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1. Full Text Discriminative stimulus properties of the atypical antipsychotic amisulpride: comparison to its isomers and to other benzamide derivatives, antipsychotic, antidepressant, and antianxiety drugs in C57BL/6 mice
by Donahue, Timothy J and Hillhouse, Todd M and Webster, Kevin A and Young, Richard and De Oliveira, Eliseu O and Porter, Joseph H
Psychopharmacology, ISSN 0033-3158, 12/2017, Volume 234, Issue 23, pp. 3507 - 3520
Racemic (RS)-amisulpride (Solian®) is an atypical antipsychotic drug used to treat schizophrenia and dysthymia. Blockade of dopamine D2/D3 and/or serotonin... 
Drug discrimination | Neurosciences | Amisulpride | Schizophrenia | Isomers | Anxiolytics | Discriminative stimulus | Antipsychotics | Biomedicine | Antidepressants | C57BL/6 mice | Benzamides | Pharmacology/Toxicology | Psychiatry | CORTICAL MEMBRANES | PSYCHIATRY | HIGH-AFFINITY | MAJOR DEPRESSION | D-2 RECEPTORS | NEUROSCIENCES | RECEPTOR ANTAGONIST | LIMBIC SELECTIVITY | 5-HT7 RECEPTOR | PHARMACOLOGY & PHARMACY | MOLECULAR-CLONING | RAT-BRAIN | DOPAMINE-RECEPTORS | Sulpiride - pharmacology | Conditioning, Operant - physiology | Male | Sulpiride - analogs & derivatives | Clozapine - pharmacology | Discrimination Learning - drug effects | Clozapine - chemistry | Conditioning, Operant - drug effects | Antidepressive Agents - chemistry | Anti-Anxiety Agents - chemistry | Antidepressive Agents - pharmacology | Benzamides - pharmacology | Quetiapine Fumarate - pharmacology | Benzamides - chemistry | Quetiapine Fumarate - chemistry | Mice, Inbred C57BL | Chlorpromazine - chemistry | Risperidone - pharmacology | Anti-Anxiety Agents - pharmacology | Chlorpromazine - pharmacology | Risperidone - chemistry | Discrimination Learning - physiology | Animals | Antipsychotic Agents - chemistry | Mice | Antipsychotic Agents - pharmacology | Sulpiride - chemistry | Dosage and administration | Antipsychotic drugs | Comparative analysis | Drug interactions | Antianxiety agents | Stereoisomers | Drugs | Neuroleptics | Olanzapine | Operant conditioning | Mental disorders | Aripiprazole | Benzamide | Metoclopramide | Chlorpromazine | Sulpiride | Serotonin S7 receptors | Psychotropic drugs | Imipramine | Receptors | Bupropion | Mianserin | Risperidone | Dopamine D2 receptors | Drug dosages | Quetiapine | Raclopride | Dopamine | Serotonin | Dopamine D3 receptors | Chlordiazepoxide | Pharmacology | Clozapine | Derivatives | Properties (attributes) | Serotonin receptors
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2. Full Text Structural basis for Na+-sensitivity in dopamine D2 and D3 receptors
by Michino, Mayako and Free, R. Benjamin and Doyle, Trevor B and Sibley, David R and Shi, Lei
Chemical Communications, ISSN 1359-7345, 2015, Volume 51, Issue 41, pp. 8618 - 8621
To understand the structural basis for the Na+-sensitivity of ligand binding to dopamine D2-like receptors, using computational analysis in combination with... 
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3. Full Text Structural basis for Na + -sensitivity in dopamine D2 and D3 receptors
by Michino, Mayako and Free, R. Benjamin and Doyle, Trevor B and Sibley, David R and Shi, Lei
Chemical Communications, ISSN 1359-7345, 05/2015, Volume 51, Issue 41, pp. 8618 - 8621
To understand the structural basis for the Na+-sensitivity of ligand binding to dopamine D2-like receptors, using computational analysis in combination with... 
