X
Search Filters
Format Format
Subjects Subjects
Subjects Subjects
X
Sort by Item Count (A-Z)
Filter by Count
aicar, aminoimidazole-4-carboxamide-1-β-d-ribofuranoside (1) 1
amino acid sequence (1) 1
ampk, amp-activated protein kinase (1) 1
animals (1) 1
anti-cancer drugs (1) 1
atf2, activating transcription factor 2 (1) 1
atm, ataxia telangiectasia mutated (1) 1
biochemistry & molecular biology (1) 1
brsk, brain-specific kinase (1) 1
cak, cyclin-dependent kinase-activating kinase (1) 1
camk, calmodulin-dependent kinase (1) 1
camkk, camk kinase (1) 1
cdk, cyclin-dependent protein kinase (1) 1
cell line (1) 1
cell-proliferation (1) 1
chk, checkpoint kinase (1) 1
ck, casein kinase (1) 1
csk, c-terminal src kinase (1) 1
cyclin-dependent kinases (1) 1
drug design (1) 1
drug discovery (1) 1
dyrk, dual-specificity tyrosine-phosphorylated and -regulated kinase (1) 1
ef2k, elongation-factor-2 kinase (1) 1
egf, epidermal growth factor (1) 1
enzyme activation (1) 1
eph-a2, ephrin a2 receptor (1) 1
erk, extracellular-signal-regulated kinase (1) 1
family-members (1) 1
fgf-r, fibroblast-growth-factor receptor (1) 1
fkbp, fk506-binding protein (1) 1
fmk, fluoromethylketone (1) 1
gak, cyclin g-associated kinase (1) 1
gsk3, glycogen synthase kinase 3 (1) 1
gst, glutathione transferase (1) 1
hek-293 cells, human embryonic kidney-293 cells (1) 1
hipk, homeodomain-interacting protein kinase (1) 1
his6, hexahistidine (1) 1
humans (1) 1
igf-1, insulin-like growth factor-1 (1) 1
ikk, inhibitory κb kinase (1) 1
il-1, interleukin 1 (1) 1
index medicus (1) 1
inhibitor specificity (1) 1
isoforms in-vitro (1) 1
jnk, c-jun n-terminal kinase (1) 1
kinase profiling (1) 1
lck, lymphocyte cell-specific protein-tyrosine kinase (1) 1
life sciences (1) 1
lps, lipopolysaccharide (1) 1
mapk, mitogen-activated protein kinase (1) 1
mapkap-k, mapk-activated protein kinase (1) 1
mark, microtubule-affinity-regulating kinase (1) 1
mbp, myelin basic protein (1) 1
melk, maternal embryonic leucine-zipper kinase (1) 1
mitogen-activated protein kinases - antagonists & inhibitors (1) 1
mitogen-activated protein kinases - metabolism (1) 1
mkk1, mapk kinase-1 (1) 1
mms, methyl methanesulfonate (1) 1
mnk, mapk-integrating protein kinase (1) 1
msk, mitogen- and stress-activated protein kinase (1) 1
mst, mammalian homologue ste20-like kinase (1) 1
ndrg, n-myc downstream-regulated gene (1) 1
nek, nima-related kinase (1) 1
nfat, nuclear factor for activated t-cells (1) 1
p38 map kinase (1) 1
p90 rsk (1) 1
pak, p21-activated protein kinase (1) 1
pdk, 3-phosphoinositide-dependent protein kinase (1) 1
ph, pleckstrin homology (1) 1
phk, phosphorylase kinase (1) 1
phosphorylation (1) 1
pi3k, phosphatidylinositol 3-kinase (1) 1
pim, provirus integration site for moloney murine leukaemia virus (1) 1
pka, camp-dependent protein kinase (1) 1
pkb, protein kinase b (1) 1
pkc, protein kinase c (1) 1
pkd, protein kinase d (1) 1
plk, polo-like kinase (1) 1
ppar, peroxisome-proliferator-activated receptor (1) 1
prak, p38-regulated activated kinase (1) 1
prk, protein kinase c-related kinase (1) 1
protein kinase (1) 1
protein kinase inhibitors - pharmacology (1) 1
pten, phosphatase and tensin homologue deleted on chromosome 10 (1) 1
receptor tyrosine kinases (1) 1
recombinant proteins - antagonists & inhibitors (1) 1
research article (1) 1
rho-associated kinase (1) 1
rip2, receptor-interacting protein 2 (1) 1
rock, rho-dependent protein kinase (1) 1
rsk, p90 ribosomal s6 kinase (1) 1
s6k1, s6 kinase 1 (1) 1
sb 203580 (1) 1
sf21, spodoptera frugiperda 21 (1) 1
sgk, serum- and glucocorticoid-induced kinase (1) 1
smmlck, smooth-muscle myosin light-chain kinase (1) 1
spodoptera (1) 1
src, sarcoma kinase (1) 1
src-i1, src inhibitor 1 (1) 1
srpk, serine-arginine protein kinase (1) 1
more...
