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Neuron (Cambridge, Mass.), ISSN 0896-6273, 06/2018, Volume 98, Issue 5, pp. 963 - 976.e5
opioid receptor | ligand-induced activation | endosome | biosensor | signaling | ligand bias | GPCR | Golgi | opioid drug | subcellular location | Neurosciences | Neurosciences & Neurology | Life Sciences & Biomedicine | Science & Technology | Dendrites - metabolism | Humans | Morphine - metabolism | Rats | Intracellular Space | Endosomes - metabolism | Narcotic Antagonists | Animals | Naloxone | Peptides - metabolism | Enkephalin, Ala-MePhe-Gly- - metabolism | Enkephalin, D-Penicillamine (2,5)- - metabolism | Enkephalin, Leucine-2-Alanine - metabolism | Biosensing Techniques | HEK293 Cells | Golgi Apparatus - metabolism | Spatio-Temporal Analysis | Cell Membrane - metabolism | Neurons - metabolism | Analgesics, Opioid - metabolism | HeLa Cells | Microscopy, Fluorescence | Receptors, Opioid - metabolism | Drugs | Neurons | Detectors | Plasma | Opioid receptors | Peptides | Narcotics | Cloning | Bias | Time series | Experiments | Neuromodulation | Golgi apparatus | Internalization | Ligands | Sensors | Biosensors | Endosomes
Journal Article
Annual review of medicine, ISSN 0066-4219, 1/2016, Volume 67, Issue 1, pp. 433 - 451
peripheral | plasticity | pain | inflammation | tolerance | addiction | Tolerance | Inflammation | Pain | Peripheral | Addiction | Plasticity | Receptors, Opioid - agonists | Chronic Pain - drug therapy | Opioid-Related Disorders - etiology | Signal Transduction | Humans | Drug Tolerance | Analgesics, Opioid - pharmacology | Analgesics, Opioid - therapeutic use | Pain - metabolism | Narcotic Antagonists - therapeutic use | Time Factors | Neuronal Plasticity | Pain - drug therapy | Ligands | Receptors, Opioid - drug effects | Receptors, Opioid - metabolism | Complications and side effects | Dosage and administration | Drug therapy | Chronic pain | Opioids | Drugs | Molecules | Side effects | Index Medicus
Journal Article
Nature neuroscience, ISSN 1097-6256, 2014, Volume 17, Issue 4, pp. 540 - 548
Neurosciences | Neurosciences & Neurology | Life Sciences & Biomedicine | Science & Technology | Endocannabinoids - metabolism | Receptors, Opioid, delta - metabolism | Neuronal Plasticity - drug effects | Male | Long-Term Synaptic Depression - drug effects | Corpus Striatum - metabolism | Receptors, Opioid - physiology | Female | Receptors, Opioid - metabolism | Long-Term Synaptic Depression - physiology | Oxycodone - administration & dosage | Receptors, Opioid, mu - drug effects | Receptors, Opioid, mu - metabolism | Mice, Inbred C57BL | Receptors, Opioid, kappa - metabolism | Rats | Receptors, Opioid, delta - drug effects | Opioid Peptides - metabolism | Rats, Sprague-Dawley | Receptors, Opioid, kappa - physiology | Receptors, Opioid, kappa - drug effects | Animals | Analgesics, Opioid - administration & dosage | Corpus Striatum - drug effects | Mice | Receptors, Opioid - drug effects | Receptors, Opioid, delta - physiology | Receptors, Opioid, mu - physiology | Drug abuse | Depression, Mental | Opioids | Physiological aspects | Corpus striatum | Health aspects | Risk factors | Index Medicus
Journal Article
Nature (London), ISSN 0028-0836, 2014, Volume 506, Issue 7487, pp. 191 - 196