SODIUM-BINDING | ANTAGONIST | INHIBITION | AFFINITY | MEMBRANE | BINDING-SITE CREVICE | PROTEIN-COUPLED RECEPTORS | ALLOSTERIC MODULATION | RESIDUES | CHEMISTRY, MULTIDISCIPLINARY | PIVOTAL ROLE | Sodium - pharmacology | Sulpiride - pharmacology | Sodium - chemistry | Protein Conformation - drug effects | Receptors, Dopamine D3 - chemistry | Receptors, Dopamine D3 - metabolism | Structure-Activity Relationship | Receptors, Dopamine D2 - metabolism | Molecular Dynamics Simulation | Dose-Response Relationship, Drug | Dopamine Antagonists - pharmacology | Salicylamides - chemistry | Receptors, Dopamine D2 - chemistry | Ligands | Benzamides - pharmacology | Molecular Structure | Receptors, Dopamine D3 - antagonists & inhibitors | Dopamine Antagonists - chemistry | Salicylamides - pharmacology | Sulpiride - chemistry | Binding Sites - drug effects | Benzamides - chemistry
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4. Full Text Development of a novel l-sulpiride-loaded quaternary microcapsule: Effect of TPGS as an absorption enhancer on physicochemical characterization and oral bioavailability
by Kim, Dong Wuk and Kim, Dong Shik and Kim, Jong Oh and Kim, Kyeong Soo and Choi, Han-Gon and Choi, Jong Seo and Seo, Youn Gee and Youn, Yu Seok and Oh, Kyung Taek and Yong, Chul Soon and Jin, Sung Giu
Colloids and Surfaces B: Biointerfaces, ISSN 0927-7765, 11/2016, Volume 147, pp. 250 - 257
The aim of this study was to assess the effect of -α-tocopheryl polyethylene glycol 1000 succinate (TPGS) on the physicochemical characterization and oral... 
Oral absorption | l-sulpiride | Quaternary microcapsule | d-α-tocopheryl polyethylene glycol 1000 succinate | Administered drug dose | L-sulpiride | D-α-tocopheryl polyethylene glycol 1000 succinate | D-alpha-tocopheryl polyethylene glycol 1000 | MATERIALS SCIENCE, BIOMATERIALS | BIOPHARMACEUTICS CLASSIFICATION-SYSTEM | DRUG-DELIVERY SYSTEM | CHEMISTRY, PHYSICAL | VITAMIN-E TPGS | succinate | SOLID LIPID NANOPARTICLES | INTESTINAL-ABSORPTION | SOLUBLE DRUG | BIOPHYSICS | MODEL-DRUG | PARTICLE-SIZE | IN-VIVO EVALUATION | AQUEOUS SOLUBILITY | Povidone - administration & dosage | Surface-Active Agents | Polymers - administration & dosage | Administration, Oral | Solubility | Drug Carriers - administration & dosage | Rats | Biological Availability | Capsules - chemistry | Male | Sulpiride - administration & dosage | Sulpiride - pharmacokinetics | Rats, Sprague-Dawley | Drug Carriers - chemistry | Drug Delivery Systems | Tissue Distribution | Povidone - chemistry | Animals | Sodium Dodecyl Sulfate - chemistry | Vitamin E - administration & dosage | Polymers - chemistry | Vitamin E - chemistry | Sulpiride - chemistry | Sodium Dodecyl Sulfate - administration & dosage | Drugstores | Pharmacy | Polyethylene glycol | Polyols | Carriers | Carriers, Drug | Drugs | Solvents | Absorption | Bioavailability
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5. Full Text Development of novel amisulpride-loaded liquid self-nanoemulsifying drug delivery systems via dual tackling of its solubility and intestinal permeability
by Gamal, Wael and Fahmy, Rania H and Mohamed, Magdy I
Drug Development and Industrial Pharmacy, ISSN 0363-9045, 09/2017, Volume 43, Issue 9, pp. 1530 - 1538
Objective: The aim of the current investigation was at enhancing the oral biopharmaceutical behavior; solubility and intestinal permeability of amisulpride... 
