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benzosultams (40) 40
chemistry, organic (34) 34
cyclization (19) 19
derivatives (12) 12
inhibitors (12) 12
1,1-dioxides (9) 9
benzosultam (9) 9
sulfonamides (9) 9
chemistry, multidisciplinary (8) 8
sultam auxiliaries (8) 8
aza-ortho-xylylenes (6) 6
stereoselective-synthesis (6) 6
synthesis (6) 6
catalysis (5) 5
catalyst (5) 5
electrophilic asymmetric fluorination (5) 5
chiral benzosultams (4) 4
diels-alder reactions (4) 4
regioselectivity (4) 4
sultams (4) 4
tmscl/nai/mecn (4) 4
1,1-dioxide (3) 3
agent (3) 3
alkenes (3) 3
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chiral toluene-2,alpha-sultam auxiliaries (3) 3
chirality (3) 3
chlorides (3) 3
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efficient (3) 3
enantiomerically pure (3) 3
generation (3) 3
ketones (3) 3
metalation (3) 3
1,2-benzisothiazole 1,1-dioxides (2) 2
1,3-dipolar cycloaddition (2) 2
2-arylethanesulfonamide (2) 2
3,4,5-trisubstituted oxazolones (2) 2
6-membered benzosultams (2) 2
[1,5] sigmatropic hydrogen shift (2) 2
alkynyl bromides (2) 2
amidations (2) 2
analysis (2) 2
anticancer (2) 2
aromatic compounds (2) 2
aryl (2) 2
arylation (2) 2
asymmetric addition (2) 2
aziridination (2) 2
benzolactam (2) 2
calpain-i inhibitors (2) 2
chemical synthesis (2) 2
chemistry, applied (2) 2
construction (2) 2
cyclic sulfonamides (2) 2
cyclizations (2) 2
dft study (2) 2
efficient agent (2) 2
enantioselective electrophilic fluorinating agent (2) 2
entry (2) 2
extrusion (2) 2
flash vacuum thermolysis (2) 2
functionalized ynamides (2) 2
hydroamination (2) 2
hydrocarbonation (2) 2
hydrogen (2) 2
hydrogenation (2) 2
index medicus (2) 2
indole (2) 2
iodine (2) 2
iodotrimethylsilane (2) 2
mcpba (2) 2
nai-mecn reagent (2) 2
natural-products (2) 2
nucleophiles (2) 2
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organic chemistry (2) 2
palladium (2) 2
photoelectron spectroscopy (2) 2
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saccharin (2) 2
six-membered (2) 2
sonogashira coupling (2) 2
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sulfonamides - chemical synthesis (2) 2
thermal extrusion (2) 2
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ynamides (2) 2
1-phenylbenzazetidine (1) 1
11-beta-hydroxysteroid dehydrogenase (1) 1
2,1-benzisothiazoline 2,2-dioxide (1) 1
2,2-dioxides (1) 1
2-arylperimidine (1) 1
3-monoarylated (1) 1
3-monosubstituted (1) 1
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Synthesis, ISSN 0039-7881, 03/2016, Volume 48, Issue 5, pp. 710 - 722
Abstract An efficient method for the synthesis of benzo-δ-sultams [(4 Z )-4-benzylidene-2-(arylmethyl)-3,4-dihydro-2 H -1,2-benzothiazine 1,1-dioxides] via... 
paper | regioselectivity | benzosultams | hydrocarbonation | DFT study
Journal Article
Tetrahedron, ISSN 0040-4020, 05/2017, Volume 73, Issue 19, pp. 2766 - 2773
Palladium-catalyzed highly regioselective synthesis of benzotriazole appended benzosultams by the tandem-cyclization of functionalized ynamides with... 
[Pd]-catalysis | Cyclization | Benzosultams | Benzotriazoles | Ynamides | ALKENES | BIOLOGICAL-ACTIVITY | CHEMISTRY, ORGANIC | SYSTEMS | DERIVATIVES | Palladium | Catalysis
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 2017, Volume 15, Issue 14, pp. 2923 - 2930
An attractive and novel methodology involving Pd/Cu-catalyzed tandem head-to-tail dimerization/ cycloisomerization of terminal ynamides for the synthesis of... 
