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The New England journal of medicine, ISSN 0028-4793, 09/2010, Volume 363, Issue 14, pp. 1303 - 1312
Medicine, General & Internal | Life Sciences & Biomedicine | General & Internal Medicine | Science & Technology | Inflammatory joint diseases | Biological and medical sciences | General aspects | Medical sciences | Diseases of the osteoarticular system | Double-Blind Method | Humans | Intracellular Signaling Peptides and Proteins - antagonists & inhibitors | Middle Aged | Male | Treatment Outcome | Methotrexate - therapeutic use | Protein Kinase Inhibitors - adverse effects | Oxazines - adverse effects | Pyridines - adverse effects | Arthritis, Rheumatoid - drug therapy | Oxazines - therapeutic use | Protein Kinase Inhibitors - therapeutic use | Statistics, Nonparametric | Aged, 80 and over | Antirheumatic Agents - adverse effects | Adult | Female | Aged | Drug Therapy, Combination | Syk Kinase | Antirheumatic Agents - therapeutic use | Protein-Tyrosine Kinases - antagonists & inhibitors | Pyridines - therapeutic use | Spleen | Hypertension | Care and treatment | Rheumatoid arthritis | Physiological aspects | Health aspects | Risk factors | Tyrosine metabolism | Drug therapy | Drug dosages | Index Medicus | Abridged Index Medicus
Journal Article
Leukemia, ISSN 0887-6924, 2012, Volume 26, Issue 7, pp. 1576 - 1583
BCR | spleen tyrosine kinase (Syk) | chronic lymphyocytic leukemia (CLL) | Oncology | Life Sciences & Biomedicine | Hematology | Science & Technology | Hematologic and hematopoietic diseases | Leukemias. Malignant lymphomas. Malignant reticulosis. Myelofibrosis | Biological and medical sciences | Medical sciences | Apoptosis - drug effects | Protein-Tyrosine Kinases - metabolism | Humans | Intracellular Signaling Peptides and Proteins - metabolism | Flow Cytometry | Cyclohexylamines - pharmacology | Stromal Cells - drug effects | Phosphorylation - drug effects | Tumor Cells, Cultured | Syk Kinase | Enzyme-Linked Immunosorbent Assay | Intracellular Signaling Peptides and Proteins - antagonists & inhibitors | Stromal Cells - metabolism | Pyrimidines - pharmacology | Cell Adhesion - drug effects | Chemotaxis | Blotting, Western | Leukemia, Lymphocytic, Chronic, B-Cell - pathology | Cell Movement - drug effects | Leukemia, Lymphocytic, Chronic, B-Cell - enzymology | Cell Proliferation - drug effects | Protein Kinase Inhibitors - pharmacology | Leukemia, Lymphocytic, Chronic, B-Cell - drug therapy | Stromal Cells - cytology | Protein-Tyrosine Kinases - antagonists & inhibitors | Tyrosine | Chronic lymphocytic leukemia | Care and treatment | Growth | Development and progression | Genetic aspects | B cells | Properties | Cell migration | Index Medicus
Journal Article
Trends in pharmacological sciences (Regular ed.), ISSN 0165-6147, 2014, Volume 35, Issue 8, pp. 414 - 422
Advanced Basic Science | leukemia | protein kinase inhibitor | fostamatinib | tyrosine phosphorylation | allergic asthma | rheumatoid arthritis | Life Sciences & Biomedicine | Pharmacology & Pharmacy | Science & Technology | Animals | Protein Kinase Inhibitors - therapeutic use | Protein-Tyrosine Kinases - metabolism | Humans | Intracellular Signaling Peptides and Proteins - antagonists & inhibitors | Intracellular Signaling Peptides and Proteins - immunology | Intracellular Signaling Peptides and Proteins - metabolism | Protein Kinase Inhibitors - pharmacology | Molecular Targeted Therapy | Syk Kinase | Protein-Tyrosine Kinases - immunology | Protein-Tyrosine Kinases - antagonists & inhibitors | Tyrosine | Health aspects | Index Medicus | tyrosine-phosphorylation
Journal Article