Amisulpride | non-everted gut sac model | bioenhancers | ex vivo permeability testing | self-nanoemulsifying | ternary phase diagrams | DESIGN | CHEMISTRY, MEDICINAL | SNEDDS | TRANSDERMAL DELIVERY | EXCIPIENTS | ORAL ABSORPTION | DISSOLUTION | PHARMACOLOGY & PHARMACY | Administration, Oral | Emulsions - chemistry | Solubility | Biological Availability | Polyethylene Glycols - chemistry | Sulpiride - administration & dosage | Permeability | Chemistry, Pharmaceutical | Particle Size | Sulpiride - analogs & derivatives | Excipients - chemistry | Ethylene Glycols - chemistry | Drug Liberation | Surface-Active Agents - chemistry | Ethylene Glycols - administration & dosage | Drug Delivery Systems - methods | Sulpiride - chemistry | Intestinal Absorption - physiology
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6. Full Text Development of novel amisulpride-loaded solid self-nanoemulsifying tablets: preparation and pharmacokinetic evaluation in rabbits
by Gamal, Wael and Fahmy, Rania H and Mohamed, Magdy I
Drug Development and Industrial Pharmacy, ISSN 0363-9045, 09/2017, Volume 43, Issue 9, pp. 1539 - 1547
Objective: The current investigation is focused on the formulation and in vivo evaluation of optimized solid self-nanoemulsifying drug delivery systems... 
pharmacokinetics | Nanoemulsions | tableting | solid-state characterization | solid self-nanoemulsifying drug delivery systems | VITRO | IMPROVE | CHEMISTRY, MEDICINAL | FORMULATION | PLASMA | DISSOLUTION | WATER-SOLUBLE DRUGS | ORAL BIOAVAILABILITY | DOUBLE-BLIND | PHARMACOLOGY & PHARMACY | DRUG-DELIVERY SYSTEMS | IN-VIVO EVALUATION | Rabbits | Administration, Oral | Emulsions - chemistry | Tablets - pharmacokinetics | Biological Availability | Polyethylene Glycols - chemistry | Ethylene Glycols - pharmacokinetics | Sulpiride - administration & dosage | Sulpiride - pharmacokinetics | Chemistry, Pharmaceutical | Drug Carriers | Particle Size | Sulpiride - analogs & derivatives | Animals | Ethylene Glycols - chemistry | Tablets - chemistry | Surface-Active Agents - chemistry | Ethylene Glycols - administration & dosage | Drug Delivery Systems - methods | Sulpiride - chemistry
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7. Full Text Sulpiride, Amisulpride, Thioridazine, and Olanzapine: Interaction with Model Membranes. Thermodynamic and Structural Aspects
by Skrobecki, Piotr and Chmielińska, Anna and Bonarek, Piotr and Stepien, Piotr and Wisniewska-Becker, Anna and Dziedzicka-Wasylewska, Marta and Polit, Agnieszka
ACS Chemical Neuroscience, ISSN 1948-7193, 07/2017, Volume 8, Issue 7, pp. 1543 - 1553
Neuroleptic drugs are widely applied in effective treatment of schizophrenia and related disorders. The lipophilic character of neuroleptics means that they... 