FUNCTIONALIZED YNAMIDES | AMIDATIONS | ALKYNYL BROMIDES | ENTRY | CHLORIDES | CHEMISTRY, ORGANIC | 3,4,5-TRISUBSTITUTED OXAZOLONES | BENZOSULTAMS | ARYL | EFFICIENT | CYCLIZATION
Journal Article
Organic Letters, ISSN 1523-7060, 04/2017, Volume 19, Issue 8, pp. 2042 - 2045
A highly diastereo- and enantioselective Ru­(II)-catalyzed dynamic kinetic resolution–asymmetric transfer hydrogenation (DKR–ATH) of α-(N-sulfonylimino) and... 
ENANTIOSELECTIVE SYNTHESIS | CONJUGATE LIGANDS | ANSA-RUTHENIUM(II) COMPLEXES | CHEMISTRY, ORGANIC | SULTAM AUXILIARIES | ARYL KETONES | STEREOSELECTIVE-SYNTHESIS | 1,1-DIOXIDES | CATALYST | INHIBITOR | CHIRAL BENZOSULTAMS
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 2018, Volume 16, Issue 28, pp. 5163 - 5166
An intramolecular annulation strategy has been developed for the synthesis of tetrahydrobenzo[e]pyrano[4,3-c][1,2]thiazine derivatives by means of coupling of... 
CALPAIN-I INHIBITORS | RADICAL CYCLIZATION | CONSTRUCTION | PIROXICAM | CHEMISTRY, ORGANIC | BENZOSULTAMS | MELOXICAM | ALDEHYDES | STEREOSELECTIVE-SYNTHESIS | SCAFFOLDS | DERIVATIVES | Organic chemistry | Silver | Toluene | Chemical reactions | Catalysis | Derivatives | Aldehydes | Chemical synthesis
Journal Article
CHEMICAL COMMUNICATIONS, ISSN 1359-7345, 2014, Volume 50, Issue 45, pp. 6046 - 6048
Intramolecular homolytic substitution (S(H)i) on the sulfur atom at acyclic N-(o-bromobenzyl)sulfinamides takes place with a complete inversion of the... 
SULTAM AUXILIARIES | BENZOSULTAMS | ASYMMETRIC-SYNTHESIS | SULFINAMIDES | INTRAMOLECULAR HOMOLYTIC SUBSTITUTION | CHEMISTRY, MULTIDISCIPLINARY
Journal Article
Organic and Biomolecular Chemistry, ISSN 1477-0520, 2018, Volume 16, Issue 16, pp. 2923 - 2931
An unprecedented Lewis acidic gold(I)-complex generated from chiral and achiral phosphines has been developed for the Mannich reaction of alpha-diazocarbonyl... 
KETONES | CYCLIZATIONS | METAL CARBENE | ISOQUINOLINE | CYCLOPROPANATION | CHEMISTRY, ORGANIC | BENZOSULTAMS | 1,1-DIOXIDE | SILYL ETHERS | DIAZOOXINDOLES | ENANTIOSELECTIVE CONSTRUCTION | Gold | Nuclear magnetic resonance--NMR | Imines | Quaternary | Phosphines
Journal Article
Advanced Synthesis & Catalysis, ISSN 1615-4150, 05/2016, Volume 358, Issue 10, pp. 1625 - 1638
Journal Article
Chemical Communications, ISSN 1359-7345, 05/2011, Volume 47, Issue 17, pp. 5052 - 5054
Journal Article
by Dong, YH and Ni, QW and Ma, ST and Liu, ZP
HETEROCYCLES, ISSN 0385-5414, 03/2010, Volume 81, Issue 3, pp. 637 - 648
3-Monoarylated five-membered benzosultams with various functional groups were prepared by simple and convenient two-step procedures. N-t-Bu-benzenesulfonamides... 