Circulation research, ISSN 0009-7330, 01/2009, Volume 104, Issue 2, pp. 210 - 218
Reactive oxygen species | Minimally oxidized LDL | RANTES | Atherosclerosis | NADPH oxidase 2 | Cardiac & Cardiovascular Systems | Peripheral Vascular Disease | Life Sciences & Biomedicine | Hematology | Cardiovascular System & Cardiology | Science & Technology | Fundamental and applied biological sciences. Psychology | Cardiology. Vascular system | Atherosclerosis (general aspects, experimental research) | Biological and medical sciences | Medical sciences | Vertebrates: cardiovascular system | Blood and lymphatic vessels | Phosphorylation | Reactive Oxygen Species - metabolism | Membrane Glycoproteins - metabolism | Muscle, Smooth, Vascular - metabolism | Protein-Tyrosine Kinases - metabolism | NADPH Oxidases - metabolism | Intracellular Signaling Peptides and Proteins - metabolism | Gene Knockdown Techniques | NADPH Oxidases - deficiency | Atherosclerosis - enzymology | Time Factors | Toll-Like Receptor 4 - deficiency | Interleukin-1beta - metabolism | Protein Kinase C - metabolism | Inflammation Mediators - metabolism | NADPH Oxidases - genetics | Chemokine CCL5 - metabolism | Lipoproteins, LDL - metabolism | Interleukin-6 - metabolism | Myocytes, Smooth Muscle - metabolism | Syk Kinase | Cell Line | Phospholipase C gamma - metabolism | Atherosclerosis - immunology | Signal Transduction | Macrophages, Peritoneal - enzymology | Myeloid Differentiation Factor 88 - genetics | Macrophages, Peritoneal - immunology | Toll-Like Receptor 4 - genetics | NADPH Oxidase 2 | Toll-Like Receptor 4 - metabolism | Membrane Glycoproteins - genetics | Mice, Knockout | Animals | Mice | Enzyme Activation | Myeloid Differentiation Factor 88 - metabolism | Membrane Glycoproteins - deficiency | Cell Movement | Index Medicus
Journal Article
British journal of dermatology (1951), ISSN 0007-0963, 10/2019, Volume 181, Issue 4, pp. 733 - 742
Life Sciences & Biomedicine | Dermatology | Science & Technology | Janus Kinase Inhibitors - pharmacokinetics | Humans | Middle Aged | E-Selectin - blood | Male | Janus Kinases - metabolism | Syk Kinase - antagonists & inhibitors | Acetonitriles - pharmacokinetics | Dermatitis, Atopic - diagnosis | Dose-Response Relationship, Drug | Young Adult | Signal Transduction - immunology | Acetonitriles - administration & dosage | Placebos - adverse effects | Dermatitis, Atopic - immunology | Pyridazines - administration & dosage | Adult | Female | Piperidines - pharmacokinetics | Placebos - administration & dosage | Pyridazines - adverse effects | Severity of Illness Index | Piperidines - administration & dosage | Double-Blind Method | Treatment Outcome | Biomarkers - blood | Acetonitriles - adverse effects | Down-Regulation - drug effects | Janus Kinases - antagonists & inhibitors | Janus Kinase Inhibitors - adverse effects | Syk Kinase - metabolism | Dermatitis, Atopic - drug therapy | Janus Kinase Inhibitors - administration & dosage | Signal Transduction - drug effects | Down-Regulation - immunology | Piperidines - adverse effects | Pyridazines - pharmacokinetics | Dermatitis, Atopic - blood | Tyrosine | Spleen | Helper cells | Lymphocytes T | Pruritus | Dermatitis | Atopic dermatitis | Arteriosclerosis | Eczema | Biomarkers | Janus kinase | Pharmacokinetics | Protein-tyrosine kinase | Index Medicus | Clinical Trial | Original
Journal Article
Leukemia research, ISSN 0145-2126, 2014, Volume 39, Issue 3, pp. 329 - 334