calorimetry | drug-membrane interactions | Neuroleptics | liposomes | ζ potential | EPR | PLASMA-MEMBRANES | CHEMISTRY, MEDICINAL | BIOCHEMISTRY & MOLECULAR BIOLOGY | drug membrane interactions | zeta potential | BLOOD-BRAIN-BARRIER | NEUROSCIENCES | LIPID-BILAYERS | CHLORPROMAZINE INTERACTION | ANTIPSYCHOTIC-DRUGS | TITRATION CALORIMETRY | RAT-BRAIN | WATER PENETRATION | PHOSPHOLIPID-BILAYERS | HYDROPHOBIC BARRIER | Protons | Sulpiride - pharmacology | Benzodiazepines - pharmacology | Electron Spin Resonance Spectroscopy | Models, Chemical | Membranes, Artificial | Phosphatidylcholines - chemistry | Sulpiride - analogs & derivatives | Thermodynamics | Phosphatidylglycerols - chemistry | Antipsychotic Agents - chemistry | Thioridazine - pharmacology | Water - chemistry | Benzodiazepines - chemistry | Thioridazine - chemistry | Calorimetry | Molecular Structure | Antipsychotic Agents - pharmacology | Sulpiride - chemistry | Dynamic Light Scattering
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8. Full Text In Vivo Evaluation of a PEO-Gellan Gum Semi-Interpenetrating Polymer Network for the Oral Delivery of Sulpiride
by Hoosain, Famida G and Hoosain, Famida G and Choonara, Yahya E and Choonara, Yahya E and Kumar, Pradeep and Kumar, Pradeep and Tomar, Lomas K and Tomar, Lomas K and Tyagi, Charu and Tyagi, Charu and du Toit, Lisa C and du Toit, Lisa C and Pillay, Viness and Pillay, Viness
AAPS PharmSciTech, ISSN 1530-9932, 4/2017, Volume 18, Issue 3, pp. 654 - 670
In this study, an optimized epichlorohydrin-crosslinked semi-interpenetrating polymer network xerogel matrix system (XePoMas) for the controlled delivery of... 
Biochemistry, general | xerogel matrix | Biotechnology | semi-interpenetrating polymer network | Biomedicine | bioavailability | Pharmacy | gellan gum | Pharmacology/Toxicology | poly(ethylene oxide) | sulpiride | CONTROLLED DRUG-DELIVERY | INTESTINAL-ABSORPTION | MATRIX TABLETS | SYSTEMS | PHARMACOLOGY & PHARMACY | CELL | RELEASE KINETICS | Polysaccharides, Bacterial - chemistry | Chemistry, Pharmaceutical - methods | Administration, Oral | Biological Availability | Delayed-Action Preparations - chemistry | Polyethylene Glycols - chemistry | Epichlorohydrin - metabolism | Drug Liberation - drug effects | Delayed-Action Preparations - metabolism | Epichlorohydrin - chemistry | Animals | Swine | Polymers - chemistry | Drug Delivery Systems - methods | Sulpiride - chemistry | Sulpiride - metabolism | Drugs | Polysaccharides | Drug delivery systems | Analysis | Epoxy resins | Ethylene oxide | Vehicles
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9. Full Text Synchronizing the release rates of salicylate and indomethacin from degradable chitosan hydrogel and its optimization by definitive screening design
by Gabbay, Racheli Sharon and Kenett, Ron S and Scaffaro, Roberto and Rubinstein, Abraham
European Journal of Pharmaceutical Sciences, ISSN 0928-0987, 12/2018, Volume 125, pp. 102 - 109
Three types of ionically crosslinked (with citric acid) chitosan discs were loaded with the highly water- soluble drug, sodium salicylate (SS) and the poorly... 
Triggered erosion | Synchronized release rates | Dual drug platform | Multifactorial definitive screening design | Crosslinked chitosan | VITRO | SULPIRIDE | CANCER | DELIVERY | IN-VIVO ANALYSIS | MATRICES | PHARMACOLOGY & PHARMACY | ABSORPTION | Salicylic Acid - chemistry | Citric Acid - chemistry | Chitosan - chemistry | Cross-Linking Reagents - chemistry | Drug Design | Drug Liberation | Indomethacin - chemistry | Hydrogels - chemistry | Drug Delivery Systems | Crosslinked polymers | Indomethacin | Analysis | Citric acid | Calcium chloride
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10. Full Text Serotonergic and dopaminergic systems are implicated in antidepressant-like effects of chotosan, a Kampo formula, in mice
by Sasaki-Hamada, Sachie and Suzuki, Azusa and Ueda, Yudai and Matsumoto, Kinzo and Oka, Jun-Ichiro
Journal of Pharmacological Sciences, ISSN 1347-8613, 02/2017, Volume 133, Issue 2, pp. 110 - 113
We previously demonstrated that (CTS), a traditional herbal formula called medicine, improves diabetes-induced cognitive deficits. In the present study, we... 