Science & Technology - Other Topics | Multidisciplinary Sciences | Science & Technology | Naltrexone - analogs & derivatives | Receptors, Opioid, delta - metabolism | Humans | Naltrexone - chemistry | Crystallography, X-Ray | Structure-Activity Relationship | Sodium - metabolism | Arrestins - metabolism | Narcotic Antagonists - chemistry | Naltrexone - pharmacology | Narcotic Antagonists - metabolism | Receptors, Opioid, delta - genetics | Receptors, Opioid, delta - antagonists & inhibitors | Asparagine - genetics | Naltrexone - metabolism | Allosteric Regulation - drug effects | Allosteric Site - genetics | Sodium - pharmacology | Allosteric Regulation - genetics | Mutagenesis, Site-Directed | Receptors, Opioid, delta - chemistry | Allosteric Site - drug effects | Models, Molecular | Signal Transduction - drug effects | beta-Arrestins | Asparagine - metabolism | Narcotic Antagonists - pharmacology | Ligands | Receptors, Opioid, delta - agonists | Index Medicus | sodium regulation | constitutive activity | human opioid receptor | arrestin | functional selectivity | GPCR signaling | allostery
Journal Article
Journal of medicinal chemistry, ISSN 0022-2623, 07/2020, Volume 63, Issue 14, pp. 7663 - 7694
Receptors, Opioid, delta - metabolism | Analgesics, Opioid - chemical synthesis | Cricetulus | Humans | Microsomes, Liver - metabolism | Narcotic Antagonists - chemical synthesis | Male | Structure-Activity Relationship | Receptors, Opioid, mu - agonists | Morphinans - metabolism | Narcotic Antagonists - metabolism | Drug Design | Receptors, Opioid, delta - antagonists & inhibitors | Molecular Structure | CHO Cells | Morphinans - therapeutic use | Pyridines - therapeutic use | Receptors, Opioid, mu - metabolism | Pyridines - chemical synthesis | Analgesics, Opioid - therapeutic use | Morphinans - chemical synthesis | Animals | Pyridines - metabolism | Narcotic Antagonists - therapeutic use | Protein Binding | Mice | Molecular Docking Simulation | Analgesics, Opioid - metabolism | Index Medicus
Journal Article
The New England journal of medicine, ISSN 0028-4793, 03/2016, Volume 374, Issue 13, pp. 1253 - 1263
Medicine, General & Internal | Life Sciences & Biomedicine | General & Internal Medicine | Science & Technology | Opioid-Related Disorders - epidemiology | Chronic Pain - drug therapy | Receptors, Opioid, mu - metabolism | Humans | Drug Tolerance | Opioid-Related Disorders - diagnosis | Analgesics, Opioid - therapeutic use | Opioid-Related Disorders - prevention & control | Chronic Pain - physiopathology | Opioid-Related Disorders - physiopathology | Prevention | Care and treatment | Dosage and administration | Chronic pain | Opioids | Drug abuse | Pain | Addiction | Abuse | Narcotics | Drug tolerance | Pain management | Chronic illnesses | Index Medicus | Abridged Index Medicus
Journal Article
Nature (London), ISSN 0028-0836, 05/2012, Volume 485, Issue 7398, pp. 327 - 332
Science & Technology - Other Topics | Multidisciplinary Sciences | Science & Technology | Structure of solids and liquids; crystallography | Structure of specific crystalline solids | Physics | Exact sciences and technology | Condensed matter: structure, mechanical and thermal properties | Organic compounds | Naltrexone - analogs & derivatives | Humans | Naltrexone - chemistry | Crystallography, X-Ray | Structure-Activity Relationship | Diterpenes, Clerodane - chemistry | Receptors, Adrenergic, beta-2 - chemistry | Piperidines - pharmacology | Tetrahydroisoquinolines - chemistry | Receptors, Opioid, kappa - chemistry | Binding Sites | Receptors, Opioid, kappa - genetics | Naltrexone - metabolism | Morphinans - chemistry | Tetrahydroisoquinolines - pharmacology | Piperidines - chemistry | Receptors, Opioid, kappa - antagonists & inhibitors | Mutagenesis, Site-Directed | Receptors, Opioid, kappa - metabolism | Models, Molecular | Receptors, CXCR4 - metabolism | Guanidines - chemistry | Diterpenes, Clerodane - metabolism | Diterpenes, Clerodane - pharmacology | Protein Conformation | Receptors, CXCR4 - chemistry | Index Medicus
Journal Article