Cytokines | Response Elements | Humans | Gene Expression Regulation | Transcription, Genetic | Mice | Dermatitis, Atopic - metabolism | Repressor Proteins - metabolism | Receptors, Glucocorticoid - agonists | Corticosteroids | Steroids | Index Medicus
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Bioorganic & medicinal chemistry letters, ISSN 0960-894X, 09/2020, Volume 30, Issue 17, pp. 127402 - 127402
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British journal of pharmacology, ISSN 0007-1188, 05/2015, Volume 172, Issue 10, pp. 2634 - 2653
Epithelial Cells - metabolism | Respiratory Mucosa - drug effects | Colforsin - pharmacology | Epithelial Cells - drug effects | Humans | Transcriptional Activation - drug effects | Cells, Cultured | Quinolones - pharmacology | Receptors, Glucocorticoid - metabolism | Adrenergic beta-2 Receptor Agonists - pharmacology | Dexamethasone - analogs & derivatives | Dexamethasone - pharmacology | Drug Interactions | Transfection | Ligands | Steroids - pharmacology | Response Elements - genetics | Respiratory Mucosa - metabolism | Benzodioxoles - pharmacology | Indans - pharmacology | Index Medicus | Research Papers
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Carcinogenesis (New York), ISSN 0143-3334, 04/2019, Volume 40, Issue 2, pp. 335 - 348
Life Sciences & Biomedicine | Oncology | Science & Technology | Cell Proliferation - genetics | Humans | Carcinogenesis - genetics | Signal Transduction - genetics | Down-Regulation - genetics | Animals | Breast Neoplasms - genetics | MCF-7 Cells | NF-kappa B - genetics | Mice, Nude | Receptors, Glucocorticoid - genetics | Cell Line, Tumor | Neoplastic Stem Cells - pathology | Female | Mice | Mice, Inbred BALB C | MicroRNAs - genetics | Index Medicus
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Pharmacological research, ISSN 1043-6618, 06/2020, Volume 156, pp. 104802 - 104802
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Journal of medicinal chemistry, ISSN 0022-2623, 06/2008, Volume 51, Issue 12, pp. 3349 - 3352
Hormones. Endocrine system | Biological and medical sciences | Medical sciences | Pharmacology. Drug treatments | Androstadienes - chemistry | Humans | Models, Molecular | Crystallography, X-Ray | Protein Conformation | Nuclear Receptor Coactivator 2 - chemistry | Binding Sites | Receptors, Glucocorticoid - chemistry | Receptors, Glucocorticoid - agonists | Index Medicus | DEXAMETHASONE | GLUCOCORTICOIDS | LIGANDS | ESTERS | CRYSTAL STRUCTURE | RECEPTORS | 60 APPLIED LIFE SCIENCES
Journal Article
The Journal of steroid biochemistry and molecular biology, ISSN 0960-0760, 02/2019, Volume 186, pp. 142 - 153
Virtual screening | MD simulations | Selective agonists | Anti-Inflammatory action | Pharmacophore model | Glucocorticoid receptor | Biochemistry & Molecular Biology | Endocrinology & Metabolism | Life Sciences & Biomedicine | Science & Technology | Benzothiazoles - pharmacology | Humans | Models, Molecular | Anti-Inflammatory Agents, Non-Steroidal - chemistry | Receptors, Glucocorticoid - metabolism | Drug Discovery | Anti-Inflammatory Agents, Non-Steroidal - pharmacology | Receptors, Glucocorticoid - agonists | Gene Expression Regulation - drug effects | NF-kappa B - genetics | Drug Design | Benzothiazoles - chemistry | HeLa Cells | Receptors, Glucocorticoid - chemistry | NF-κB protein | Side effects | Inflammation | Antiinflammatory agents | Glucocorticoids | Benzothiazole | Index Medicus
Journal Article
Journal of bone and mineral research, ISSN 0884-0431, 11/2012, Volume 27, Issue 11, pp. 2238 - 2241
Life Sciences & Biomedicine | Endocrinology & Metabolism | Science & Technology | Receptors, Glucocorticoid - metabolism | Animals | Bone Density | Humans | Physiological aspects | Corticosteroids | Steroids | Index Medicus | Obesity | Antiinflammatory agents | Glucocorticoids | Diabetes mellitus | Cushing's syndrome | Glucocorticoid receptors | Atrophy | Glucose tolerance | Osteoporosis | Side effects | Skin | Bone | Myopathy
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Journal of medicinal chemistry, ISSN 0022-2623, 03/2015, Volume 58, Issue 6, pp. 2658 - 2677
Cell Line | Anti-Inflammatory Agents - pharmacology | Humans | Matrix Metalloproteinase 13 - genetics | Tumor Necrosis Factor-alpha - blood | Models, Molecular | Crystallography, X-Ray | Receptors, Glucocorticoid - metabolism | Receptors, Glucocorticoid - agonists | Up-Regulation - drug effects | Phenanthrenes - chemistry | Phenanthrenes - pharmacology | Animals | Dexamethasone - pharmacology | Interleukin-1 - immunology | Tumor Necrosis Factor-alpha - immunology | Mice | Mammary Tumor Virus, Mouse - genetics | Index Medicus
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Non-steroidal glucocorticoid agonists—The discovery of aryl pyrazoles as A-ring mimetics
Bioorganic & medicinal chemistry letters, ISSN 0960-894X, 2007, Volume 17, Issue 17, pp. 4737 - 4745
Aryl pyrazole | Agonist | Glucocorticoid | Non-steroidal | Dissociated | Tetrahydronaphthalene | Physical Sciences | Chemistry | Chemistry, Organic | Life Sciences & Biomedicine | Pharmacology & Pharmacy | Chemistry, Medicinal | Science & Technology | Biological and medical sciences | Medical sciences | Pharmacology. Drug treatments | Bones, joints and connective tissue. Antiinflammatory agents | Chemistry, Pharmaceutical - methods | Models, Chemical | Stereoisomerism | Molecular Conformation | Receptors, Glucocorticoid - agonists | Pyrazoles - chemistry | Drug Design | Amides - chemistry | Inhibitory Concentration 50 | Drug Evaluation, Preclinical | Binding Sites | Glucocorticoids - agonists | Steroids - chemistry | Index Medicus
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