Monoamine | Chotosan | Antidepressants | DEMENTIA | AMELIORATION | GEISSOSCHIZINE METHYL-ETHER | PHARMACOLOGY & PHARMACY | ANIMAL-MODEL | YOKUKANSAN | RECEPTORS | BRAIN | COGNITIVE DEFICITS | Ketanserin - pharmacology | Sulpiride - pharmacology | Pyridines - chemistry | Ketanserin - chemistry | Metergoline - chemistry | Drugs, Chinese Herbal - pharmacology | Male | Piperazines - chemistry | Imipramine - chemistry | Piperazines - pharmacology | Yohimbine - chemistry | Locomotion | Animals | Serotonin Agents - pharmacology | Dopamine Agents - pharmacology | Fenclonine - chemistry | Antidepressive Agents - pharmacology | Mice | Pyridines - pharmacology | Swimming | Imipramine - pharmacology | Medicine, Kampo | Sulpiride - chemistry | Disease Models, Animal | Care and treatment | Medicine, Botanic | Patient outcomes | Depression, Mental | Serotoninergic mechanisms | Medicine, Herbal | Dopaminergic mechanisms | Health aspects | Methods
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11. Full Text Effective determination of a pharmaceutical, sulpiride, in river water by online SPE-LC–MS using a molecularly imprinted polymer as a preconcentration medium
by Kubo, Takuya and Kuroda, Kenta and Tominaga, Yuichi and Naito, Toyohiro and Sueyoshi, Kenji and Hosoya, Ken and Otsuka, Koji
Journal of Pharmaceutical and Biomedical Analysis, ISSN 0731-7085, 02/2014, Volume 89, pp. 111 - 117
We report an effective and a quantitative analysis method for one of pharmaceuticals, sulpiride, in river water by online solid phase extraction (SPE)... 
Solid phase extraction | Interval recognition | Pharmaceutical | Molecular imprinting | Sulpiride | MULTIPLE PHARMACEUTICALS | CHEMISTRY, ANALYTICAL | PERSONAL CARE PRODUCTS | FEATHER MEAL | REENTRY | LIQUID-CHROMATOGRAPHY | DRUGS | SURFACE | PREVIOUSLY UNRECOGNIZED ROUTE | PHARMACOLOGY & PHARMACY | CATALYSTS | SOLID-PHASE EXTRACTION | Chromatography, High Pressure Liquid - methods | Solvents - chemistry | Water Pollutants, Chemical - chemistry | Fresh Water - chemistry | Water Pollutants, Chemical - analysis | Molecular Imprinting - methods | Adsorption | Rivers - chemistry | Solid Phase Extraction - methods | Polymers - chemistry | Fresh Water - analysis | Chromatography, Liquid - methods | Mass Spectrometry - methods | Sulpiride - chemistry | Polymers | Polymer industry | Usage | Analysis | Nitriles | Liquid chromatography | Mass spectrometry
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12. Full Text Measurement of clozapine, norclozapine, and amisulpride in plasma and in oral fluid obtained using 2 different sampling systems
by Fisher, Danielle S and Beyer, Chad and Van Schalkwyk, Gerrit and Seedat, Soraya and Flanagan, Robert J
Therapeutic Drug Monitoring, ISSN 0163-4356, 2017, Volume 39, Issue 2, pp. 109 - 117
Background: There is a poor correlation between total concentrations of proton-accepting compounds (most basic drugs) in unstimulated oral fluid and in plasma.... 