Language Language
Publication Date Publication Date
Click on a bar to filter by decade
Slide to change publication date range


Biochemical Journal, ISSN 0264-6021, 12/2007, Volume 408, Issue 3, pp. 297 - 315
The specificities of 65 compounds reported to be relatively specific inhibitors of protein kinases have been profiled against a panel of 70-80 protein kinases.... 
Drug discovery | Kinase profiling | Protein kinase | Anti-cancer drugs | Inhibitor specificity | RHO-ASSOCIATED KINASE | TUMOR PROGRESSION | FAMILY-MEMBERS | BIOCHEMISTRY & MOLECULAR BIOLOGY | CELL-PROLIFERATION | protein kinase | P38 MAP KINASE | CYCLIN-DEPENDENT KINASES | RECEPTOR TYROSINE KINASES | drug discovery | kinase profiling | SB 203580 | anti-cancer drugs | ISOFORMS IN-VITRO | P90 RSK | inhibitor specificity | Amino Acid Sequence | Cell Line | Phosphorylation | Recombinant Proteins - antagonists & inhibitors | Animals | Mitogen-Activated Protein Kinases - antagonists & inhibitors | Humans | Drug Design | Protein Kinase Inhibitors - pharmacology | Enzyme Activation | Mitogen-Activated Protein Kinases - metabolism | Spodoptera | Index Medicus | Yes1, Yamaguchi sarcoma viral oncogene homologue 1 | CSK, C-terminal Src kinase | Lck, lymphocyte cell-specific protein-tyrosine kinase | EGF, epidermal growth factor | FGF-R, fibroblast-growth-factor receptor | PAK, p21-activated protein kinase | PDK, 3-phosphoinositide-dependent protein kinase | PI3K, phosphatidylinositol (phosphoinositide) 3-kinase | NEK, NIMA (never in mitosis in Aspergillus nidulans)-related kinase | RSK, p90 ribosomal S6 kinase | HEK-293 cells, human embryonic kidney-293 cells | VEGF, vascular endothelial growth factor (vasoendothelial growth factor) | EF2K, elongation-factor-2 kinase | CK, casein kinase | PTEN, phosphatase and tensin homologue deleted on chromosome 10 | ERK, extracellular-signal-regulated kinase | ATM, ataxia telangiectasia mutated | SRPK, serine-arginine protein kinase | IL-1, interleukin 1 | MNK, MAPK-integrating protein kinase | ROCK, Rho-dependent protein kinase | CaMKK, CaMK kinase | GST, glutathione transferase | MKK1, MAPK kinase-1 (also called MEK1, MAPK or ERK kinase 1) | GAK, cyclin G-associated kinase | FMK, fluoromethylketone | MST, mammalian homologue Ste20-like kinase | PKA, cAMP-dependent protein kinase | FKBP, FK506-binding protein | PPAR, peroxisome-proliferator-activated receptor | IKK, inhibitory κB kinase | PH, pleckstrin homology | MBP, myelin basic protein | AICAR, aminoimidazole-4-carboxamide-1-β-D-ribofuranoside | MAPKAP-K, MAPK-activated protein kinase | Sf21, Spodoptera frugiperda (fall armyworm) 21 | MARK, microtubule-affinity-regulating kinase | PIM, provirus integration site for Moloney murine leukaemia virus | LPS, lipopolysaccharide | MSK, mitogen- and stress-activated protein kinase | MAPK, mitogen-activated protein kinase | MELK, maternal embryonic leucine-zipper kinase | His6, hexahistidine | CAK, cyclin-dependent kinase-activating kinase | Eph-A2, Ephrin A2 receptor | PLK, polo-like kinase | ATF2, activating transcription factor 2 | PKD, protein kinase D | Src, sarcoma kinase | AMPK, AMP-activated protein kinase | MMS, methyl methanesulfonate | CHK, checkpoint kinase | JNK, c-Jun N-terminal kinase | TORC1, mTOR (mammalian target of rapamycin)–raptor (regulatory associated protein of mTOR) complex | BRSK, brain-specific kinase | RIP2, receptor-interacting protein 2 | IGF-1, insulin-like growth factor-1 | S6K1, S6 kinase 1 | DYRK, dual-specificity tyrosine-phosphorylated and -regulated kinase | HIPK, homeodomain-interacting protein kinase | ZMP, aminoimidazole-4-carboxamide-1-β-D-ribofuranoside monophosphate | PRAK, p38-regulated activated kinase | PKC, protein kinase C | Src-I1, Src inhibitor 1 | TANK, TRAF (tumour-necrosis-factor-receptor-associated factor)-family-member-associated nuclear factor κB activator | NFAT, nuclear factor for activated T-cells | PHK, phosphorylase kinase | GSK3, glycogen synthase kinase 3 | PKB, protein kinase B (also called Akt) | CaMK, calmodulin-dependent kinase | CDK, cyclin-dependent protein kinase | NDRG, N-myc downstream-regulated gene | SmMLCK, smooth-muscle myosin light-chain kinase | TBK1, TANK-binding kinase 1 | PRK, protein kinase C-related kinase | SGK, serum- and glucocorticoid-induced kinase
Journal Article
No results were found for your search.

Cannot display more than 1000 results, please narrow the terms of your search.