6-MEMBERED BENZOSULTAMS | CONVERSION | NAI-MECN REAGENT | CHEMISTRY, ORGANIC | SULFONAMIDES | 1,1-DIOXIDE | ELECTROPHILIC ASYMMETRIC FLUORINATION | Iodotrimethylsilane | Benzosultam | ENANTIOMERICALLY PURE | Cyclization | SULTAM AUXILIARIES | INHIBITORS | EFFICIENT AGENT | NaI/TMSCl/MeCN | Iodine
Journal Article
Heterocycles, ISSN 0385-5414, 06/2009, Volume 78, Issue 6, pp. 1387 - 1412
Recent developments in the novel synthesis of saccharin related five- and six-membered benzosultams are reviewed. 
Saccharin Derivative | Cyclization | Benzosultam | Intramolecular C-H Amination | Intramolecular Aziridination | HYDROGENATION | AZIRIDINATION | CONSTRUCTION | AMIDATION | CHEMISTRY, ORGANIC | SULFONAMIDES | ACCESS
Journal Article
Organic Letters, ISSN 1523-7060, 10/2003, Volume 5, Issue 22, pp. 4175 - 4177
A practical synthesis of sultams was developed via intramolecular sulfonamide dianion alkylation. This method has been applied toward the synthesis of chiral... 
AGENT | AUXILIARIES | METALATION | DIELS-ALDER REACTIONS | CAMPHOR | CHEMISTRY, ORGANIC | BENZOSULTAMS | ELECTROPHILIC ASYMMETRIC FLUORINATION | 1,1-DIOXIDES | INHIBITORS
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 06/2018, Volume 59, Issue 23, pp. 2260 - 2263
[Display omitted] •A methodology for the preparation of medicinally important Benzosultams.•Molecules are completely new and applied Sonogashira coupling for... 
Sonogashira coupling | C[sbnd]H arylation | Hydroamination | Indole | Benzosultams
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 09/2009, Volume 50, Issue 38, pp. 5354 - 5357
Journal Article
Tetrahedron, ISSN 0040-4020, 05/2020, Volume 76, Issue 21, p. 131201
An efficient Ni(ClO4)2·6H2O/SMI-PHOX catalyzed enantioselective addition of arylboronic acids to cyclic N-sulfonyl aldimines is envisioned to afford excellent... 
Cyclic N-Sulfonyl aldimines | Chiral benzosultams | Asymmetric addition | Spiro phosphine-oxazoline ligands | HYDRAZONES | ARYLATION | COMPLEXES | CHEMISTRY, ORGANIC | BORONIC ACIDS | LIGANDS | CHLORIDES | COUPLINGS | ASYMMETRIC HYDROGENATION | CARBOXYLIC-ACIDS | AMIDES
Journal Article
Heterocycles, ISSN 0385-5414, 11/2007, Volume 71, Issue 11, pp. 2377 - 2388
3-Monosubstituted six-membered benzosultams with a wide range of functional groups were prepared by simple and convenient two-step procedures. o-Lithiation of... 
Metalation | TMSCI/Nal/MeCN | Sulfonamide | Cyclization | Benzosultam | AGENT | CHEMISTRY, ORGANIC | SULFONAMIDES | ELECTROPHILIC ASYMMETRIC FLUORINATION | 1,1-DIOXIDES | DERIVATIVES
Journal Article
Tetrahedron Letters, ISSN 0040-4039, 06/2018, Volume 59, Issue 23, pp. 2260 - 2263
A one-pot Sonogashira coupling, hydroamination of alkyne and C–H arylation reactions for the synthesis of indole-fused benzosultams are described. This method... 
Sonogashira coupling | Hydroamination | Benzosultams | C–H arylation | Indole | ALKENES | REGIOSELECTIVE SYNTHESIS | CHEMISTRY, ORGANIC | SULTAMS | INHIBITORS | C-H arylation | AMINE | CYCLIZATION
Journal Article
Synthesis (Germany), ISSN 0039-7881, 10/2016, Volume 48, Issue 20, pp. 3544 - 3550
An efficient method for the synthesis of bioactive heterocycles containing 1,2-benzothiazine 1,1-dioxide derivatives via Pd-catalyzed intramolecular Heck... 
regioselectivity | XRD | Heck cyclization | sultams | CHEMISTRY, ORGANIC | BENZOSULTAMS | SULFUR | INHIBITORS | CATALYZED TANDEM CYCLIZATION
Journal Article
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