Amisulpride | Oral fluid | Plasma:oral fluid distribution | Clozapine | TDM | METABOLITES | SERUM | MS/MS | SALIVA | WHOLE-BLOOD | amisulpride | ANTIPSYCHOTICS | plasma:oral fluid distribution | oral fluid | DRUGS | clozapine | PHARMACOLOGY & PHARMACY | TOXICOLOGY | MEDICAL LABORATORY TECHNOLOGY | BINDING | Antipsychotic Agents - blood | Humans | Middle Aged | Body Fluids - chemistry | Male | Clozapine - analogs & derivatives | Drug Monitoring - methods | Mouth - chemistry | Sulpiride - analogs & derivatives | Young Adult | Tandem Mass Spectrometry | Antipsychotic Agents - chemistry | Clozapine - chemistry | Plasma - chemistry | Adult | Female | Aged | Clozapine - blood | Chromatography, Liquid - methods | Sulpiride - chemistry | Sulpiride - blood | Index Medicus
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13. Full Text Amisulpride–CD-Loaded Liposomes: Optimization and In Vivo Evaluation
by Shukr, Marwa H and Ahmed Farid, Omar A
AAPS PharmSciTech, ISSN 1530-9932, 8/2018, Volume 19, Issue 6, pp. 2658 - 2671
Amisulpride (AMS) is an atypical antipsychotic agent used for the treatment of schizophrenia. The effect of different variables, i.e., the type of... 
Biochemistry, general | Biotechnology | amisulpride | Biomedicine | liposomes | Pharmacy | Pharmacology/Toxicology | atypical antipsychotic | double loading | cyclodextrins | SYSTEM | MEMBRANE CONTACTOR | DRUG-DELIVERY | STABILITY | SCHIZOPHRENIA | RELEASE | RECEPTOR ANTAGONIST | CYCLODEXTRIN COMPLEXES | INTEGRITY | LIMBIC SELECTIVITY | PHARMACOLOGY & PHARMACY | 2-Hydroxypropyl-beta-cyclodextrin - metabolism | Rats, Wistar | Tablets | Amisulpride | Drug Carriers - administration & dosage | Biological Availability | Male | Sulpiride - administration & dosage | Drug Carriers - chemistry | Sulpiride - analogs & derivatives | Drug Liberation - physiology | Drug Evaluation, Preclinical - methods | Drug Carriers - metabolism | beta-Cyclodextrins - metabolism | Rats | 2-Hydroxypropyl-beta-cyclodextrin - administration & dosage | Antipsychotic Agents - administration & dosage | Particle Size | Animals | Antipsychotic Agents - chemistry | beta-Cyclodextrins - chemistry | 2-Hydroxypropyl-beta-cyclodextrin - chemistry | Antipsychotic Agents - metabolism | Liposomes | Sulpiride - chemistry | Sulpiride - metabolism
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14. Full Text An Epichlorohydrin-Crosslinked Semi-Interpenetrating GG-PEO Network as a Xerogel Matrix for Sustained Release of Sulpiride
by Hoosain, Famida G and Choonara, Yahya E and Kumar, Pradeep and Tomar, Lomas K and Tyagi, Charu and du Toit, Lisa C and Pillay, Viness
AAPS PharmSciTech, ISSN 1865-1372, 10/2014, Volume 15, Issue 5, pp. 1292 - 1306
The current study involved the development of a novel sustained release crosslinked semi-IPN xerogel matrix tablet prepared by chemical crosslinking of... 