Hematology, Oncology and Palliative Medicine | Flow cytometry | Dasatinib | Chronic Myeloid Leukemia (CML) | Spleen tyrosine kinase (Syk) | pSyk348 | PSyk | Oncology | Life Sciences & Biomedicine | Hematology | Science & Technology | Phosphorylation | Prognosis | Follow-Up Studies | Protein-Tyrosine Kinases - metabolism | Humans | Middle Aged | Leukemia, Myelogenous, Chronic, BCR-ABL Positive - drug therapy | Male | Intracellular Signaling Peptides and Proteins - metabolism | Biomarkers, Tumor | Young Adult | Protein-Tyrosine Kinases - genetics | Flow Cytometry | Leukemia, Myelogenous, Chronic, BCR-ABL Positive - pathology | Aged, 80 and over | Adult | Female | Tumor Cells, Cultured | Blast Crisis | Child | Intracellular Signaling Peptides and Proteins - genetics | Leukemia, Myelogenous, Chronic, BCR-ABL Positive - mortality | Real-Time Polymerase Chain Reaction | Syk Kinase | Oxazines - pharmacology | RNA, Messenger - genetics | Antineoplastic Combined Chemotherapy Protocols | Survival Rate | Pyrimidines - pharmacology | Reverse Transcriptase Polymerase Chain Reaction | Disease Progression | Adolescent | Leukemia, Myelogenous, Chronic, BCR-ABL Positive - metabolism | Aged | Protein Kinase Inhibitors - pharmacology | Pyridines - pharmacology | Thiazoles - pharmacology | Chronic Disease | Tyrosine | RNA | Index Medicus
Journal Article
Cancer research (Chicago, Ill.), ISSN 0008-5472, 04/2019, Volume 79, Issue 8, pp. 1831 - 1843
Journal Article
ChemMedChem, ISSN 1860-7179, 01/2016, Volume 11, Issue 2, pp. 217 - 233
imidazotriazines | drug discovery | spleen tyrosine kinase | free-energy perturbation | molecular modeling | Protein Kinase Inhibitors - chemical synthesis | Triazines - pharmacology | Protein-Tyrosine Kinases - metabolism | Humans | Intracellular Signaling Peptides and Proteins - antagonists & inhibitors | Imidazoles - chemistry | Models, Molecular | Imidazoles - pharmacology | Intracellular Signaling Peptides and Proteins - metabolism | Structure-Activity Relationship | Dose-Response Relationship, Drug | Thermodynamics | Protein Kinase Inhibitors - chemistry | Triazines - chemical synthesis | Triazines - chemistry | Molecular Structure | Protein Kinase Inhibitors - pharmacology | Imidazoles - chemical synthesis | Syk Kinase | Protein-Tyrosine Kinases - antagonists & inhibitors | Autoimmunity | Tyrosine | Phenols | Analysis | Spleen | Index Medicus
Journal Article
Journal of allergy and clinical immunology, ISSN 0091-6749, 03/2019, Volume 143, Issue 3, pp. 1100 - 1107.e11
Human | Fc receptors | allergy | basophil | Allergy | Immunology | Life Sciences & Biomedicine | Science & Technology | Autoantibodies - immunology | Immunoglobulin E - immunology | Humans | Basophils - immunology | Cells, Cultured | Receptors, IgE - immunology | Urticaria - immunology | Chronic Disease | Syk Kinase - immunology | Tyrosine | Spleen | CD34 antigen | Immunoglobulins | Autoantibodies | Urticaria | Secretion | Variability | Antibodies | Immunoglobulin E | Kinases | Patients | Asthma | Hemopoiesis | Histamine | Hypotheses | Algorithms | Peripheral blood | Syk protein | Mast cells | Leukocytes (basophilic) | Protein-tyrosine kinase | Index Medicus | Abridged Index Medicus
Journal Article
The Journal of biological chemistry, ISSN 0021-9258, 05/2019, Volume 294, Issue 19, pp. 7658 - 7668
Life Sciences & Biomedicine | Biochemistry & Molecular Biology | Science & Technology | Phosphorylation | Syk Kinase - metabolism | Models, Chemical | Humans | src-Family Kinases - metabolism | Enzyme Activation | src-Family Kinases - chemistry | Amino Acid Motifs | Syk Kinase - chemistry | src Homology Domains | Index Medicus | ITAM (immune-receptor tyrosine activation motif) | enzyme activation | autophosphorylation | non-receptor tyrosine kinase (nRTK) | cell signaling | spleen tyrosine kinase (SYK) | immunity | Enzymology | conformational change | phosphorylation | enzyme kinetics | tonic signalling
Journal Article