Biochemistry, general | Biotechnology | semi-interpenetrating polymer network | Biomedicine | epichlorohydrin | sustained release | Pharmacy | matrix tablet | Pharmacology/Toxicology | sulpiride | GELLAN GUM | BEHAVIOR | POLYMER ELECTROLYTES | MECHANICAL-PROPERTIES | GRANULES | TABLETS | PHARMACOLOGY & PHARMACY | DRUG-DELIVERY SYSTEMS | WATER | Polysaccharides, Bacterial - chemistry | Excipients | Powders | Cross-Linking Reagents - chemistry | Hardness Tests | Solubility | Polyethylene Glycols - chemistry | Sulpiride - administration & dosage | Chemistry, Pharmaceutical | Antipsychotic Agents - administration & dosage | Epichlorohydrin - chemistry | Algorithms | Antipsychotic Agents - chemistry | Delayed-Action Preparations | Sulpiride - chemistry | Drugs | Polysaccharides | Drug delivery systems | Crosslinked polymers | Epoxy resins | Electron microscopy | Vehicles
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15. Full Text Photolysis of the antidepressants amisulpride and desipramine in wastewaters: Identification of transformation products formed and their fate
by Gros, Meritxell and Williams, Mike and Llorca, Marta and Rodriguez-Mozaz, Sara and Barceló, Damià and Kookana, Rai S and Sveriges lantbruksuniversitet
Science of the Total Environment, ISSN 0048-9697, 10/2015, Volume 530-531, pp. 434 - 444
Attenuation of pharmaceuticals due to natural sunlight is expected to be an important removal pathway in wastewater treatment plants using treatment lagoon... 
Transformation products | High-resolution mass spectrometry | Sewage | Lagoon | Photolysis | Pharmaceuticals | ENVIRONMENTAL SCIENCES | REMOVAL | WASTE-WATER | PHOTODEGRADATION | CARBAMAZEPINE | MICROPOLLUTANTS | Desipramine - analysis | Sulpiride - analogs & derivatives | Environmental Monitoring | Sulpiride - analysis | Antidepressive Agents - analysis | Desipramine - chemistry | Waste Water - chemistry | Antidepressive Agents - chemistry | Water Pollutants, Chemical - chemistry | Water Pollutants, Chemical - analysis | Sulpiride - chemistry | Purification | Wastewater | Mass spectrometry | Antidepressants, Tricyclic | Index Medicus | Miljövetenskap | Environmental Sciences
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16. Full Text Efficacy of surface charge in targeting pegylated nanoparticles of sulpiride to the brain
by Parikh, Tapan and Bommana, Murali Mohan and Squillante, Emilio
European Journal of Pharmaceutics and Biopharmaceutics, ISSN 0939-6411, 2010, Volume 74, Issue 3, pp. 442 - 450
The objective of the study was to formulate sulpiride-loaded nanoparticles (NPs) that can improve bioretention and achieve dose reduction by passively... 
Nanoparticles | Surface charge | Adsorption | Microscopy | Pegylation | Albumin | Cationized bovine serum albumin | CNS | Drug targeting | Sulpiride | Blood–brain barrier | DRUG | BARRIER | DELIVERY | Blood-brain barrier | PHARMACOLOGY & PHARMACY | Injections, Intravenous | Nanoparticles - chemistry | Male | Polyethylene Glycols - chemistry | Sulpiride - administration & dosage | Drug Carriers - chemistry | Brain - metabolism | Tissue Distribution | Cattle | Maleimides - chemical synthesis | Surface Properties | Drug Compounding | Serum Albumin, Bovine - chemistry | Microscopy, Electron, Scanning | Sulpiride - urine | Rats | Sulpiride - pharmacokinetics | Rats, Sprague-Dawley | Brain - drug effects | Particle Size | Polyesters - chemistry | Animals | Polyethylene Glycols - chemical synthesis | Maleimides - chemistry | Drug Delivery Systems - methods | Sulpiride - blood
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17. Full Text Spectroscopic investigation on the inclusion complex formation between amisulpride and γ-cyclodextrin
by Negi, Jeetendra Singh and Singh, Shivpal
Carbohydrate Polymers, ISSN 0144-8617, 02/2013, Volume 92, Issue 2, pp. 1835 - 1843
► Inclusion complex formation between amisulpride and gamma cyclodextrin was investigated. ► Bulky molecule of amisulpride was completely included inside...